List of works - William Tieu

89Zr-pro-MMP-9 F(ab')2 detects colitis induced intestinal and kidney fibrosis

scientific article published on 23 November 2020

Advanced Resistance Studies Identify Two Discrete Mechanisms in Staphylococcus aureus to Overcome Antibacterial Compounds that Target Biotin Protein Ligase

scientific article published on 06 April 2020

Analogues of desferrioxamine B (DFOB) with new properties and new functions generated using precursor-directed biosynthesis

scientific article published on 30 January 2019

Biotin analogues with antibacterial activity are potent inhibitors of biotin protein ligase

scientific article

Crystal structure of highly glycosylated human leukocyte elastase in complex with an S2' site binding inhibitor

scientific article published on 26 July 2018

Dimeric and trimeric homo- and heteroleptic hydroxamic acid macrocycles formed using mixed-ligand Fe(III)-based metal-templated synthesis

scientific article published in August 2017

Exploiting the biosynthetic machinery of Streptomyces pilosus to engineer a water-soluble zirconium(iv) chelator

scientific article

Exploring hydroxamic acid inhibitors of HDAC1 and HDAC2 using small molecule tools and molecular or homology modelling

scientific article published on 02 August 2019

Forward and reverse (retro) iron(III) or gallium(III) desferrioxamine E and ring-expanded analogues prepared using metal-templated synthesis from endo-hydroxamic acid monomers

scientific article

Heterocyclic acyl-phosphate bioisostere-based inhibitors of Staphylococcus aureus biotin protein ligase

scientific article published on 19 August 2014

Immuno-PET of innate immune markers CD11b and IL-1β detect inflammation in murine colitis

scientific article published on 09 November 2018

Improved Synthesis of Biotinol-5'-AMP: Implications for Antibacterial Discovery

scientific article

New Series of BPL Inhibitors To Probe the Ribose-Binding Pocket of Staphylococcus aureus Biotin Protein Ligase.

scientific article published on 10 October 2016

New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds.

scientific article

Octadentate Zirconium(IV)-Loaded Macrocycles with Varied Stoichiometry Assembled From Hydroxamic Acid Monomers using Metal-Templated Synthesis

scientific article published on 28 February 2017

Optimising in situ click chemistry: the screening and identification of biotin protein ligase inhibitors

article

Rapid and automated production of [68Ga]gallium chloride and [68Ga]Ga-DOTA-TATE on a medical cyclotron

scientific article published on 12 July 2019

Reverse Biosynthesis: Generating Combinatorial Pools of Drug Leads from Enzyme-Mediated Fragmentation of Natural Products

scientific article

Selective inhibition of Biotin Protein Ligase from Staphylococcus aureus

scientific article

Structure guided design of biotin protein ligase inhibitors for antibiotic discovery

scientific article published on January 2014

Sulfonamide-Based Inhibitors of Biotin Protein Ligase as New Antibiotic Leads

scientific article published on 21 August 2019

The chemical biology and coordination chemistry of putrebactin, avaroferrin, bisucaberin, and alcaligin

scientific article published on 26 June 2018

List of works by William Tieu

89Zr-pro-MMP-9 F(ab')2 detects colitis induced intestinal and kidney fibrosis

Advanced Resistance Studies Identify Two Discrete Mechanisms in Staphylococcus aureus to Overcome Antibacterial Compounds that Target Biotin Protein Ligase

Analogues of desferrioxamine B (DFOB) with new properties and new functions generated using precursor-directed biosynthesis

Biotin analogues with antibacterial activity are potent inhibitors of biotin protein ligase

Crystal structure of highly glycosylated human leukocyte elastase in complex with an S2' site binding inhibitor

Dimeric and trimeric homo- and heteroleptic hydroxamic acid macrocycles formed using mixed-ligand Fe(III)-based metal-templated synthesis

Exploiting the biosynthetic machinery of Streptomyces pilosus to engineer a water-soluble zirconium(iv) chelator

Exploring hydroxamic acid inhibitors of HDAC1 and HDAC2 using small molecule tools and molecular or homology modelling

Forward and reverse (retro) iron(III) or gallium(III) desferrioxamine E and ring-expanded analogues prepared using metal-templated synthesis from endo-hydroxamic acid monomers

Heterocyclic acyl-phosphate bioisostere-based inhibitors of Staphylococcus aureus biotin protein ligase

Immuno-PET of innate immune markers CD11b and IL-1β detect inflammation in murine colitis

Improved Synthesis of Biotinol-5'-AMP: Implications for Antibacterial Discovery

New Series of BPL Inhibitors To Probe the Ribose-Binding Pocket of Staphylococcus aureus Biotin Protein Ligase.

New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds.

Octadentate Zirconium(IV)-Loaded Macrocycles with Varied Stoichiometry Assembled From Hydroxamic Acid Monomers using Metal-Templated Synthesis

Optimising in situ click chemistry: the screening and identification of biotin protein ligase inhibitors

Rapid and automated production of [68Ga]gallium chloride and [68Ga]Ga-DOTA-TATE on a medical cyclotron

Reverse Biosynthesis: Generating Combinatorial Pools of Drug Leads from Enzyme-Mediated Fragmentation of Natural Products

Selective inhibition of Biotin Protein Ligase from Staphylococcus aureus

Structure guided design of biotin protein ligase inhibitors for antibiotic discovery

Sulfonamide-Based Inhibitors of Biotin Protein Ligase as New Antibiotic Leads

The chemical biology and coordination chemistry of putrebactin, avaroferrin, bisucaberin, and alcaligin