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List of works by Pasquale Linciano

Aryl thiosemicarbazones for the treatment of trypanosomatidic infections

scientific article published on 30 January 2018

Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth

scientific article published on 26 September 2019

Discovery of RC-752, a Novel Sigma-1 Receptor Antagonist with Antinociceptive Activity: A Promising Tool for Fighting Neuropathic Pain

scientific article published in 2023

Druggability profile of stilbene-derived PPAR agonists: determination of physicochemical properties and PAMPA study

scientific article published on 15 August 2019

Excited-state intramolecular proton transfer in a bioactive flavonoid provides fluorescence observables for recognizing its engagement with target proteins

scientific article published on 22 March 2019

Fibrate-derived N-(methylsulfonyl)amides with antagonistic properties on PPARα

scientific article published on 23 October 2012

High-resolution crystal structure of Trypanosoma brucei pteridine reductase 1 in complex with an innovative tricyclic-based inhibitor

scientific article published on 29 May 2020

Identification of a Potent and Selective 5-HT<sub>1A</sub> Receptor Agonist with <i>In Vitro</i> and <i>In Vivo</i> Antinociceptive Activity

scientific article published on 02 December 2020

Isolation of a High-Affinity Cannabinoid for the Human CB1 Receptor from a Medicinal Cannabis sativa Variety: Δ9-Tetrahydrocannabutol, the Butyl Homologue of Δ9-Tetrahydrocannabinol

scientific article published on 31 December 2019

Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds.

scientific article

Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance.

scientific article published on 22 January 2018

Structural development studies of PPARs ligands based on tyrosine scaffold

scientific article published on 31 October 2014

Synthesis and structure-activity relationships of fibrate-based analogues inside PPARs

scientific article published on 06 October 2012

Tackling Antimicrobial Resistance with Small Molecules Targeting LsrK: Challenges and Opportunities

scientific article published on 05 November 2020

Ten Years with New Delhi Metallo-β-lactamase-1 (NDM-1): From Structural Insights to Inhibitor Design

scientific article published on 28 November 2018

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