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List of works by Sebastian Demkowicz

Geometry optimization of steroid sulfatase inhibitors - the influence on the free binding energy with STS

New clicked full agonists of the estrogen receptor β

scholarly article in RSC Advances, vol. 3 no. 11, 2013

New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1<i>H</i>-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives

scientific article published on 01 December 2021

Novel steroid sulfatase inhibitors based on N-thiophosphorylated 3-(4-aminophenyl)-coumarin-7-O-sulfamates

scientific article published on 13 July 2019

Phosphate and thiophosphate biphenyl analogs as steroid sulfatase inhibitors

scientific article published on 01 March 2015

Recent progress in the development of steroid sulphatase inhibitors - examples of the novel and most promising compounds from the last decade

scientific article published on 01 December 2020

Steroid Sulfatase Inhibitors Based on Phosphate and Thiophosphate Flavone Analogs

scientific article published on 28 September 2015

Synthesis and Biological Evaluation of Fluorinated 3-Phenylcoumarin-7-O-Sulfamate Derivatives as Steroid Sulfatase Inhibitors

scientific article published on 14 September 2015

Synthesis and Cholinesterase Inhibitory Activity of N-Phosphorylated / N-Tiophosphorylated Tacrine

scientific article published on 16 July 2019

Synthesis and biological evaluation of N-acylated tyramine sulfamates containing C-F bonds as steroid sulfatase inhibitors.

scientific article

Synthesis and biological evaluation of fluorinated N-benzoyl and N-phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7-O-sulfamate as steroid sulfatase inhibitors.

scientific article published on 22 January 2017

Synthesis and biological evaluation of thiophosphate tricyclic coumarin derivatives as steroid sulfatase inhibitors

scientific article published on 13 August 2015

Synthesis of bicoumarin thiophosphate derivatives as steroid sulfatase inhibitors

scientific article published on 02 July 2015

Taurine as a water structure breaker and protein stabilizer

scientific article published on 17 October 2017

Towards β-selectivity in functional estrogen receptor antagonists

scientific article published on 01 September 2012