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List of works by Luigi André Agrofoglio

3'-(1,2,3-Triazol-1-yl)-3'-deoxythymidine analogs as substrates for human and Ureaplasma parvum thymidine kinase for structure-activity investigations.

scientific article

Active site labeling of cysteine cathepsins by a straightforward diazomethylketone probe derived from the N-terminus of human cystatin C.

scientific article

Alkyne-Azide Click Chemistry Mediated Carbanucleosides Synthesis

article

Analysis and validation of the phosphorylated metabolites of two anti-human immunodeficiency virus nucleotides (stavudine and didanosine) by pressure-assisted CE-ESI-MS/MS in cell extracts: sensitivity enhancement by the use of perfluorinated acids

scientific article published on 01 June 2006

Artificial receptors for the extraction of nucleoside metabolite 7-methylguanosine from aqueous media made by molecular imprinting.

scientific article

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2.

scientific article published on 28 December 2017

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3

scientific article published on 30 June 2018

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5

scientific article published on 30 June 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6

scientific article published on 28 December 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes⁻4

scientific article published on 31 December 2018

Combination of computational methods, adsorption isotherms and selectivity tests for the conception of a mixed non-covalent-semi-covalent molecularly imprinted polymer of vanillin.

scientific article published on 27 June 2013

Cross-Metathesis Mediated Synthesis of New Acyclic Nucleoside Phosphonates

scientific article published on 01 January 2007

Design and Synthesis of Various 5'-Deoxy-5'-(4-Substituted-1,2,3-Triazol-1-yl)-Uridine Analogues as Inhibitors of Mycobacterium tuberculosis Mur Ligases

scientific article published on 26 October 2020

Determination at ppb level of an anti-human immunodeficiency virus nucleoside drug by capillary electrophoresis-electrospray ionization tandem mass spectrometry.

scientific article published in October 2000

Efficient synthesis of D-[1'-13C]-ribonucleosides for incorporation into oligo-RNA

scientific article published on 01 April 2001

Efficient synthesis of unprotected C-5-aryl/heteroaryl-2'-deoxyuridine via a Suzuki-Miyaura reaction in aqueous media.

scientific article

Evaluation of molecularly imprinted polymers using 2',3',5'-tri-O-acyluridines as templates for pyrimidine nucleoside recognition

scientific article published on 31 July 2014

HPLC and mass spectrometry analysis of the enzymatic hydrolysis of anti-HIV pronucleotide diastereomers.

scientific article

Highly convergent synthesis and antiviral activity of (E)-but-2-enyl nucleoside phosphonoamidates

scientific article published on 31 January 2018

Human and viral nucleoside/nucleotide kinases involved in antiviral drug activation: structural and catalytic properties.

scientific article published on April 2010

Inhibition of human immunodeficiency virus type 1 reverse transcriptase by the 5'-triphosphate beta enantiomers of cytidine analogs

scientific article

Liquid chromatographic separation of phosphoramidate diastereomers on a polysaccharide-type chiral stationary phase.

scientific article

Looking for new pyrimidine acyclic nucleotide analogues designed for phosphorylation by human UMP-CMP kinase.

scientific article published in January 2007

Love Acoustic Wave-Based Devices and Molecularly-Imprinted Polymers as Versatile Sensors for Electronic Nose or Tongue for Cancer Monitoring.

scientific article

Mass spectrometry based methods for analysis of nucleosides as antiviral drugs and potential tumor biomarkers

scientific article published on 01 January 2007

Microwave-Assisted Silylation-Amination of Uracil Acyclonucleosides to 4-Alkylamino-2(1H)-Pyrimidinone Analogues

Microwave-assisted syntheses of nucleosides and their precursors.

scientific article published on February 2010

Molecularly imprinted polymer of 5-methyluridine for solid-phase extraction of pyrimidine nucleoside cancer markers in urine.

scientific article

Novel antiviral C5-substituted pyrimidine acyclic nucleoside phosphonates selected as human thymidylate kinase substrates

scientific article

Nucleotide binding to human UMP-CMP kinase using fluorescent derivatives -- a screening based on affinity for the UMP-CMP binding site

scientific article

Olefin metathesis route to antiviral nucleosides

scientific article

Palladium-assisted routes to nucleosides.

scientific article

Phosphorylation of dGMP analogs by vaccinia virus TMP kinase and human GMP kinase

scientific article published on 23 July 2009

Potential and perspectives of cyclonucleosides.

scientific article published on January 2010

Preparation of acyclo nucleoside phosphonate analogues based on cross-metathesis

article

Recent progress for the synthesis of selected carbocyclic nucleosides

scientific article published on 29 September 2015

Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs

scientific article published on 19 July 2018

Simultaneous analysis of several antiretroviral nucleosides in rat-plasma by high-performance liquid chromatography with UV using acetic acid/hydroxylamine buffer Test of this new volatile medium-pH for HPLC-ESI-MS/MS.

scientific article published in July 2005

Simultaneous quantitation of nucleoside HIV-1 reverse transcriptase inhibitors by short-end injection capillary electrochromatography on a beta-cyclodextrin-bonded silica stationary phase.

scientific article published in August 2001

Sonication-Assisted Synthesis of(E)-2-Methyl-but-2-enyl Nucleoside Phosphonate Prodrugs

Specificity enhancement with LC-positive ESI-MS/MS for the measurement of nucleotides: application to the quantitative determination of carbovir triphosphate, lamivudine triphosphate and tenofovir diphosphate in human peripheral blood mononuclear ce

scientific article published in February 2008

Straightforward synthesis of 2,4,6-trisubstituted 1,3,5-triazine compounds targeting cysteine cathepsins K and S.

scientific article published on 6 May 2016

Study of Copper(I) Catalysts for the Synthesis of Carbanucleosides via Azide-Alkyne 1,3-Dipolar Cycloaddition

Study of Different Copper (I) Catalysts for the “Click Chemistry” Approach to Carbanucleosides

scientific article published on 01 January 2007

Synthesis and Anti-HIV Evaluation of 3′-Triazolo Nucleosides ⬇️

scientific article published on April 1, 2011

Synthesis and antiviral activity of novel acyclic nucleosides in the 5-alkynyl- and 6-alkylfuro[2,3-d]pyrimidine series.

scientific article published on February 2005

Synthesis and antiviral evaluation of C5-substituted-(1,3-diyne)-2'-deoxyuridines.

scientific article published on 21 April 2012

Synthesis and antiviral evaluation of bis(POM) prodrugs of (E)-[4′-phosphono-but-2′-en-1′-yl]purine nucleosides

article

Synthesis and broad spectrum antiviral evaluation of bis(POM) prodrugs of novel acyclic nucleosides

scientific article published on 4 July 2013

Synthesis and characterization of various 5'-dye-labeled ribonucleosides

scientific article published on 01 September 2018

Synthesis of 1,2,3-triazolo-carbanucleoside analogues of ribavirin targeting an HCV in replicon.

scientific article published in August 2003

Synthesis of 5'-thioalkyl, sulfoxide and sulfone pyrimidine nucleosides

scientific article published on 01 April 1999

Synthesis of 5-haloethynyl- and 5-(1,2-dihalo)vinyluracil nucleosides: antiviral activity and cellular toxicity.

scientific article published on November 2005

Synthesis of a molecularly imprinted polymer to isolate glucosamine from plant extracts by an ionic-non-covalent dual approach

scientific article published on 20 January 2015

Synthesis of a novel heterocyclic ring system: 2-thia-3,5,6,7,9-pentaazabenz[cd]azulenes

scientific article published in January 2002

Synthesis of dihydropyrimidine α,γ-diketobutanoic acid derivatives targeting HIV integrase

scientific article

Synthesis of isotopically labeled D-[1'-13C]ribonucleoside phosphoramidites

scientific article published on 01 March 2001

Synthesis of new C5-(1-substituted-1,2,3-triazol-4 or 5-yl)-2'-deoxyuridines and their antiviral evaluation

scientific article published on 21 December 2010

Synthesis of water-compatible imprinted polymers of in situ produced fructosazine and 2,5-deoxyfructosazine ⬇️

scientific article published on July 22, 2012

The Preparation of Trisubstituted Alkenyl Nucleoside Phosphonates under Ultrasound-Assisted Olefin Cross-Metathesis

scientific article published on 20 August 2013

Thiopurine Derivative-Induced Fpg/Nei DNA Glycosylase Inhibition: Structural, Dynamic and Functional Insights

scientific article published on 17 March 2020

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