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List of works by François Crestey

A small molecule activator of Nav 1.1 channels increases fast-spiking interneuron excitability and GABAergic transmission in vitro and has anti-convulsive effects in vivo.

scientific article published on 21 June 2017

A strategic approach to [6,6]-bicyclic lactones: application towards the CD fragment of DHβE

scientific article

Chemo- and Regioselective Functionalization of Nortrilobolide: Application for Semisynthesis of the Natural Product 2-Acetoxytrilobolide

scientific article published on 16 June 2015

Design, synthesis, and biological evaluation of Erythrina alkaloid analogues as neuronal nicotinic acetylcholine receptor antagonists.

scientific article

Dual Nicotinic Acetylcholine Receptors α4β2 Antagonists/α7 Agonists: Synthesis, Docking Studies and Pharmacological Evaluation of Tetrahydroisoquinolines and Tetrahydroisoquinolinium Salts.

scientific article published on 31 January 2018

Expedite protocol for construction of chiral regioselectively N-protected monosubstituted piperazine, 1,4-diazepane, and 1,4-diazocane building blocks.

scientific article

Identification and electrophysiological evaluation of 2-methylbenzamide derivatives as Nav1.1 modulators

scientific article

Microwave-Assisted Ring-Opening of Activated Aziridines with Resin-Bound Amines

scientific article published on 01 April 2008

Radiosynthesis and preclinical evaluation of [11 C]Cimbi-701 - Towards the imaging of cerebral 5-HT7 receptors

scientific article published on 06 January 2020

Total synthesis of ascididemin via anionic cascade ring closure

scientific article published on 03 August 2012

Trifunctionalization of the purine scaffold using Mg and Zn organometallic intermediates

scientific article published on 19 January 2011

Tying up Nicotine: New Selective Competitive Antagonist of the Neuronal Nicotinic Acetylcholine Receptors.

scientific article published on 4 March 2015

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