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List of works by Francesca Bartoccini

A novel one-pot approach of hexahydropyrrolo[2,3-b]indole nucleus by a cascade addition/cyclization strategy: synthesis of (+/-)-esermethole.

scientific article published on September 2010

A simple, modular synthesis of C4-substituted tryptophan derivatives

scientific article published on 01 October 2016

Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin

scientific article published on 06 September 2019

Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist.

scientific article published in August 2010

Direct, regioselective, and chemoselective preparation of novel boronated tryptophans by Friedel-Crafts alkylation

scientific article published on 30 December 2011

Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions.

scientific article

Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen

scientific article published on 26 July 2017

Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position

scientific article published on 17 September 2018

Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives

scientific article published on 20 May 2016

Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands

scientific article published on 07 May 2015

Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease.

scientific article published on 24 June 2013

Synthesis of (-)-epi-indolactam V by an intramolecular Buchwald-Hartwig C-N coupling cyclization reaction.

scientific article published on 25 July 2013

Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors.

scientific article published on 16 January 2013

Synthesis of (±)-cis-clavicipitic acid by a Rh(I)-catalyzed intramolecular imine reaction

scientific article published on 14 March 2014

Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration.

scientific article published on 26 August 2014

Synthesis of benzo[1,2-d;3,4-d']diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists.

scientific article published in August 2007

Synthesis of new C-6 alkyliden penicillin derivatives as beta-lactamase inhibitors.

scientific article

Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation

scientific article published on 05 June 2019