List of works - Shinichiro Fuse

6-Azido-6-deoxy-l-idose as a Hetero-Bifunctional Spacer for the Synthesis of Azido-Containing Chemical Probes.

scientific article

A Formal Total Synthesis of Taxol Aided by an Automated Synthesizer

article

A rapid and clean synthetic approach to cyclic peptides via micro-flow peptide chain elongation and photochemical cyclization: synthesis of a cyclic RGD peptide.

scientific article published on 16 November 2016

Anti-influenza virus compound from Streptomyces sp. RI18.

scientific article published on October 2010

Asymmetric Total Synthesis of ent-Pyripyropene A.

scientific article published on 26 May 2015

Complete characterization of the seventeen step moenomycin biosynthetic pathway

scientific article published on September 2009

Continuous in situ generation and reaction of phosgene in a microflow system

scientific article published on 31 October 2011

Continuous-flow synthesis of activated vitamin D3 and its analogues

scientific article published on 16 May 2012

Continuous-flow synthesis of vitamin D3.

scientific article published on 28 September 2010

Design, synthesis and evaluation of carbamate-modified (-)-N(1)-phenethylnorphysostigmine derivatives as selective butyrylcholinesterase inhibitors.

scientific article published on 20 January 2010

Design, synthesis, and evaluation of azo D-π-A dyes as photothermal agents

scientific article published on 01 December 2019

Design, synthesis, evaluation and QSAR analysis of N(1)-substituted norcymserine derivatives as selective butyrylcholinesterase inhibitors.

scientific article published on 20 January 2010

Development of 1-aryl-3-furanyl/thienyl-imidazopyridine templates for inhibitors against hypoxia inducible factor (HIF)-1 transcriptional activity.

scientific article published on 5 November 2016

Development of dual targeting inhibitors against aggregations of amyloid-β and tau protein.

scientific article published on 26 July 2014

Directing/protecting-group-free synthesis of tetraaryl-substituted pyrazoles through four direct arylations on an unsubstituted pyrazole scaffold

scientific article published on 21 August 2015

Efficient amide bond formation through a rapid and strong activation of carboxylic acids in a microflow reactor

scientific article published on 2 December 2013

Elucidating the structure-property relationships of donor-π-acceptor dyes for dye-sensitized solar cells (DSSCs) through rapid library synthesis by a one-pot procedure.

scientific article

Elucidation of the structure-property relationship of p-type organic semiconductors through rapid library construction via a one-pot, Suzuki-Miyaura coupling reaction.

scientific article

Functional and Structural Analysis of a Key Region of the Cell Wall Inhibitor Moenomycin

scientific article

Generation of an 4-Isoxazolyl Anion Species: Facile Access to Multifunctionalized Isoxazoles

scientific article published on 26 September 2016

Gold(I)-Catalyzed Intramolecular SEAr Reaction: Efficient Synthesis of Isoxazole-Containing Fused Heterocycles.

scientific article published on 5 January 2018

JBIR-56 and JBIR-57, 2(1H)-pyrazinones from a marine sponge-derived Streptomyces sp. SpD081030SC-03.

scientific article published on 5 July 2011

Micro-flow synthesis and structural analysis of sterically crowded diimine ligands with five aryl rings

scientific article published on November 2013

Micro-flow synthesis of β-amino acid derivatives via a rapid dual activation approach

scientific article published on 03 April 2020

One-pot, three-component coupling approach to the synthesis of α-iminocarboxamides

scientific article published on 03 August 2012

Peptide Synthesis Utilizing Micro-flow Technology

article

Peptide-Chain Elongation Using Unprotected Amino Acids in a Micro-Flow Reactor

scientific article published on 24 October 2019

Photodynamic therapy using a cytotoxic photosensitizer porphyrus envelope that targets the cell membrane

scientific article published on 24 October 2017

Rapid Synthesis of D-A'-π-A Dyes through a One-Pot Three-Component Suzuki-Miyaura Coupling and an Evaluation of their Photovoltaic Properties for Use in Dye-Sensitized Solar Cells

scientific article

Rapid Synthesis of Thiophene-Based, Organic Dyes for Dye-Sensitized Solar Cells (DSSCs) by a One-Pot, Four-Component Coupling Approach.

scientific article published on 28 May 2015

Rapid and Mild Synthesis of Amino Acid N -Carboxy Anhydrides: Basic-to-Acidic Flash Switching in a Microflow Reactor

scientific article published on 24 July 2018

Rapid assembly of resorcylic acid lactone frameworks through sequential palladium-catalyzed coupling reactions.

scientific article

Recent progresses in the synthesis of functionalized isoxazoles

Ribosomal synthesis of backbone-macrocyclic peptides containing γ-amino acids.

scientific article

Sequential S(N)Ar Reaction/Suzuki-Miyaura Coupling/C-H Direct Arylations Approach for the Rapid Synthesis of Tetraaryl-Substituted Pyrazoles

scientific article published on 19 June 2015

Sequential coupling approach to the synthesis of nickel(II) complexes with N-aryl-2-amino phenolates.

scientific article

Single-Step, Rapid, and Mild Synthesis of β-Amino Acid N-Carboxy Anhydrides Using Micro-Flow Technology

scientific article published on 28 November 2019

Solution-phase automated synthesis of an α-amino aldehyde as a versatile intermediate.

scientific article published on 17 January 2017

Structural Analysis of the Contacts Anchoring Moenomycin to Peptidoglycan Glycosyltransferases and Implications for Antibiotic Design

scientific article

Synthesis of bicyclic enediynes that possess a photosensitive triggering device and exhibit strong DNA cleaving activity.

scientific article published on 2 July 2010

The Design, Synthesis, and Evaluation of 1,5,7-Trisubstituted-3-Pyridyl-Xanthones for Use as Insecticides Starting from Pyripyropene A.

scientific article published on 9 November 2016

The Synthesis of trans-Flavan-3-ol Gallates by Regioselective Oxidative Etherification and Their Cytotoxicity Mediated by 67 LR.

scientific article published on 13 July 2016

The design, synthesis, and evaluation of organic dithienopyrrole-based D-π-A dyes for use as sensitizers in photodynamic therapy

scientific article published on 17 July 2018

The α-Glycosidation of Partially Unprotected N-Acetyl and N-Glycolyl Sialyl Donors in the Absence of a Nitrile Solvent Effect.

scientific article published on 8 April 2016

Total synthesis and stereochemistry revision of mannopeptimycin aglycone

scientific article published on 13 August 2014

Total synthesis of feglymycin based on a linear/convergent hybrid approach using micro-flow amide bond formation.

scientific article published on 28 November 2016

Total synthesis of spiruchostatin B aided by an automated synthesizer

scientific article published on 29 March 2011

List of works by Shinichiro Fuse

6-Azido-6-deoxy-l-idose as a Hetero-Bifunctional Spacer for the Synthesis of Azido-Containing Chemical Probes.

A Formal Total Synthesis of Taxol Aided by an Automated Synthesizer

A rapid and clean synthetic approach to cyclic peptides via micro-flow peptide chain elongation and photochemical cyclization: synthesis of a cyclic RGD peptide.

Anti-influenza virus compound from Streptomyces sp. RI18.

Asymmetric Total Synthesis of ent-Pyripyropene A.

Complete characterization of the seventeen step moenomycin biosynthetic pathway

Continuous in situ generation and reaction of phosgene in a microflow system

Continuous-flow synthesis of activated vitamin D3 and its analogues

Continuous-flow synthesis of vitamin D3.

Design, synthesis and evaluation of carbamate-modified (-)-N(1)-phenethylnorphysostigmine derivatives as selective butyrylcholinesterase inhibitors.

Design, synthesis, and evaluation of azo D-π-A dyes as photothermal agents

Design, synthesis, evaluation and QSAR analysis of N(1)-substituted norcymserine derivatives as selective butyrylcholinesterase inhibitors.

Development of 1-aryl-3-furanyl/thienyl-imidazopyridine templates for inhibitors against hypoxia inducible factor (HIF)-1 transcriptional activity.

Development of dual targeting inhibitors against aggregations of amyloid-β and tau protein.

Directing/protecting-group-free synthesis of tetraaryl-substituted pyrazoles through four direct arylations on an unsubstituted pyrazole scaffold

Efficient amide bond formation through a rapid and strong activation of carboxylic acids in a microflow reactor

Elucidating the structure-property relationships of donor-π-acceptor dyes for dye-sensitized solar cells (DSSCs) through rapid library synthesis by a one-pot procedure.

Elucidation of the structure-property relationship of p-type organic semiconductors through rapid library construction via a one-pot, Suzuki-Miyaura coupling reaction.

Functional and Structural Analysis of a Key Region of the Cell Wall Inhibitor Moenomycin

Generation of an 4-Isoxazolyl Anion Species: Facile Access to Multifunctionalized Isoxazoles

Gold(I)-Catalyzed Intramolecular SEAr Reaction: Efficient Synthesis of Isoxazole-Containing Fused Heterocycles.

JBIR-56 and JBIR-57, 2(1H)-pyrazinones from a marine sponge-derived Streptomyces sp. SpD081030SC-03.

Micro-flow synthesis and structural analysis of sterically crowded diimine ligands with five aryl rings

Micro-flow synthesis of β-amino acid derivatives via a rapid dual activation approach

One-pot, three-component coupling approach to the synthesis of α-iminocarboxamides

Peptide Synthesis Utilizing Micro-flow Technology

Peptide-Chain Elongation Using Unprotected Amino Acids in a Micro-Flow Reactor

Photodynamic therapy using a cytotoxic photosensitizer porphyrus envelope that targets the cell membrane

Rapid Synthesis of D-A'-π-A Dyes through a One-Pot Three-Component Suzuki-Miyaura Coupling and an Evaluation of their Photovoltaic Properties for Use in Dye-Sensitized Solar Cells

Rapid Synthesis of Thiophene-Based, Organic Dyes for Dye-Sensitized Solar Cells (DSSCs) by a One-Pot, Four-Component Coupling Approach.

Rapid and Mild Synthesis of Amino Acid N -Carboxy Anhydrides: Basic-to-Acidic Flash Switching in a Microflow Reactor

Rapid assembly of resorcylic acid lactone frameworks through sequential palladium-catalyzed coupling reactions.

Recent progresses in the synthesis of functionalized isoxazoles

Ribosomal synthesis of backbone-macrocyclic peptides containing γ-amino acids.

Sequential S(N)Ar Reaction/Suzuki-Miyaura Coupling/C-H Direct Arylations Approach for the Rapid Synthesis of Tetraaryl-Substituted Pyrazoles

Sequential coupling approach to the synthesis of nickel(II) complexes with N-aryl-2-amino phenolates.

Single-Step, Rapid, and Mild Synthesis of β-Amino Acid N-Carboxy Anhydrides Using Micro-Flow Technology

Solution-phase automated synthesis of an α-amino aldehyde as a versatile intermediate.

Structural Analysis of the Contacts Anchoring Moenomycin to Peptidoglycan Glycosyltransferases and Implications for Antibiotic Design

Synthesis of bicyclic enediynes that possess a photosensitive triggering device and exhibit strong DNA cleaving activity.

The Design, Synthesis, and Evaluation of 1,5,7-Trisubstituted-3-Pyridyl-Xanthones for Use as Insecticides Starting from Pyripyropene A.

The Synthesis of trans-Flavan-3-ol Gallates by Regioselective Oxidative Etherification and Their Cytotoxicity Mediated by 67 LR.

The design, synthesis, and evaluation of organic dithienopyrrole-based D-π-A dyes for use as sensitizers in photodynamic therapy

The α-Glycosidation of Partially Unprotected N-Acetyl and N-Glycolyl Sialyl Donors in the Absence of a Nitrile Solvent Effect.

Total synthesis and stereochemistry revision of mannopeptimycin aglycone

Total synthesis of feglymycin based on a linear/convergent hybrid approach using micro-flow amide bond formation.

Total synthesis of spiruchostatin B aided by an automated synthesizer