List of works - Gianfabio Giorgioni

1-[3-(4-Butylpiperidin-1-yl)propyl]-1,2,3,4-tetrahydroquinolin-2-one (77-LH-28-1) as a Model for the Rational Design of a Novel Class of Brain Penetrant Ligands with High Affinity and Selectivity for Dopamine D4 Receptor.

scientific article published on 28 March 2018

A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus

scientific article published on 15 March 2016

Chemical–physical properties and cytotoxicity of N -decanoyl amino acid-based surfactants: Effect of polar heads

Correlation among chemical structure, surface properties and cytotoxicity of N-acyl alanine and serine surfactants

scientific article published on 28 September 2016

Cu(I) and Cu(II) Complexes Based on Lonidamine-Conjugated Ligands Designed to Promote Synergistic Antitumor Effects

scientific article published on 14 March 2022

Design, synthesis, and preliminary pharmacological evaluation of new imidazolinones as L-DOPA prodrugs.

scientific article published on 25 January 2010

Dopamine D5 receptors: a challenge to medicinal chemists.

scientific article published on September 2008

Evaluation of P(L)LA-PEG-P(L)LA as processing aid for biodegradable particles from gas saturated solutions (PGSS) process

scientific article published on 18 April 2014

Evaluation of methoxy polyethylene glycol-polylactide diblock copolymers as additive in hypromellose film coating

Evaluation of polymer mucoadhesiveness by the use of acoustic spectroscopy

scientific article

Glycosyl and polyalcoholic prodrugs of lonidamine.

scientific article

Ibuprofen and lipoic acid diamide as co-drug with neuroprotective activity: pharmacological properties and effects in beta-amyloid (1-40) infused Alzheimer's disease rat model.

scientific article published on April 2010

Investigation of the Role of Chirality in the Interaction with σ Receptors and Effect on Binge Eating Episode of a Potent σ1 Antagonist Analogue of Spipethiane

scientific article published on 23 July 2019

Monitoring the aggregation behaviour of self-assembling polymers through high-resolution ultrasonic spectroscopy

scientific article published on 07 January 2010

Multitarget 1,4-Dioxane Compounds Combining Favorable D2-like and 5-HT1A Receptor Interactions with Potential for the Treatment of Parkinson's Disease or Schizophrenia

scientific article published on 09 January 2019

New L-dopa codrugs as potential antiparkinson agents

scientific article published in July 2008

New flurbiprofen derivatives: synthesis, membrane affinity and evaluation of in vitro effect on β-amyloid levels

scientific article published on 3 September 2013

Novel imidazoline compounds as partial or full agonists of D2-like dopamine receptors inspired by I2-imidazoline binding sites ligand 2-BFI.

scientific article published on 6 August 2010

Novel muscarinic acetylcholine receptor hybrid ligands embedding quinuclidine and 1,4-dioxane fragments.

scientific article published on 3 June 2017

Preparation and pharmacological characterization of trans-2-amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes as D2-like dopamine receptor agonists

scientific article published in April 2005

Quaternary Ammonium Leucine-Based Surfactants: The Effect of a Benzyl Group on Physicochemical Properties and Antimicrobial Activity

scientific article published on 19 June 2019

Synthesis and Cytotoxic Activity Evaluation of New Cu(I) Complexes of Bis(pyrazol-1-yl) Acetate Ligands Functionalized with an NMDA Receptor Antagonist

scientific article published on 09 April 2020

Synthesis and biological evaluation of GABA derivatives able to cross the blood–Brain barrier in rats ⬇️

scientific article published on November 3, 2003

Synthesis and preliminary pharmacological evaluation of 5-hydroxy- and 5,6-dihydroxy-1,2,3,7,12,12a-hexahydrobenzo[5,6]cyclohepta[1,2,3-ij]isoquinoline derivatives as dopamine receptor ligands.

scientific article published in June 2001

Synthesis of L-(+)-3-(3-hydroxy-4-pivaloyloxybenzyl)-2,5-diketomorpholine as potential prodrug of L-dopa.

scientific article published in June 2000

Synthesis of novel 4-aryl-1,2,3,4-tetrahydroisoquinolines as probes for dopamine receptor ligands

scientific article published on 01 July 2012

Synthesis, Biological, and Computational Evaluations of Conformationally Restricted NAD-Mimics as Discriminant Inhibitors of Human NMN-Adenylyltransferase Isozymes

scientific article published in 2024

Synthesis, resolution, and preliminary evaluation of trans-2-amino-6(5)-hydroxy-1-phenyl-2,3-dihydro-1H-indenes and related derivatives as dopamine receptors ligands

scientific article published on 01 October 1996

The Versatile 2-Substituted Imidazoline Nucleus as a Structural Motif of Ligands Directed to the Serotonin 5-HT1A Receptor

scientific article published on 30 September 2016

The replacement of the 2-methoxy substituent of N-((6,6-diphenyl-1,4-dioxan-2-yl)methyl)-2-(2-methoxyphenoxy)ethan-1-amine improves the selectivity for 5-HT1A receptor over α1-adrenoceptor and D2-like receptor subtypes

scientific article published on 9 September 2016

Thermosensitive Self-Assembling Block Copolymers as Drug Delivery Systems

Underlying Susceptibility to Eating Disorders and Drug Abuse: Genetic and Pharmacological Aspects of Dopamine D4 Receptors

scientific article published on 30 July 2020

List of works by Gianfabio Giorgioni