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List of works by David Wifling

Basal Histamine H4 Receptor Activation: Agonist Mimicry by the Diphenylalanine Motif

scientific article published on 16 October 2019

Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity

scientific article published on 22 May 2019

Dibenzodiazepinone-type muscarinic receptor antagonists conjugated to basic peptides: Impact of the linker moiety and unnatural amino acids on M2R selectivity

scientific article published in 2021

Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H2 Receptor Agonists

scientific article published on 09 March 2018

Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts

scientific article (publication date: 2013)

Mimicking of Arginine by Functionalized Nω-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples

scientific article published on 11 February 2016

Molecular determinants for the high constitutive activity of the human histamine H4 receptor: functional studies on orthologues and mutants

scientific article published on 5 September 2014

Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M2 Muscarinic Acetylcholine Receptor.

scientific article

Structural basis of ligand binding modes at the neuropeptide Y Y1 receptor

scientific article published on 18 April 2018

Structure-Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands

article

The extracellular loop 2 (ECL2) of the human histamine H4 receptor substantially contributes to ligand binding and constitutive activity

scientific article published on 28 January 2015

Universal Activation Index for Class A GPCRs

scientific article published on 06 September 2019