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List of works by Garrett C Moraski

A dual read-out assay to evaluate the potency of compounds active against Mycobacterium tuberculosis

scientific article

Advancement of Imidazo[1,2-a]pyridines with Improved Pharmacokinetics and Nanomolar Activity Against Mycobacterium tuberculosis

scientific article published on July 2013

Advent of Imidazo[1,2-a]pyridine-3-carboxamides with Potent Multi- and Extended Drug Resistant Antituberculosis Activity

scientific article

Allylic thiocyanates as a new class of antitubercular agents

scientific article published on 21 August 2012

Bactericidal activity of an imidazo[1, 2-a]pyridine using a mouse M. tuberculosis infection model

scientific article (publication date: 2014)

ChemInform Abstract: One-Step Syntheses of Nitrofuranyl Benzimidazoles that Are Active Against Multidrug-Resistant Bacteria

ChemInform Abstract: Utilization of the Suzuki Coupling to Enhance the Antituberculosis Activity of Aryloxazoles

Design, synthesis, and study of a mycobactin-artemisinin conjugate that has selective and potent activity against tuberculosis and malaria

scientific article

Generation and exploration of new classes of antitubercular agents: The optimization of oxazolines, oxazoles, thiazolines, thiazoles to imidazo[1,2-a]pyridines and isomeric 5,6-fused scaffolds

scientific article published on 16 February 2012

Imidazo[1,2-a]Pyridine-3-Carboxamides Are Active Antimicrobial Agents against Mycobacterium avium Infection In Vivo

scientific article published on 23 May 2016

N-((1-benzyl-1H-1,2,3-triazol-4-yl)methyl)arylamide as a new scaffold that provides rapid access to antimicrotubule agents: synthesis and evaluation of antiproliferative activity against select cancer cell lines

scientific article

One-step syntheses of nitrofuranyl benzimidazoles that are active against multidrug-resistant bacteria

scientific article

Preparation and Evaluation of Potent Pentafluorosulfanyl-Substituted Anti-Tuberculosis Compounds.

scientific article published on 27 June 2017

Scaffold-switching: an exploration of 5,6-fused bicyclic heteroaromatics systems to afford antituberculosis activity akin to the imidazo[1,2-a]pyridine-3-carboxylates

scientific article

Streamlined Processes for the Synthesis of a Farnesyl Transferase Inhibitor Drug Candidate

Structure-Based Mechanism for Oxidative Decarboxylation Reactions Mediated by Amino Acids and Heme Propionates in Coproheme Decarboxylase (HemQ).

scientific article published on 12 December 2016

Structure-activity relationship of new anti-tuberculosis agents derived from oxazoline and oxazole benzyl esters

scientific article

Syntheses and biological studies of novel spiropiperazinyl oxazolidinone antibacterial agents using a spirocyclic diene derived acylnitroso Diels-Alder reaction

scientific article

Thiolates chemically induce redox activation of BTZ043 and related potent nitroaromatic anti-tuberculosis agents

scientific article published on 25 February 2013

UTILIZTION OF THE SUZUKI COUPLING TO ENHANCE THE ANTITUBERCULOSIS ACTIVITY OF ARYL OXAZOLES.

scientific article

Unusual Peroxide-Dependent, Heme-Transforming Reaction Catalyzed by HemQ.

scientific article published on 23 June 2015

Utilization of microbial iron assimilation processes for the development of new antibiotics and inspiration for the design of new anticancer agents

scientific article published on 07 January 2009

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