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List of works by Raphael Terreux

6-halogenochromones bearing tryptamine: one-step access to potent and highly selective inhibitors of breast cancer resistance protein

scientific article published on 21 May 2012

A cyclic PNA-based compound targeting domain IV of HCV IRES RNA inhibits in vitro IRES-dependent translation

scientific article published in October 2005

Active site coupling in Plasmodium falciparum GMP synthetase is triggered by domain rotation

scientific article

Bacterial tyrosine-kinases: structure-function analysis and therapeutic potential

scientific article published on 27 August 2009

Bioinspired Design and Oriented Synthesis of Immunogenic Site-Specifically Penicilloylated Peptides.

scientific article

C(16)-methyl corticosteroids are far less allergenic than the non-methylated molecules

scientific article published on 19 April 2011

Calcineurin A versus NS5A-TP2/HD domain containing 2: a case study of site-directed low-frequency random mutagenesis for dissecting target specificity of peptide aptamers

scientific article

Collateral sensitivity of resistant MRP1-overexpressing cells to flavonoids and derivatives through GSH efflux

scientific article

Construction of atomic models of full hepatitis B vaccine particles at different stages of maturation

scientific article published on 09 April 2020

Cyclic PNA-based compound directed against HIV-1 TAR RNA: modelling, liquid-phase synthesis and TAR binding

scientific article published on 27 November 2003

Daclatasvir-like inhibitors of NS5A block early biogenesis of hepatitis C virus-induced membranous replication factories, independent of RNA replication

scientific article

Deciphering the molecular mechanisms underlying the binding of the TWIST1/E12 complex to regulatory E-box sequences

scientific article published on 05 May 2016

Degradation of High Energy Materials Using Biological Reduction: A Rational Way to Reach Bioremediation

scientific article published on 07 November 2019

Delayed hypersensitivity to corticosteroids in a series of 315 patients: clinical data and patch test results

scientific article

Destabilization of the TWIST1/E12 complex dimerization following the R154P point-mutation of TWIST1: an in silico approach.

scientific article

Determination of ddATP levels in human immunodeficiency virus-infected patients treated with dideoxyinosine

scientific article published on February 2004

Flavonoids and tyrosine nitration: structure-activity relationship correlation with enthalpy of formation

scientific article published in March 2005

Identification of structural and molecular determinants of the tyrosine-kinase Wzc and implications in capsular polysaccharide export

scientific article

In Silico, in Vitro, and in Vivo Evaluation of New Candidates for α-Synuclein PET Imaging

scientific article published on 25 July 2018

Interhelical loops within the bHLH domain are determinant in maintaining TWIST1-DNA complexes.

scientific article published on 25 March 2013

Investigation of chalcones as selective inhibitors of the breast cancer resistance protein: critical role of methoxylation in both inhibition potency and cytotoxicity

scientific article published on 02 April 2012

Isoflavonoids in non-leguminous families: an update.

scientific article

Localization of putative binding sites for cyclic guanosine monophosphate and the anti-cancer drug 5-fluoro-2'-deoxyuridine-5'-monophosphate on ABCC11 in silico models

scientific article

MBL-II-141, a chromone derivative, enhances irinotecan (CPT-11) anticancer efficiency in ABCG2-positive xenografts

scientific article

Modelling, synthesis and biological evaluation of an ethidium-arginine conjugate linked to a ribonuclease mimic directed against TAR RNA of HIV-1.

scientific article

Molecular Dynamics Studies of Poly(Lactic Acid) Nanoparticles and Their Interactions with Vitamin E and TLR Agonists Pam1CSK4 and Pam3CSK4

scientific article published on 05 November 2020

Molecular modelling of TLR agonist Pam3CSK4 entrapment in PLA nanoparticles as a tool to explain loading efficiency and functionality

scientific article published on 26 July 2019

Multidrug resistance ABC transporter structure predictions by homology modeling approaches

scientific article published on March 2011

New structure-activity relationships of chalcone inhibitors of breast cancer resistance protein: polyspecificity toward inhibition and critical substitutions against cytotoxicity

scientific article published on 30 September 2013

Potent and fully noncompetitive peptidomimetic inhibitor of multidrug resistance P-glycoprotein.

scientific article

Pyrolysis patterns of 5 close Corynebacterium species analyzed by artificial neural networks.

scientific article published in May 2004

Quantification and kinetic study in plasma and tissues of (E)-1,1,4,4-tetramethyl-2-tetrazene, a liquid propellant and a transformation product of 1,1-dimethyl hydrazine

scientific article published on 17 June 2015

Quinoxaline-substituted chalcones as new inhibitors of breast cancer resistance protein ABCG2: polyspecificity at B-ring position

scientific article

Relative antioxidant capacities of propofol and its main metabolites

scientific article published on 10 July 2004

Structure-activity relationship of natural and synthetic coumarins inhibiting the multidrug transporter P-glycoprotein.

scientific article published on 7 July 2006

Substituted chromones as highly potent nontoxic inhibitors, specific for the breast cancer resistance protein

scientific article published on 06 January 2012

Surface charge modulation of rifampicin-loaded PLA nanoparticles to improve antibiotic delivery in Staphylococcus aureus biofilms

scientific article published on 07 January 2021

Tyrosine dephosphorylation of the syndecan-1 PDZ binding domain regulates syntenin-1 recruitment

scientific article

Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2

scientific article published on 12 November 2020

X-ray structures of human bile-salt activated lipase conjugated to nerve agents surrogates

scientific article published on 22 October 2018

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