List of works - Kathleen A Farley

A new and useful method for the macrocyclization of linear peptides

scientific article published on 21 May 2012

An asymmetric synthesis of (2S,5S)-5-substituted azepane-2-carboxylate derivatives.

scientific article published on 28 January 2011

Comparative pharmacokinetic profile of cyclosporine (CsA) with a decapeptide and a linear analogue

scientific article published on 07 March 2017

Cyclic Peptide Design Guided by Residual Dipolar Couplings, J-Couplings, and Intramolecular Hydrogen Bond Analysis

scientific article published on 15 January 2019

Delineating the role of cooperativity in the design of potent PROTACs for BTK.

scientific article published on 16 July 2018

Design and evaluation of a 2-(2,3,6-trifluorophenyl)acetamide derivative as an agonist of the GPR119 receptor ⬇️

scientific article published on January 25, 2011

Discovery of azetidinyl ketolides for the treatment of susceptible and multidrug resistant community-acquired respiratory tract infections.

scientific article published in December 2009

Discovery of cytotoxic dolastatin 10 analogues with N-terminal modifications

scientific article

Efficient use of the iron ortho-nitrophenylporphyrin chloride to mimic biological oxidations of dimethylaminoantipyrine

scientific article published in October 2007

Integrating Intramolecular Hydrogen Bonding (IMHB) Considerations in Drug Discovery Using ΔlogP As a Tool

scientific article published on 12 June 2013

Macrocyclizations for medicinal chemistry: synthesis of druglike macrocycles by high-concentration Ullmann coupling.

scientific article

Optimizing PK properties of cyclic peptides: the effect of side chain substitutions on permeability and clearance().

scientific article published on October 2012

Revisiting N-to-O acyl shift for synthesis of natural product-like cyclic depsipeptides

scientific article published on 20 November 2014

Screening of compound libraries for protein binding using flow-injection nuclear magnetic resonance spectroscopy.

scientific article

Structural analysis of bovine somatotropin using monoclonal antibodies and the conformation-sensitive immunoassay

scientific article published on 01 June 1996

Utilizing on- and off-line monitoring tools to follow a kinetic resolution step during flow synthesis

scientific article published on 11 August 2016

List of works by Kathleen A Farley

A new and useful method for the macrocyclization of linear peptides

An asymmetric synthesis of (2S,5S)-5-substituted azepane-2-carboxylate derivatives.

Comparative pharmacokinetic profile of cyclosporine (CsA) with a decapeptide and a linear analogue

Cyclic Peptide Design Guided by Residual Dipolar Couplings, J-Couplings, and Intramolecular Hydrogen Bond Analysis

Delineating the role of cooperativity in the design of potent PROTACs for BTK.

Design and evaluation of a 2-(2,3,6-trifluorophenyl)acetamide derivative as an agonist of the GPR119 receptor ⬇️

Discovery of azetidinyl ketolides for the treatment of susceptible and multidrug resistant community-acquired respiratory tract infections.

Discovery of cytotoxic dolastatin 10 analogues with N-terminal modifications

Efficient use of the iron ortho-nitrophenylporphyrin chloride to mimic biological oxidations of dimethylaminoantipyrine

Integrating Intramolecular Hydrogen Bonding (IMHB) Considerations in Drug Discovery Using ΔlogP As a Tool

Macrocyclizations for medicinal chemistry: synthesis of druglike macrocycles by high-concentration Ullmann coupling.

Optimizing PK properties of cyclic peptides: the effect of side chain substitutions on permeability and clearance().

Revisiting N-to-O acyl shift for synthesis of natural product-like cyclic depsipeptides

Screening of compound libraries for protein binding using flow-injection nuclear magnetic resonance spectroscopy.

Structural analysis of bovine somatotropin using monoclonal antibodies and the conformation-sensitive immunoassay

Utilizing on- and off-line monitoring tools to follow a kinetic resolution step during flow synthesis