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List of works by Jessica Iegre

A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066.

scientific article published on 30 April 2017

Binding Mode and Induced Fit Predictions for Prospective Computational Drug Design.

scientific article published on 14 March 2016

Database Extraction of Metabolite Information of Drug Candidates: Analysis of 27 AstraZeneca Compounds with Human Absorption, Distribution, Metabolism, and Excretion Data

scientific article

Efficient development of stable and highly functionalised peptides targeting the CK2α/CK2β protein-protein interaction.

scientific article published on 12 April 2019

General dual functionalisation of biomacromolecules via a cysteine bridging strategy

scientific article published on 20 May 2020

Oxime-based inhibitors of glucose transporter 1 displaying antiproliferative effects in cancer cells.

scientific article published on 28 September 2013

Peptides as a platform for targeted therapeutics for cancer: peptide-drug conjugates (PDCs)

scientific article published on 21 December 2020

Salicylketoximes That Target Glucose Transporter 1 Restrict Energy Supply to Lung Cancer Cells

scientific article published on September 2015

Second-generation CK2α inhibitors targeting the αD pocket.

scientific article

Stapled peptides as a new technology to investigate protein-protein interactions in human platelets.

scientific article published on 25 April 2018

Targeted covalent inhibitors of MDM2 using electrophile-bearing stapled peptides

scientific article published on 21 June 2019

Two-Component Stapling of Biologically Active and Conformationally Constrained Peptides: Past, Present, and Future

scholarly article published 7 August 2018