List of works by Kristoffer Sahlholm

A Neanderthal Sodium Channel Increases Pain Sensitivity in Present-Day Humans

scientific article published on 15 July 2020

A truncated Kv1.1 protein in the brain of the megencephaly mouse: expression and interaction

scientific article

Agonist-specific voltage sensitivity at the dopamine D2S receptor--molecular determinants and relevance to therapeutic ligands.

scientific article published on 5 July 2011

Antipsychotic-Like Efficacy of Dopamine D2 Receptor-Biased Ligands is Dependent on Adenosine A2A Receptor Expression

scientific article published on 5 August 2017

Antipsychotics with similar association kinetics at dopamine D receptors differ in extrapyramidal side-effects

scientific article published in Nature Communications

Behavioral control by striatal adenosine A2A -dopamine D2 receptor heteromers

scientific article

Cocaine produces D2R-mediated conformational changes in the adenosine A(2A)R-dopamine D2R heteromer

scientific article

Differential voltage-sensitivity of D2-like dopamine receptors

scientific article published on 22 July 2008

Discovery and biological characterization of a novel scaffold for potent inhibitors of peripheral serotonin synthesis

scientific article published on 05 August 2020

Dopamine D Receptor Agonist Binding Kinetics-Role of a Conserved Serine Residue

scientific article published in 2021

Effects of the Dopamine Stabilizer, Pridopidine, on Basal and Phencyclidine- Induced Locomotion: Role of Dopamine D2 and Sigma-1 Receptors

scientific article published on 01 January 2018

Electrophysiology-based analysis of human histamine H(4) receptor pharmacology using GIRK channel coupling in Xenopus oocytes

scientific article published on 12 June 2008

Evidence for oligomerization between GABAB receptors and GIRK channels containing the GIRK1 and GIRK3 subunits

scientific article published on 16 September 2010

Facilitated Anion Transport Induces Hyperpolarization of the Cell Membrane That Triggers Differentiation and Cell Death in Cancer Stem Cells

scientific article published on 3 December 2015

G protein-gated inwardly rectifying potassium channel subunits 1 and 2 are down-regulated in rat dorsal root ganglion neurons and spinal cord after peripheral axotomy

scientific article published on 22 July 2015

Highly Selective Dopamine D3 Receptor Antagonists with Arylated Diazaspiro Alkane Cores.

scientific article published on 10 November 2017

In Vitro Comparison of Ulotaront (SEP-363856) and Ralmitaront (RO6889450): Two TAAR1 Agonist Candidate Antipsychotics

Ligand with Two Modes of Interaction with the Dopamine D2 Receptor-An Induced-Fit Mechanism of Insurmountable Antagonism

scientific article published on 15 September 2020

Point mutation of a conserved aspartate, D69, in the muscarinic M2 receptor does not modify voltage-sensitive agonist potency

scientific article published on 2 January 2018

Pridopidine Reverses Phencyclidine-Induced Memory Impairment.

scientific article

Pridopidine selectively occupies sigma-1 rather than dopamine D2 receptors at behaviorally active doses

scientific article published on 11 July 2015

Sigma-2 receptor binding is decreased in female, but not male, APP/PS1 mice.

scientific article published on 18 March 2015

The Beta-Arrestin-Biased Dopamine D2 Receptor Ligand, UNC9994, Is a Partial Agonist at G-Protein-Mediated Potassium Channel Activation

article

The dopamine stabilizers ACR16 and (−)-OSU6162 display nanomolar affinities at the σ-1 receptor

scientific article published on 21 February 2012

The fast-off hypothesis revisited: A functional kinetic study of antipsychotic antagonism of the dopamine D2 receptor

scientific article published on 14 January 2016

The human histamine H3 receptor couples to GIRK channels in Xenopus oocytes

scientific article

The role of RGS protein in agonist-dependent relaxation of GIRK currents in Xenopus oocytes

scientific article published on 29 October 2011

The role of beta-arrestin2 in shaping fMRI BOLD responses to dopaminergic stimulation

scientific article

Typical and atypical antipsychotics do not differ markedly in their reversibility of antagonism of the dopamine D2 receptor

scientific article

Voltage sensitivities and deactivation kinetics of histamine H₃ and H₄ receptors

scientific article published on 2 August 2012

Voltage-dependence of the human dopamine D2 receptor

scientific article published in June 2008

Voltage-sensitivity at the human dopamine D2S receptor is agonist-specific

scientific article

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