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List of works by Paolo Guglielmi

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

scientific article published on 01 December 2019

A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms.

scientific article published on 20 January 2016

Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent.

scientific article

Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity

scientific article published on 01 December 2019

Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors

scientific article published on 04 July 2018

Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles

scientific article published on 29 January 2019

Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents

scientific article published on 19 October 2017

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold

scientific article published on 01 December 2019

Enantiomers of triclabendazole sulfoxide: Analytical and semipreparative HPLC separation, absolute configuration assignment, and transformation into sodium salt.

scientific article published on 16 March 2017

Inhibition of Human Monoamine Oxidase: Biological and Molecular Modeling Studies on Selected Natural Flavonoids.

scientific article

Magnetic Metal-Organic Framework Composite by Fast and Facile Mechanochemical Process.

scientific article published on 7 February 2018

Natural compounds and extracts as novel antimicrobial agents

scientific article published on 17 November 2020

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation

scientific article published on 01 December 2020

Novel therapies for glaucoma: a patent review (2013-2019)

scientific article published on 11 August 2019

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms.

scientific article

Protective Effects Induced by Microwave-Assisted Aqueous Harpagophytum Extract on Rat Cortex Synaptosomes Challenged with Amyloid β-Peptide

scientific article published on 21 June 2017

Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives.

scientific article published on December 2017

Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma.

scientific article published on 22 October 2015

The Up-Regulation of Oxidative Stress as a Potential Mechanism of Novel MAO-B Inhibitors for Glioblastoma Treatment

scientific article published on 25 May 2019

The sodium salt of the enantiomers of ricobendazole: Preparation, solubility and chiroptical properties.

scientific article published on 20 February 2017