List of works - Craig Jamieson

A Multicomponent Route to Functionalized Amides and Oxazolidinones

scientific article published on 01 December 2017

A fragment-like approach to PYCR1 inhibition

scientific article published on 25 July 2019

Amidation of esters with amino alcohols using organobase catalysis

scientific article published on 16 September 2014

Amidation of unactivated ester derivatives mediated by trifluoroethanol

scientific article published on 01 April 2017

Atom Efficient Synthesis of Selectively Difluorinated Carbocycles through a Gold(I)-Catalyzed Cyclization

scientific article published on 30 July 2018

Catalytic amidation of unactivated ester derivatives mediated by trifluoroethanol

scientific article published on 01 June 2015

Cyrene as a bio-based solvent for HATU mediated amide coupling

scientific article published on 01 April 2018

Dioxo-triazines as a novel series of cathepsin K inhibitors

scientific article

Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD Integrins.

scientific article published on 30 January 2017

Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease

scientific article

Functional analysis of a novel positive allosteric modulator of AMPA receptors derived from a structure-based drug design strategy

scientific article

Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replacement within an LpPLA2 Inhibitor.

scientific article published on 15 November 2016

Metal-free C-C bond formation via coupling of nitrile imines and boronic acids

scientific article published on 27 September 2019

One-Pot, Three-Step Synthesis of Cyclopropylboronic Acid Pinacol Esters from Synthetically Tractable Propargylic Silyl Ethers.

scientific article published on 6 July 2017

Organobase-Catalyzed Amidation of Esters with Amino Alcohols

scientific article published on 02 May 2013

Photocatalytic E → Z Isomerization of β-Ionyl Derivatives

scientific article published on 20 November 2019

Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor.

scientific article published on October 2010

Practical synthesis of pharmaceutically relevant molecules enriched in sp3 character.

scientific article published on 30 November 2017

Rational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators

scientific article

Rational Design of a Novel AMPA Receptor Modulator through a Hybridization Approach

scientific article

Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulation

scientific article (publication date: 2016)

Structurally Diverse Mitochondrial Branched Chain Aminotransferase (BCATm) Leads with Varying Binding Modes Identified by Fragment Screening

scientific article

Structure based evolution of a novel series of positive modulators of the AMPA receptor

scientific article

Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode

scientific article

Surface Functionalization with Carboxylic Acids by Photochemical Microcontact Printing and Tetrazole Chemistry

scientific article published on 16 January 2018

Synthesis of the originally proposed structures of elatenyne and an enyne from Laurencia majuscula

scientific article published on 20 November 2008

The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits

scientific article

List of works by Craig Jamieson

A Multicomponent Route to Functionalized Amides and Oxazolidinones

A fragment-like approach to PYCR1 inhibition

Amidation of esters with amino alcohols using organobase catalysis

Amidation of unactivated ester derivatives mediated by trifluoroethanol

Atom Efficient Synthesis of Selectively Difluorinated Carbocycles through a Gold(I)-Catalyzed Cyclization

Catalytic amidation of unactivated ester derivatives mediated by trifluoroethanol

Cyrene as a bio-based solvent for HATU mediated amide coupling

Dioxo-triazines as a novel series of cathepsin K inhibitors

Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD Integrins.

Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease

Functional analysis of a novel positive allosteric modulator of AMPA receptors derived from a structure-based drug design strategy

Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replacement within an LpPLA2 Inhibitor.

Metal-free C-C bond formation via coupling of nitrile imines and boronic acids

One-Pot, Three-Step Synthesis of Cyclopropylboronic Acid Pinacol Esters from Synthetically Tractable Propargylic Silyl Ethers.

Organobase-Catalyzed Amidation of Esters with Amino Alcohols

Photocatalytic E → Z Isomerization of β-Ionyl Derivatives

Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor.

Practical synthesis of pharmaceutically relevant molecules enriched in sp3 character.

Rational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators

Rational Design of a Novel AMPA Receptor Modulator through a Hybridization Approach

Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulation

Structurally Diverse Mitochondrial Branched Chain Aminotransferase (BCATm) Leads with Varying Binding Modes Identified by Fragment Screening

Structure based evolution of a novel series of positive modulators of the AMPA receptor

Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode

Surface Functionalization with Carboxylic Acids by Photochemical Microcontact Printing and Tetrazole Chemistry

Synthesis of the originally proposed structures of elatenyne and an enyne from Laurencia majuscula

The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits