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List of works by Janos Sapi

4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies

scientific article

Chemical biology: contribution to molecular therapeutic innovation--a new role for chemistry? Report from the thematic symposium organized by the SCT (French Medicinal Chemistry Society), November 26th, 2013

scientific article published on 01 April 2014

Condensation of beta-diester titanium enolates with carbonyl substrates: a combined DFT and experimental investigation

scientific article published in November 2009

Cyclopropyl-tryptamine analogues: synthesis and biological evaluation as 5-HT(6) receptor ligands

scientific article published on 05 November 2012

Cytotoxic bis-3,4-dihydro-beta-carbolines and bis-beta-carbolines

Design, Synthesis, and Use of MMP-2 Inhibitor-Conjugated Quantum Dots in Functional Biochemical Assays

scientific article published in March 2016

Diastereomer Interconversion via Enolization: A Case Study

scientific article published on 04 September 2015

Direct chiral separation of unnatural amino acids by high‐performance liquid chromatography on a ristocetin a‐bonded stationary phase ⬇️

scientific article published on January 1, 2001

First domino radical cyclisation/Smiles rearrangement combination

scientific article published on 23 January 2012

Indirect high-performance liquid chromatographic separation of stereoisomers of beta-alkyl-substituted amino acids by the application of (S)-N-(4-nitrophenoxycarbonyl)phenylalanine methoxyethyl ester as chiral derivatizing agent.

scientific article

Inhibition of human leukocyte elastase, plasmin and matrix metalloproteinases by oleic acid and oleoyl-galardin derivative(s)

scientific article published on 10 December 2010

Interfacing chemical biology and drug discovery: report from the 50th International Conference on Medicinal Chemistry of the SCT (French Medicinal Chemistry Society), July 2-4, 2014, Rouen, France.

scientific article published on 5 December 2014

Introduction of the 4-(4-bromophenyl)benzenesulfonyl group to hydrazide analogs of Ilomastat leads to potent gelatinase B (MMP-9) inhibitors with improved selectivity

scientific article

Multicomponent reactions studies: Yonemitsu-type trimolecular condensations promoted by Ti(IV) derivatives

Multifunctional Nanoprobes for Cancer Cell Targeting, Imaging and Anticancer Drug Delivery

scientific article published in 2015

Multiple dual-mode centrifugal partition chromatography, a semi-continuous development mode for routine laboratory-scale purifications

article

Palladium nanoparticles in catalytic carbon nanoreactors: the effect of confinement on Suzuki–Miyaura reactions

Palladium nanoparticles on carbon nanotubes as catalysts of cross-coupling reactions

Photochemical aryl radical cyclizations to give (E)-3-ylideneoxindoles

scientific article published on 30 September 2014

Radical Smiles Rearrangement: An Update

scientific article

Simultaneous presence of unsaturation and long alkyl chain at P'1 of Ilomastat confers selectivity for gelatinase A (MMP-2) over gelatinase B (MMP-9) inhibition as shown by molecular modelling studies

scientific article published on 06 May 2007

Synthesis and anticancer activity of new pyrrolocarbazoles and pyrrolo-beta-carbolines.

scientific article

Synthesis of two new heteroaromatic beta-carboline-fused pentacycles. Observation of a new intercalating agent.

scientific article

The NC1 domain of type XIX collagen inhibits melanoma cell migration

scientific article published on 14 September 2010

TiCl4-promoted condensation of methyl acetoacetate, isobutyraldehyde, and indole: a theoretical and experimental study

scientific article published on 09 March 2015

TiCl4/Et3N-promoted three-component condensation between aromatic heterocycles, aldehydes, and active methylene compounds

scientific article published on 9 August 2008

Yonemitsu-type condensations catalysed by proline and Eu(OTf)3

scholarly article in RSC Advances, vol. 4 no. 89, 2014

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