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List of works by Mark Blaskovich

A new antibiotic with potent activity targets MscL.

scientific article published on 4 February 2015

Activity and Predicted Nephrotoxicity of Synthetic Antibiotics Based on Polymyxin B.

scientific article published on 6 January 2016

An amphipathic peptide with antibiotic activity against multidrug-resistant Gram-negative bacteria

scientific article published on 23 June 2020

An azido-oxazolidinone antibiotic for live bacterial cell imaging and generation of antibiotic variants

scientific article published on 14 June 2014

Anti-cooperative ligand binding and dimerisation in the glycopeptide antibiotic dalbavancin

scientific article published on April 2014

Antibacterial serrulatane diterpenes from the Australian native plant Eremophila microtheca.

scientific article published on 18 April 2013

Antibiotics in the clinical pipeline at the end of 2015.

scientific article

Antibiotics in the clinical pipeline in 2013.

scientific article published on 04 September 2013

Antimicrobial Silver in Medicinal and Consumer Applications: A Patent Review of the Past Decade (2007⁻2017)

article

Antitubercular and Antiparasitic 2-Nitroimidazopyrazinones with Improved Potency and Solubility

scientific article published on 05 November 2020

Can octapeptin antibiotics combat extensively drug-resistant (XDR) bacteria?

scientific article published on 26 June 2018

Cell- and biomarker-based assays for predicting nephrotoxicity

scientific article

Chemical philanthropy: a path forward for antibiotic discovery?

scientific article

Chemical synthesis of human trefoil factor 1 (TFF1) and its homodimer provides novel insights into their mechanisms of action

scientific article published on 11 May 2020

Clostridium difficile drug pipeline: challenges in discovery and development of new agents

scientific article published on 30 March 2015

Contribution of Amphipathicity and Hydrophobicity to the Antimicrobial Activity and Cytotoxicity of β-Hairpin Peptides

scientific article published on 29 April 2016

Correction: Chemical synthesis of human trefoil factor 1 (TFF1) and its homodimer provides novel insights into their mechanisms of action

scientific article published on 17 June 2020

Cover Feature: Nontoxic Cobalt(III) Schiff Base Complexes with Broad‐Spectrum Antifungal Activity (Chem. Eur. J. 6/2021)

scientific article published on 24 November 2020

CryoEM structure of the outer membrane secretin channel pIV from the f1 filamentous bacteriophage

CryoEM structure of the outer membrane secretin channel pIV from the f1 filamentous bacteriophage

scientific article published on 2 November 2021

Design and synthesis of phosphotyrosine mimetics.

scientific article published in June 2003

Design, synthesis and biological evaluation of 2-nitroimidazopyrazin-one/-es with antitubercular and antiparasitic activity

scientific article published on 11 December 2018

Detection and Investigation of Eagle Effect Resistance to Vancomycin in Clostridium difficile With an ATP-Bioluminescence Assay.

scientific article published on 2 July 2018

Developments in Glycopeptide Antibiotics

scientific article

Discovery of functionally selective C5aR2 ligands: novel modulators of C5a signalling.

scientific article

Drug discovery and protein tyrosine phosphatases.

scientific article

Effects of Microplate Type and Broth Additives on Microdilution MIC Susceptibility Assays

scientific article published on 21 December 2018

Elucidating the Lipid Binding Properties of Membrane-Active Peptides Using Cyclised Nanodiscs

scientific article published on 16 April 2019

Enhancement of antibiotic-activity through complexation with metal ions - Combined ITC, NMR, enzymatic and biological studies.

scientific article published on 24 November 2016

Evaluation of biomarkers for in vitro prediction of drug-induced nephrotoxicity: comparison of HK-2, immortalized human proximal tubule epithelial, and primary cultures of human proximal tubular cells

scientific article published on 15 May 2015

Fluorescent Antibiotics: New Research Tools to Fight Antibiotic Resistance.

scientific article published on 22 February 2018

Fluorescent Trimethoprim Conjugate Probes To Assess Drug Accumulation in Wild Type and Mutant Escherichia coli

scientific article published on 16 August 2016

Fluoroquinolone-derived fluorescent probes for studies of bacterial penetration and efflux

scientific article published on 17 May 2019

Glycopeptide antibiotics: back to the future.

scientific article published on 13 August 2014

Helping Chemists Discover New Antibiotics.

scientific article published on 13 May 2015

Highly efficient and versatile synthesis of libraries of constrained beta-strand mimetics

scientific article

How to Stimulate and Facilitate Early Stage Antibiotic Discovery

scientific article published on 01 June 2020

In vitro Antimicrobial Activity of Acne Drugs Against Skin-Associated Bacteria

scientific article published on 10 October 2019

Institutional profile: Community for Open Antimicrobial Drug Discovery - crowdsourcing new antibiotics and antifungals

scientific article published on 24 March 2017

Investigating the Interaction of Octapeptin A3 with Model Bacterial Membranes

scientific article

Light-Activated Rhenium Complexes with Dual Mode of Action against Bacteria

scientific article published on 30 January 2020

Lipoamino acids as major components of absorption promoters in drug delivery.

scientific article published on January 2012

Loss of YhcB results in dysregulation of coordinated peptidoglycan, LPS and phospholipid synthesis during Escherichia coli cell growth

scientific article published on 23 December 2021

Loss of β-Ketoacyl Acyl Carrier Protein Synthase III Activity Restores Multidrug-Resistant Escherichia coli Sensitivity to Previously Ineffective Antibiotics

scientific article published in 2022

Metal Complexes as Antifungals? From a Crowd-Sourced Compound Library to the First <i>In Vivo</i> Experiments

scientific article published in 2022

Metal complexes as a promising source for new antibiotics

scientific article published on 12 February 2020

Metronidazole-triazole conjugates: activity against Clostridium difficile and parasites

scientific article published on 18 June 2015

Mucin Binding Reduces Colistin Antimicrobial Activity.

scientific article

Multifactorial Chromosomal Variants Regulate Polymyxin Resistance In Extensively Drug-Resistant Klebsiella pneumoniae

Multifactorial chromosomal variants regulate polymyxin resistance in extensively drug-resistant Klebsiella pneumoniae

scientific article published on 12 February 2018

Natural products as anthelmintics: safeguarding animal health

scientific article published in January 2023

Nitroimidazole carboxamides as antiparasitic agents targeting Giardia lamblia, Entamoeba histolytica and Trichomonas vaginalis.

scientific article published on 27 April 2016

Nitroimidazoles: Molecular Fireworks That Combat a Broad Spectrum of Infectious Diseases.

scientific article

Non-antibiotic Small-Molecule Regulation of DHFR-Based Destabilizing Domains In Vivo

scientific article published on 15 August 2019

Non-toxic Cobalt(III) Schiff Base Complexes with Broad Spectrum Antifungal Activity

scientific article published on 30 July 2020

Nontoxic Cobalt(III) Schiff Base Complexes with Broad-Spectrum Antifungal Activity

scientific article published on 24 November 2020

Octapeptin C4 Induces Less Resistance and Novel Mutations in an Epidemic Carbapenemase-producing Klebsiella pneumoniae ST258 Clinical Isolate Compared to Polymyxins

article by Miranda Pitt et al published 28 April 2018 in bioRxiv

Octapeptin C4 and polymyxin resistance occur via distinct pathways in an epidemic XDR Klebsiella pneumoniae ST258 isolate

scientific article published on 01 March 2019

Old dogs and new tricks in antimicrobial discovery.

scientific article published on 2 June 2016

Polishing the tarnished silver bullet: the quest for new antibiotics

scientific article published on February 2017

Protein-inspired antibiotics active against vancomycin- and daptomycin-resistant bacteria.

scientific article published on 2 January 2018

Quinolone antibiotics

scientific article published on 28 June 2019

Repurposing a neurodegenerative disease drug to treat Gram-negative antibiotic-resistant bacterial sepsis

scientific article published on 01 November 2020

Resolving biofilm infections: current therapy and drug discovery strategies.

scientific article published on October 2012

Self-assembling lipopeptides with a potent activity against Gram-positive bacteria, including multidrug resistant strains.

scientific article published in November 2015

Short cationic lipopeptides as effective antibacterial agents: Design, physicochemical properties and biological evaluation.

scientific article published on 30 March 2016

Silver bullets: A new lustre on an old antimicrobial agent

scientific article published on 27 May 2018

Structure, Function, and Biosynthetic Origin of Octapeptin Antibiotics Active against Extensively Drug-Resistant Gram-Negative Bacteria.

scientific article published on 23 January 2018

Structure-Activity and -Toxicity Relationships of the Antimicrobial Peptide Tachyplesin-1.

scientific article published on 29 September 2017

Structure-Function Studies of Polymyxin B Lipononapeptides

scientific article published on 02 February 2019

Surface Ligand Density of Antibiotic-Nanoparticle Conjugates Enhances Target Avidity and Membrane Permeabilization of Vancomycin-Resistant Bacteria.

scientific article

Synthesis of octapeptin C4 and biological profiling against NDM-1 and polymyxin-resistant bacteria.

scientific article published on 12 April 2017

The Eagle Effect and Antibiotic-Induced Persistence: Two Sides of the Same Coin?

scientific article published on 15 November 2018

The Fight Against Antimicrobial Resistance Is Confounded by a Global Increase in Antibiotic Usage

scientific article published on 14 May 2018

Tyrosinase inhibitors as potential antibacterial agents

scientific article published on 18 November 2019

Unusual Amino Acids in Medicinal Chemistry

scientific article

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