List of works - Mikhail Reibarkh

13C NMR-Based Approaches for Solving Challenging Stereochemical Problems.

scientific article published on 22 May 2019

1J(CC)-edited HSQC-1,n-ADEQUATE: a new paradigm for simultaneous direct and long-range carbon-carbon correlation

scientific article published on 19 September 2012

A multifunctional catalyst that stereoselectively assembles prodrugs.

scientific article

A new class of prolylcarboxypeptidase inhibitors, part 2: the aminocyclopentanes.

scientific article published in March 2012

Asymmetric synthesis of cyclic indole aminals via 1,3-stereoinduction

scientific article published on 03 September 2014

Band-Selective 2D HSQMBC: A Universal Technique for Detection and Measurement of 35,37Cl Isotope Effects for 13C Nuclei

scientific article published on 28 September 2016

Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety

scientific article published on 21 March 2019

Broadband inversion of 1J(CC) responses in 1,n-ADEQUATE spectra

scientific article published on 9 August 2013

Complex macrocycle exploration: parallel, heuristic, and constraint-based conformer generation using ForceGen.

scientific article

Coniothyrione: anatomy of a structure revision

scientific article published on 15 May 2013

Discovery of N-[Bis(4-methoxyphenyl)methyl]-4-hydroxy-2-(pyridazin-3-yl)pyrimidine-5-carboxamide (MK-8617), an Orally Active Pan-Inhibitor of Hypoxia-Inducible Factor Prolyl Hydroxylase 1-3 (HIF PHD1-3) for the Treatment of Anemia

scientific article published on 30 November 2016

Discovery of Novel Indoline Cholesterol Ester Transfer Protein Inhibitors (CETP) through a Structure-Guided Approach

scientific article published on 4 January 2016

Discovery of a Photoinduced Dark Catalytic Cycle Using in Situ LED-NMR Spectroscopy

scientific article published on 10 October 2018

Discovery of highly potent and efficacious MC4R agonists with spiroindane N-Me-1,2,4-triazole privileged structures for the treatment of obesity

scientific article published on 19 September 2010

Eukaryotic initiation factor (eIF) 1 carries two distinct eIF5-binding faces important for multifactor assembly and AUG selection

scientific article

Facile Quantum Yield Determination via NMR Actinometry.

scientific article published on 28 March 2018

Identification of individual protein-ligand NOEs in the limit of intermediate exchange

scientific article published on 09 September 2006

Interatomic potentials and solvation parameters from protein engineering data for buried residues

scientific article

Investigation of Cardiovascular Effects of Tetrahydro-β-carboline sstr3 antagonists.

scientific article published on 21 April 2014

NMR study of monomer-dimer equilibrium of barstar in solution.

scientific article published in March 2001

Oxyfunctionalization of the Remote C-H Bonds of Aliphatic Amines by Decatungstate Photocatalysis

scientific article

PBLG as a versatile liquid crystalline medium for anisotropic NMR data acquisition

scientific article published on 01 April 2019

Promotion of a Ti-Mediated Mannich Reaction by a Proton Source

scientific article published on 21 December 2015

SAR exploration at the C-3 position of tetrahydro-β-carboline sstr3 antagonists

scientific article published on 10 February 2016

Secondary amine selective Petasis (SASP) bioconjugation

scientific article published on 07 November 2019

Selective pharmacological targeting of a DEAD box RNA helicase.

scientific article

Small molecule inhibition of phosphatidylinositol-3,4,5-triphosphate (PIP3) binding to pleckstrin homology domains ⬇️

scientific article published on November 16, 2010

Small-molecule inhibition of the interaction between the translation initiation factors eIF4E and eIF4G

scientific article

Structure elucidation of uniformly (13)C labeled small molecule natural products

scientific article published in December 2015

Structure elucidation of uniformly 13C labeled small molecule natural products ⬇️

scientific article published on December 2015

Substituted fused bicyclic pyrrolizinones as potent, orally bioavailable hNK1 antagonists.

scientific article

The C-terminal domain of eukaryotic initiation factor 5 promotes start codon recognition by its dynamic interplay with eIF1 and eIF2β

scientific article

The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes.

scientific article

The protecting-group free selective 3'-functionalization of nucleosides

scientific article published on 18 January 2017

Three-dimensional structure of toxin OSK1 from Orthochirus scrobiculosus scorpion venom

scientific article

Three‐dimensional structure of binase in solution ⬇️

scientific article published on July 17, 1998

Trapping‐Enrichment Multi‐dimensional Liquid Chromatography with On‐Line Deuterated Solvent Exchange for Streamlined Structure Elucidation at the Microgram Scale

Use of hydrostatic pressure for modulation of protein chemical modification and enzymatic selectivity

scientific article published on 18 April 2016

Using Electron Paramagnetic Resonance Spectroscopy To Facilitate Problem Solving in Pharmaceutical Research and Development.

scientific article published on 20 June 2016

Visualizing small differences using subtractive chromatographic analysis.

scientific article published on 13 September 2016

[I87E mutation prevents barstar dimerization]

scientific article published on 01 November 2004

pK measurements for the SAMPL6 prediction challenge for a set of kinase inhibitor-like fragments

scientific article published on 01 October 2018

List of works by Mikhail Reibarkh

13C NMR-Based Approaches for Solving Challenging Stereochemical Problems.

1J(CC)-edited HSQC-1,n-ADEQUATE: a new paradigm for simultaneous direct and long-range carbon-carbon correlation

A multifunctional catalyst that stereoselectively assembles prodrugs.

A new class of prolylcarboxypeptidase inhibitors, part 2: the aminocyclopentanes.

Asymmetric synthesis of cyclic indole aminals via 1,3-stereoinduction

Band-Selective 2D HSQMBC: A Universal Technique for Detection and Measurement of 35,37Cl Isotope Effects for 13C Nuclei

Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety

Broadband inversion of 1J(CC) responses in 1,n-ADEQUATE spectra

Complex macrocycle exploration: parallel, heuristic, and constraint-based conformer generation using ForceGen.

Coniothyrione: anatomy of a structure revision

Discovery of N-[Bis(4-methoxyphenyl)methyl]-4-hydroxy-2-(pyridazin-3-yl)pyrimidine-5-carboxamide (MK-8617), an Orally Active Pan-Inhibitor of Hypoxia-Inducible Factor Prolyl Hydroxylase 1-3 (HIF PHD1-3) for the Treatment of Anemia

Discovery of Novel Indoline Cholesterol Ester Transfer Protein Inhibitors (CETP) through a Structure-Guided Approach

Discovery of a Photoinduced Dark Catalytic Cycle Using in Situ LED-NMR Spectroscopy

Discovery of highly potent and efficacious MC4R agonists with spiroindane N-Me-1,2,4-triazole privileged structures for the treatment of obesity

Eukaryotic initiation factor (eIF) 1 carries two distinct eIF5-binding faces important for multifactor assembly and AUG selection

Facile Quantum Yield Determination via NMR Actinometry.

Identification of individual protein-ligand NOEs in the limit of intermediate exchange

Interatomic potentials and solvation parameters from protein engineering data for buried residues

Investigation of Cardiovascular Effects of Tetrahydro-β-carboline sstr3 antagonists.

NMR study of monomer-dimer equilibrium of barstar in solution.

Oxyfunctionalization of the Remote C-H Bonds of Aliphatic Amines by Decatungstate Photocatalysis

PBLG as a versatile liquid crystalline medium for anisotropic NMR data acquisition

Promotion of a Ti-Mediated Mannich Reaction by a Proton Source

SAR exploration at the C-3 position of tetrahydro-β-carboline sstr3 antagonists

Secondary amine selective Petasis (SASP) bioconjugation

Selective pharmacological targeting of a DEAD box RNA helicase.

Small molecule inhibition of phosphatidylinositol-3,4,5-triphosphate (PIP3) binding to pleckstrin homology domains ⬇️

Small-molecule inhibition of the interaction between the translation initiation factors eIF4E and eIF4G

Structure elucidation of uniformly (13)C labeled small molecule natural products

Structure elucidation of uniformly 13C labeled small molecule natural products ⬇️

Substituted fused bicyclic pyrrolizinones as potent, orally bioavailable hNK1 antagonists.

The C-terminal domain of eukaryotic initiation factor 5 promotes start codon recognition by its dynamic interplay with eIF1 and eIF2β

The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes.

The protecting-group free selective 3'-functionalization of nucleosides

Three-dimensional structure of toxin OSK1 from Orthochirus scrobiculosus scorpion venom

Three‐dimensional structure of binase in solution ⬇️

Trapping‐Enrichment Multi‐dimensional Liquid Chromatography with On‐Line Deuterated Solvent Exchange for Streamlined Structure Elucidation at the Microgram Scale

Use of hydrostatic pressure for modulation of protein chemical modification and enzymatic selectivity

Using Electron Paramagnetic Resonance Spectroscopy To Facilitate Problem Solving in Pharmaceutical Research and Development.

Visualizing small differences using subtractive chromatographic analysis.

[I87E mutation prevents barstar dimerization]

pK measurements for the SAMPL6 prediction challenge for a set of kinase inhibitor-like fragments

pKa measurements for the SAMPL6 prediction challenge for a set of kinase inhibitor-like fragments