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List of works by Marta Artola

1,6-Cyclophellitol Cyclosulfates: A New Class of Irreversible Glycosidase Inhibitor

scientific article published on 13 July 2017

A Divergent Synthesis ofl-arabino- andd-xylo-Configured Cyclophellitol Epoxides and Aziridines

Activity-Based Probes for Glycosidases: Profiling and Other Applications

scientific article

Activity-based probes for functional interrogation of retaining β-glucuronidases

scientific article

An overview of activity-based probes for glycosidases

scientific article published on 13 August 2019

Carba-cyclophellitols Are Neutral Retaining-Glucosidase Inhibitors.

scientific article published on 2 May 2017

Chemical Proteomics Identifies SLC25A20 as a Functional Target of the Ingenol Class of Actinic Keratosis Drugs

scientific article published on 6 December 2017

Competitive and Covalent Inhibitors of Human Lysosomal Retaining Exoglucosidases

Direct Stereoselective Aziridination of Cyclohexenols with 3-Amino-2-(trifluoromethyl)quinazolin-4(3H )-one in the Synthesis of Cyclitol Aziridine Glycosidase Inhibitors

scientific article published on 11 January 2019

Discovering the Microbial Enzymes Driving Drug Toxicity with Activity-Based Protein Profiling

scientific article published on 12 December 2019

Distinguishing the differences in beta-glycosylceramidase folds, dynamics, and actions informs therapeutic uses

article

Effective GTP-Replacing FtsZ Inhibitors and Antibacterial Mechanism of Action

scientific article published on 30 December 2014

Functionalized Cyclophellitols Are Selective Glucocerebrosidase Inhibitors and Induce a Bona Fide Neuropathic Gaucher Model in Zebrafish

scientific article published on 04 March 2019

Gluco-1 H-imidazole: A New Class of Azole-Type β-Glucosidase Inhibitor.

scientific article published on 30 March 2018

Glycosphingolipids and lysosomal storage disorders as illustrated by gaucher disease

scientific article published on 26 November 2019

Human glucocerebrosidase mediates formation of xylosyl-cholesterol by β-xylosidase and transxylosidase reactions

scientific article published on 23 December 2020

Identification of a Novel Orally Bioavailable Phosphodiesterase 10A (PDE10A) Inhibitor with Efficacy in Animal Models of Schizophrenia

scientific article published on 12 January 2015

In vivo inactivation of glycosidases by conduritol B epoxide and cyclophellitol as revealed by activity-based protein profiling

scientific article published on 02 February 2019

New irreversible α-L-iduronidase inhibitors and activity-based probes

scientific article published on 26 November 2018

New synthetic inhibitors of fatty acid synthase with anticancer activity

scientific article published on 16 May 2012

Novel activity-based probes for N-acylethanolamine acid amidase

scientific article published on 16 October 2017

Plant Glycosides and Glycosidases: A Treasure-Trove for Therapeutics

scientific article published on 07 April 2020

Rational Design of Mechanism-Based Inhibitors and Activity-Based Probes for the Identification of Retaining α-l-Arabinofuranosidases

scientific article published on 26 February 2020

Role of cannabinoid receptor CB2 in HER2 pro-oncogenic signaling in breast cancer

scientific article

Role of β-glucosidase 2 in aberrant glycosphingolipid metabolism: model of glucocerebrosidase deficiency in zebrafish

scientific article published on 27 September 2019

Structure of a GH51 α-L-arabinofuranosidase from Meripilus giganteus: conserved substrate recognition from bacteria to fungi

scientific article published on 16 October 2020

Synthetic inhibitors of bacterial cell division targeting the GTP-binding site of FtsZ.

scientific article

The Synthesis of Cyclophellitol-Aziridine and Its Configurational and Functional Isomers

The structural assembly switch of cell division protein FtsZ probed with fluorescent allosteric inhibitors.

scientific article published on 21 October 2016

Towards broad spectrum activity-based glycosidase probes: synthesis and evaluation of deoxygenated cyclophellitol aziridines.

scientific article published on 8 November 2017

Xylose-Configured Cyclophellitols as Selective Inhibitors for Glucocerebrosidase

scientific article published on 13 September 2021

α-galactosidase A1.1 can functionally complement human α-galactosidase A deficiency associated with Fabry disease

scientific article published in Journal of Biological Chemistry

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