List of works by João Neres

2-Carboxyquinoxalines kill mycobacterium tuberculosis through noncovalent inhibition of DprE1

scientific article

Aryl acid adenylating enzymes involved in siderophore biosynthesis: fluorescence polarization assay, ligand specificity, and discovery of non-nucleoside inhibitors via high-throughput screening.

scientific article published on 18 October 2008

Benzoic acid and pyridine derivatives as inhibitors of Trypanosoma cruzi trans-sialidase

scientific article published on 15 December 2006

Biochemical and Structural Characterization of Bisubstrate Inhibitors of BasE, the Self-Standing Nonribosomal Peptide Synthetase Adenylate-Forming Enzyme of Acinetobactin Synthesis,

scientific article

Biological and structural characterization of the Mycobacterium smegmatis nitroreductase NfnB, and its role in benzothiazinone resistance

scientific article

Continuous fluorimetric assay for high-throughput screening of inhibitors of trans-sialidase from Trypanosoma cruzi

scientific article published in October 2006

Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure-activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-D-ribose 2'-oxidase

scientific article

Discovery of novel inhibitors of Trypanosoma cruzi trans-sialidase from in silico screening

scientific article published on 24 December 2008

DprE1--from the discovery to the promising tuberculosis drug target.

scientific article published on January 2014

Inhibition of siderophore biosynthesis by 2-triazole substituted analogues of 5'-O-[N-(salicyl)sulfamoyl]adenosine: antibacterial nucleosides effective against Mycobacterium tuberculosis

scientific article published on December 2008

Inhibition of siderophore biosynthesis in Mycobacterium tuberculosis with nucleoside bisubstrate analogues: structure-activity relationships of the nucleobase domain of 5'-O-[N-(salicyl)sulfamoyl]adenosine

scientific article

Inhibitors of the Salicylate Synthase (MbtI) from Mycobacterium tuberculosis Discovered by High‐Throughput Screening

scientific article published on December 3, 2010

Mechanism of a Standalone β-Lactone Synthetase: New Continuous Assay for a Widespread ANL Superfamily Enzyme

scientific article published on 16 May 2019

Non-nucleoside inhibitors of BasE, an adenylating enzyme in the siderophore biosynthetic pathway of the opportunistic pathogen Acinetobacter baumannii

scientific article published on 13 March 2013

Pyridomycin bridges the NADH- and substrate-binding pockets of the enoyl reductase InhA

scientific article

Rational drug design in parasitology: trans-sialidase as a case study for Chagas disease.

scientific article published on February 2008

Selective detection of epimeric pentose saccharides at physiological pH using a fluorescent receptor

scientific article published on 15 February 2014

Structural Basis for Benzothiazinone-Mediated Killing of Mycobacterium tuberculosis

scientific article

The global virulence regulators VsrAD and PhcA control secondary metabolism in the plant pathogen Ralstonia solanacearum

scientific article published on 01 November 2009

Towards a new combination therapy for tuberculosis with next generation benzothiazinones

scientific article

Towards a new tuberculosis drug: pyridomycin - nature's isoniazid

scientific article

Tryptophan as a molecular shovel in the glycosyl transfer activity of Trypanosoma cruzi trans-sialidase.

scientific article