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List of works by Christophe Verlinde

Dialkylimidazole inhibitors of Trypanosoma cruzi sterol 14α-demethylase as anti-Chagas disease agents

scientific article

Efficacy, Pharmacokinetics, and Metabolism of Tetrahydroquinoline Inhibitors of Plasmodium falciparum Protein Farnesyltransferase

scientific article

Glycogen synthase kinase 3 is a potential drug target for African trypanosomiasis therapy

scientific article published on 21 July 2008

Leishmania donovani tyrosyl-tRNA synthetase structure in complex with a tyrosyl adenylate analog and comparisons with human and protozoan counterparts

scientific article published on 18 April 2017

Pharmacological Characterization, Structural Studies, and In Vivo Activities of Anti-Chagas Disease Lead Compounds Derived from Tipifarnib

scientific article

Rational modification of a candidate cancer drug for use against Chagas disease

scientific article published on March 2009

Second generation analogues of the cancer drug clinical candidate tipifarnib for anti-Chagas disease drug discovery.

scientific article

Second generation tetrahydroquinoline-based protein farnesyltransferase inhibitors as antimalarials

scientific article published on 28 August 2007

Structural genomics of pathogenic protozoa: an overview

scientific article

Structurally simple farnesyltransferase inhibitors arrest the growth of malaria parasites

scientific article published in August 2005

Structurally simple inhibitors of lanosterol 14alpha-demethylase are efficacious in a rodent model of acute Chagas disease.

scientific article published on June 2009

Synthesis and Conformational Analysis of 2?-Deoxy-2?-(3-methoxybenzamido)adenosine, a rational-designed inhibitor of trypanosomal glyceraldehyde phosphate dehydrogenase (GAPDH)

article

The protein farnesyltransferase inhibitor Tipifarnib as a new lead for the development of drugs against Chagas disease

scientific article published on August 2005

The structure of the D3 domain of Plasmodium falciparum myosin tail interacting protein MTIP in complex with a nanobody

scientific article