List of works - Antonio Massa

2,3-Dihydro-1,2-Diphenyl-substituted 4H-Pyridinone derivatives as new anti Flaviviridae inhibitors

scientific article published on 17 March 2011

3-Carboxylate-Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions

Active Methylene Compounds in the Synthesis of 3-substituted Isobenzofuranones, Isoindolinones and Related Compounds

Active methylene compounds in a very effective approach to 3-substituted isobenzofuranones through tandem aldol/lactonization reactions

article published in 2012

Asymmetric tandem hemiaminal-heterocyclization-aza-Mannich reaction of 2-formylbenzonitriles and amines using chiral phase transfer catalysis: an experimental and theoretical study

scholarly article in RSC Advances, vol. 6 no. 38, 2016

Bifunctional phase-transfer catalysis in the asymmetric synthesis of biologically active isoindolinones

scientific article published on 15 December 2015

Cascade reactions of glycine Schiff bases and chiral phase transfer catalysts in the synthesis of α-amino acids 3-substituted phthalides or isoindolinones

scholarly article in RSC Advances, vol. 4 no. 9, 2014

Chiral Phase Transfer Catalysis in the Asymmetric Synthesis of a 3,3-Disubstituted Isoindolinone and Determination of Its Absolute Configuration by VCD Spectroscopy

scientific article published on 12 May 2020

Chiral sulfoxides as activators of allyl trichlorosilanes in the stereoselective allylation of aldehydes

scientific article published on 17 May 2010

Chiral sulfoxides in the enantioselective allylation of aldehydes with allyltrichlorosilane: a kinetic study

scientific article published on 09 November 2012

Combined electrochemical/chemical methods for the synthesis and the molecular diversifying of isoindolinone-based heterocyclic scaffolds.

scientific article published on 12 January 2014

Cyclohexa-2,5-diene-1,4-dione-based antiproliferative agents: design, synthesis, and cytotoxic evaluation.

scientific article published on 30 April 2013

Design of chiral urea-quaternary ammonium salt hybrid catalysts for asymmetric reactions of glycine Schiff bases

scientific article

Design of inhibitors of influenza virus membrane fusion: synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series

scientific article published on 22 May 2013

Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based omega-acidic amino acids as glutamate receptors ligands

scientific article published on 14 November 2008

Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands

scientific article published on September 2011

Determination of the absolute configuration of a novel tetrasubstituted isoindolinone by vibrational circular dichroism.

scientific article published on 4 May 2017

Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication

scientific article published on 31 October 2016

Electrochemically Initiated Tandem and Sequential Conjugate Addition Processes: One-Pot Synthesis of Diverse Functionalized Isoindolinones

article

Exploring the role of chloro and methyl substitutions in 2-phenylthiomethyl-benzoindole derivatives for 5-LOX enzyme inhibition

scientific article published on 07 December 2015

Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase

scientific article published on 14 May 2014

Highly diastereo- and enantioselective organocatalytic synthesis of new heterocyclic hybrids isoindolinone-imidate and isoindolinone-phthalide

scholarly article in RSC Advances, vol. 6 no. 65, 2016

Isoindolinones as Michael Donors under Phase Transfer Catalysis: Enantioselective Synthesis of Phthalimidines Containing a Tetrasubstituted Carbon Stereocenter

scientific article published on 12 May 2015

Metal-Free Air Oxidation in a Convenient Cascade Approach for the Access to Isoquinoline-1,3,4(2H)-triones

scientific article published on 10 June 2019

Model-averaging of ab initio spectra for the absolute configuration assignment via vibrational circular dichroism

scientific article published on 17 October 2017

Multi-component, regio-selective aldol addition of β-ketoesters to aldehydes: scope and applications

article

New chelating agents for Cu(II), Fe(III), Al(III), and Zn(II) based on β-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone

Novel Highly Regioselective VO(acac)2/TBHP Mediated Oxidation of o-Alkenyl Phenols to o-Hydroxybenzyl Ketones ⬇️

scientific article published on May 2, 2003

Organocatalysts and sequential asymmetric cascade reactions in the synthesis of functionalized isoindolinones and benzoindolizidinones

scholarly article in RSC Advances, vol. 3 no. 42, 2013

Organocatalytic asymmetric synthesis of highly functionalized pyrrolizidines via cascade Michael/hemi-aminalization reactions of isoindolinones

Quick and easy access to N-Mannich bases of 1-isoindolinones by catalytic electroactivation of primary and secondary amines and tandem reaction with 2-formylbenzonitriles

article by Laura Palombi et al published 2015 in New Journal of Chemistry

Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures

Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture.

scientific article

Synthesis of new chiral 2,2'-bipyridine ligands and their application in copper-catalyzed asymmetric allylic oxidation and cyclopropanation.

scientific article

The Aldol Reactions of Active Methylene Compounds

The first organocatalytic asymmetric synthesis of 3-substituted isoindolinones

scholarly article in RSC Advances, vol. 2 no. 9, 2012

Trimethylchlorosilane and Silicon Tetrachloride in Two Novel Methodologies for the Efficient and Mild Aldol Addition of β-Keto Esters and Malonates to Aldehydes

article

List of works by Antonio Massa

2,3-Dihydro-1,2-Diphenyl-substituted 4H-Pyridinone derivatives as new anti Flaviviridae inhibitors

3-Carboxylate-Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions

Active Methylene Compounds in the Synthesis of 3-substituted Isobenzofuranones, Isoindolinones and Related Compounds

Active methylene compounds in a very effective approach to 3-substituted isobenzofuranones through tandem aldol/lactonization reactions

Asymmetric tandem hemiaminal-heterocyclization-aza-Mannich reaction of 2-formylbenzonitriles and amines using chiral phase transfer catalysis: an experimental and theoretical study

Bifunctional phase-transfer catalysis in the asymmetric synthesis of biologically active isoindolinones

Cascade reactions of glycine Schiff bases and chiral phase transfer catalysts in the synthesis of α-amino acids 3-substituted phthalides or isoindolinones

Chiral Phase Transfer Catalysis in the Asymmetric Synthesis of a 3,3-Disubstituted Isoindolinone and Determination of Its Absolute Configuration by VCD Spectroscopy

Chiral sulfoxides as activators of allyl trichlorosilanes in the stereoselective allylation of aldehydes

Chiral sulfoxides in the enantioselective allylation of aldehydes with allyltrichlorosilane: a kinetic study

Combined electrochemical/chemical methods for the synthesis and the molecular diversifying of isoindolinone-based heterocyclic scaffolds.

Cyclohexa-2,5-diene-1,4-dione-based antiproliferative agents: design, synthesis, and cytotoxic evaluation.

Design of chiral urea-quaternary ammonium salt hybrid catalysts for asymmetric reactions of glycine Schiff bases

Design of inhibitors of influenza virus membrane fusion: synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series

Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based omega-acidic amino acids as glutamate receptors ligands

Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands

Determination of the absolute configuration of a novel tetrasubstituted isoindolinone by vibrational circular dichroism.

Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication

Electrochemically Initiated Tandem and Sequential Conjugate Addition Processes: One-Pot Synthesis of Diverse Functionalized Isoindolinones

Exploring the role of chloro and methyl substitutions in 2-phenylthiomethyl-benzoindole derivatives for 5-LOX enzyme inhibition

Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase

Highly diastereo- and enantioselective organocatalytic synthesis of new heterocyclic hybrids isoindolinone-imidate and isoindolinone-phthalide

Isoindolinones as Michael Donors under Phase Transfer Catalysis: Enantioselective Synthesis of Phthalimidines Containing a Tetrasubstituted Carbon Stereocenter

Metal-Free Air Oxidation in a Convenient Cascade Approach for the Access to Isoquinoline-1,3,4(2H)-triones

Model-averaging of ab initio spectra for the absolute configuration assignment via vibrational circular dichroism

Multi-component, regio-selective aldol addition of β-ketoesters to aldehydes: scope and applications

New chelating agents for Cu(II), Fe(III), Al(III), and Zn(II) based on β-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone

Novel Highly Regioselective VO(acac)2/TBHP Mediated Oxidation of o-Alkenyl Phenols to o-Hydroxybenzyl Ketones ⬇️

Organocatalysts and sequential asymmetric cascade reactions in the synthesis of functionalized isoindolinones and benzoindolizidinones

Organocatalytic asymmetric synthesis of highly functionalized pyrrolizidines via cascade Michael/hemi-aminalization reactions of isoindolinones

Quick and easy access to N-Mannich bases of 1-isoindolinones by catalytic electroactivation of primary and secondary amines and tandem reaction with 2-formylbenzonitriles

Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures

Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture.

Synthesis of new chiral 2,2'-bipyridine ligands and their application in copper-catalyzed asymmetric allylic oxidation and cyclopropanation.

The Aldol Reactions of Active Methylene Compounds

The first organocatalytic asymmetric synthesis of 3-substituted isoindolinones

Trimethylchlorosilane and Silicon Tetrachloride in Two Novel Methodologies for the Efficient and Mild Aldol Addition of β-Keto Esters and Malonates to Aldehydes