List of works - Maria Luisa Gelmi

1-Aminocyclopentane-1,2,4-tricarboxylic acids screening on glutamatergic and serotonergic systems

scientific article published on 12 September 2007

1H-Azepine-2-oxo-5-amino-5-carboxylic Acid: A 310 Helix Inducer and an Effective Tool for Functionalized Gold Nanoparticles

scientific article published on 14 May 2015

1H-Azepine-4-amino-4-carboxylic acid: a new α,α-disubstituted ornithine analogue capable of inducing helix conformations in short Ala-Aib pentapeptides

scientific article published on 11 June 2012

A New Synthesis of Functionalized 2-Alkylidenetetrahydro-5-furanones by Tandem Alkylation and Translactonization Reactions of 5(4H)-Oxazolones

scientific article published on 01 March 1996

A Novel Class of Conformationally Constrained, Masked Cysteines: Synthesis of 2-Alkyl- and 2-Arylsulfanyl-1-aminocyclopropanecarboxylic Acids

scientific article published on 01 February 1999

A highly diastereoselective synthesis of new polyhydroxy 2-aminonorbornanecarboxylic acids

scientific article published on 01 July 2001

A highly diastereoselective synthesis of α-hydroxy-β-amino acid derivatives via a Lewis acid catalyzed three-component condensation reaction.

scientific article published on November 2010

A new scaffold of topoisomerase I inhibitors: Design, synthesis and biological evaluation.

scientific article published on 23 August 2016

Alpha,gamma-diamino acids: asymmetric synthesis of new constrained 6-amino-3-azabicyclo[3.2.1]octane-6-carboxylic acids

scientific article published on 01 October 2006

An efficient route to all stereoisomeric enantiopure 6-amino-3-alkyl-3- azabicyclo[3.2.1]octane-6-carboxylic acids.

scientific article published on 8 November 2007

Antiproliferative activity on human prostate carcinoma cell lines of new peptidomimetics containing the spiroazepinoindolinone scaffold

scientific article published on 13 June 2013

Asymmetric Modular Synthesis of a Semirigid Dipeptide Mimetic by Cascade Cycloaddition/Ring Rearrangement and Borohydride Reduction

scientific article published on 25 March 2014

Chemotactic effect of prorenin on human aortic smooth muscle cells: a novel function of the (pro)renin receptor.

scientific article published on 21 June 2012

Construction of ratiometric fluorescent sensors by ribonucleopeptides.

scientific article

Cycloaddition reactions of 2,4-diphenyl-3-methyl-1,3-oxazolium 5-oxide with 4-methylene-4,5-dihydroisoxazoles: 1H and 13C nuclear magnetic resonance stereochemical assignments of the products

Diastereoselective 14beta-hydroxylation of baccatin III derivatives

scientific article

Diastereoselective protocols for the synthesis of 2,3-trans- and 2,3-cis-6-methoxy-morpholine-2-carboxylic acid derivatives

scientific article published on 21 March 2012

Dipeptide Nanotubes Containing Unnatural Fluorine-Substituted β(2,3)-Diarylamino Acid and L-Alanine as Candidates for Biomedical Applications

scientific article published on 03 September 2015

Efforts towards the design of 'teflon' proteins: in vivo translation with trifluorinated leucine and methionine analogues.

scientific article published in October 2004

Expedient chemical synthesis of 75mer DNA binding domain of MafA: an insight on its binding to insulin enhancer

scientific article published on 04 April 2012

Isothiazole dioxides: synthesis and inhibition of Trypanosoma brucei protein farnesyltransferase.

scientific article

Isothiazoles. Part 13: Synthesis of sulfamic esters, [1,2]thiazete S,S-dioxides, benzo[e][1,2]thiazine S,S-dioxides or triazoles by reaction of isothiazole dioxides with sodium azide

MediaChrom: Discovering a Class of Pyrimidoindolone-Based Polarity-Sensitive Dyes

scientific article published on 16 October 2015

Model peptides containing the 3-sulfanyl-norbornene amino acid, a conformationally constrained cysteine analogue effective inducer of 310-helix secondary structures

article

Molecular dynamics and tubulin polymerization kinetics study on 1,14-heterofused taxanes: evidence of stabilization of the tubulin head-to-tail dimer-dimer interaction.

scientific article

Molecular insights into dimerization inhibition of c-Maf transcription factor

scholarly article by Sara Pellegrino published in December 2014

N-Deacetyl-N-aminoacylthiocolchicine Derivatives: Synthesis and Biological Evaluation on MDR-Positive and MDR-Negative Human Cancer Cell Lines

scientific article published on 01 December 1999

New taxane derivatives: synthesis of baccatin[14,1-d]furan-2-one nucleus and its condensation with the norstatine side chain

scientific article published in October 2004

Non-natural 3-Arylmorpholino-β-amino Acid as a PPII Helix Inducer

scientific article published on 30 July 2020

Novel 3-O-glycosyl-3-demethylthiocolchicines as ligands for glycine and gamma-aminobutyric acid receptors.

scientific article

Peptide modulators of Rac1/Tiam1 protein-protein interaction: An alternative approach for cardiovascular diseases.

scientific article published on 27 November 2017

Rational Design of a User-Friendly Aptamer/Peptide-Based Device for the Detection of Staphylococcus aureus

scientific article published on 02 September 2020

Self-assembly of an amphipathic ααβ-tripeptide into cationic spherical particles for intracellular delivery

scientific article published on 01 August 2017

Stabilization of the cysteine-rich conotoxin MrIA by using a 1,2,3-triazole as a disulfide bond mimetic

scientific article published on 5 December 2014

Synthesis, structural, and biological evaluation of bis-heteroarylmaleimides and bis-heterofused imides

scientific article published on 16 August 2011

Synthetic peptides containing a conserved sequence motif of the Id protein family modulate vascular smooth muscle cell phenotype

scientific article published on 01 October 2009

Tandem Tetrahydroisoquinoline-4-carboxylic Acid/β-Alanine as a New Construct Able To Induce a Flexible Turn

scientific article

Tetrahydro-4 H-(pyrrolo[3,4- d]isoxazol-3-yl)methanamine: A Bicyclic Diamino Scaffold Stabilizing Parallel Turn Conformations

scientific article published on 18 September 2018

Unusual chemoselective Rh(II)-catalysed transformations of α-diazocarbonyl piperidine cores

scientific article published on 24 November 2014

β-Hairpin mimics containing a piperidine-pyrrolidine scaffold modulate the β-amyloid aggregation process preserving the monomer species.

scientific article published on 7 October 2016

List of works by Maria Luisa Gelmi

1-Aminocyclopentane-1,2,4-tricarboxylic acids screening on glutamatergic and serotonergic systems

1H-Azepine-2-oxo-5-amino-5-carboxylic Acid: A 310 Helix Inducer and an Effective Tool for Functionalized Gold Nanoparticles

1H-Azepine-4-amino-4-carboxylic acid: a new α,α-disubstituted ornithine analogue capable of inducing helix conformations in short Ala-Aib pentapeptides

A New Synthesis of Functionalized 2-Alkylidenetetrahydro-5-furanones by Tandem Alkylation and Translactonization Reactions of 5(4H)-Oxazolones

A Novel Class of Conformationally Constrained, Masked Cysteines: Synthesis of 2-Alkyl- and 2-Arylsulfanyl-1-aminocyclopropanecarboxylic Acids

A highly diastereoselective synthesis of new polyhydroxy 2-aminonorbornanecarboxylic acids

A highly diastereoselective synthesis of α-hydroxy-β-amino acid derivatives via a Lewis acid catalyzed three-component condensation reaction.

A new scaffold of topoisomerase I inhibitors: Design, synthesis and biological evaluation.

Alpha,gamma-diamino acids: asymmetric synthesis of new constrained 6-amino-3-azabicyclo[3.2.1]octane-6-carboxylic acids

An efficient route to all stereoisomeric enantiopure 6-amino-3-alkyl-3- azabicyclo[3.2.1]octane-6-carboxylic acids.

Antiproliferative activity on human prostate carcinoma cell lines of new peptidomimetics containing the spiroazepinoindolinone scaffold

Asymmetric Modular Synthesis of a Semirigid Dipeptide Mimetic by Cascade Cycloaddition/Ring Rearrangement and Borohydride Reduction

Chemotactic effect of prorenin on human aortic smooth muscle cells: a novel function of the (pro)renin receptor.

Construction of ratiometric fluorescent sensors by ribonucleopeptides.

Cycloaddition reactions of 2,4-diphenyl-3-methyl-1,3-oxazolium 5-oxide with 4-methylene-4,5-dihydroisoxazoles: 1H and 13C nuclear magnetic resonance stereochemical assignments of the products

Diastereoselective 14beta-hydroxylation of baccatin III derivatives

Diastereoselective protocols for the synthesis of 2,3-trans- and 2,3-cis-6-methoxy-morpholine-2-carboxylic acid derivatives

Dipeptide Nanotubes Containing Unnatural Fluorine-Substituted β(2,3)-Diarylamino Acid and L-Alanine as Candidates for Biomedical Applications

Efforts towards the design of 'teflon' proteins: in vivo translation with trifluorinated leucine and methionine analogues.

Expedient chemical synthesis of 75mer DNA binding domain of MafA: an insight on its binding to insulin enhancer

Isothiazole dioxides: synthesis and inhibition of Trypanosoma brucei protein farnesyltransferase.

Isothiazoles. Part 13: Synthesis of sulfamic esters, [1,2]thiazete S,S-dioxides, benzo[e][1,2]thiazine S,S-dioxides or triazoles by reaction of isothiazole dioxides with sodium azide

MediaChrom: Discovering a Class of Pyrimidoindolone-Based Polarity-Sensitive Dyes

Model peptides containing the 3-sulfanyl-norbornene amino acid, a conformationally constrained cysteine analogue effective inducer of 310-helix secondary structures

Molecular dynamics and tubulin polymerization kinetics study on 1,14-heterofused taxanes: evidence of stabilization of the tubulin head-to-tail dimer-dimer interaction.

Molecular insights into dimerization inhibition of c-Maf transcription factor

N-Deacetyl-N-aminoacylthiocolchicine Derivatives: Synthesis and Biological Evaluation on MDR-Positive and MDR-Negative Human Cancer Cell Lines

New taxane derivatives: synthesis of baccatin[14,1-d]furan-2-one nucleus and its condensation with the norstatine side chain

Non-natural 3-Arylmorpholino-β-amino Acid as a PPII Helix Inducer

Novel 3-O-glycosyl-3-demethylthiocolchicines as ligands for glycine and gamma-aminobutyric acid receptors.

Peptide modulators of Rac1/Tiam1 protein-protein interaction: An alternative approach for cardiovascular diseases.

Rational Design of a User-Friendly Aptamer/Peptide-Based Device for the Detection of Staphylococcus aureus

Self-assembly of an amphipathic ααβ-tripeptide into cationic spherical particles for intracellular delivery

Stabilization of the cysteine-rich conotoxin MrIA by using a 1,2,3-triazole as a disulfide bond mimetic

Synthesis, structural, and biological evaluation of bis-heteroarylmaleimides and bis-heterofused imides

Synthetic peptides containing a conserved sequence motif of the Id protein family modulate vascular smooth muscle cell phenotype

Tandem Tetrahydroisoquinoline-4-carboxylic Acid/β-Alanine as a New Construct Able To Induce a Flexible Turn

Tetrahydro-4 H-(pyrrolo[3,4- d]isoxazol-3-yl)methanamine: A Bicyclic Diamino Scaffold Stabilizing Parallel Turn Conformations

Unusual chemoselective Rh(II)-catalysed transformations of α-diazocarbonyl piperidine cores

β-Hairpin mimics containing a piperidine-pyrrolidine scaffold modulate the β-amyloid aggregation process preserving the monomer species.