List of works by Dimitrios Evangelopoulos

A new plant-derived antibacterial is an inhibitor of efflux pumps in Staphylococcus aureus

scientific article published on 16 September 2013

A new strategy for hit generation: Novel in cellulo active inhibitors of CYP121A1 from Mycobacterium tuberculosis via a combined X-ray crystallographic and phenotypic screening approach (XP screen)

scientific article published on 11 January 2022

An antibacterial from Hypericum acmosepalum inhibits ATP-dependent MurE ligase from Mycobacterium tuberculosis

scientific article published on 10 November 2011

Antagonistic effects of indoloquinazoline alkaloids on antimycobacterial activity of evocarpine

scientific article published on 04 February 2015

Anti-tubercular screening of natural products from Colombian plants: 3-methoxynordomesticine, an inhibitor of MurE ligase of Mycobacterium tuberculosis.

scientific article published on 18 August 2010

Antimycobacterials from lovage root (Ligusticum officinale Koch)

scientific article published on 16 August 2012

Antitubercular activity of Arctium lappa and Tussilago farfara extracts and constituents.

scientific article published on 20 June 2014

Antitubercular specific activity of ibuprofen and the other 2-arylpropanoic acids using the HT-SPOTi whole-cell phenotypic assay

scientific article

Assessment of treatment response by colony forming units, time to culture positivity and the molecular bacterial load assay compared in a mouse tuberculosis model

scientific article published on 8 May 2017

Characterisation of ATP-dependent Mur ligases involved in the biogenesis of cell wall peptidoglycan in Mycobacterium tuberculosis

scientific article

Characterisation of a putative AraC transcriptional regulator from Mycobacterium smegmatis

scientific article published on December 2014

Characterization of an oxidoreductase from the arylamine N-acetyltransferase operon in Mycobacterium smegmatis

scientific article

Comparative fitness analysis of D-cycloserine resistant mutants reveals both fitness-neutral and high-fitness cost genotypes

scientific article published on 13 September 2019

DNA sequence-selective C8-linked pyrrolobenzodiazepine-heterocyclic polyamide conjugates show anti-tubercular-specific activities.

scientific article

Design and Synthesis of 1-((1,5-Bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethylocta-2,6-dienyl)ethane-1,2-diamine (SQ109) Pyrrole Hybrid Derivatives: Discovery of Potent Antitu

scientific article published on 23 February 2016

Effective anti-tuberculosis therapy correlates with plasma small RNA.

scientific article published on 5 March 2015

Gene analysis of the N-terminal region of the estrogen receptor alpha in preeclampsia

scientific article published on 01 September 2001

Improving the tuberculosis drug development pipeline

scientific article published on 16 March 2015

Interaction of N-methyl-2-alkenyl-4-quinolones with ATP-dependent MurE ligase of Mycobacterium tuberculosis: antibacterial activity, molecular docking and inhibition kinetics

scientific article

Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach

scientific article

Molecular analysis of the estrogen receptor alpha gene in men with coronary artery disease: association with disease status ⬇️

scientific article published on May 1, 2003

Optimising molecular diagnostic capacity for effective control of tuberculosis in high-burden settings

scientific article published on August 2016

Pediatric tuberculosis-human immunodeficiency virus co-infection in the United Kingdom highlights the need for better therapy monitoring tools: a case report

scientific article published on 26 February 2017

Polymersomes Eradicating Intracellular Bacteria

scientific article published on 09 June 2020

Posterior stabilization of cervical spine injuries using the Roy-Camille plates: a long-term follow-up

scientific article published on 10 December 2013

ProTides of N-(3-(5-(2'-deoxyuridine))prop-2-ynyl)octanamide as potential anti-tubercular and anti-viral agents.

scientific article published on 15 March 2014

Profiling persistent tubercule bacilli from patient sputa during therapy predicts early drug efficacy

scientific article

Rapid methods for testing inhibitors of mycobacterial growth

scientific article published on 01 January 2010

Synthesis and biological evaluation of purpurealidin E-derived marine sponge metabolites: aplysamine-2, aplyzanzine A, and suberedamines A and B.

scientific article published on 23 May 2012

Tetrahydroisoquinolines affect the whole-cell phenotype of Mycobacterium tuberculosis by inhibiting the ATP-dependent MurE ligase.

scientific article published on 4 February 2015

Understanding anti-tuberculosis drug efficacy: rethinking bacterial populations and how we model them

scientific article

Versatile routes to marine sponge metabolites through benzylidene rhodanines.

scientific article published on 12 December 2012

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