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List of works by Danny J Scholten

At-line coupling of LC-MS to bioaffinity and selectivity assessment for metabolic profiling of ligands towards chemokine receptors CXCR1 and CXCR2.

scientific article published on 10 August 2015

C(X)CR in silico: Computer-aided prediction of chemokine receptor-ligand interactions

scientific article published on January 2012

Chemical subtleties in small-molecule modulation of peptide receptor function: the case of CXCR3 biaryl-type ligands

scientific article

Identification of overlapping but differential binding sites for the high-affinity CXCR3 antagonists NBI-74330 and VUF11211.

scientific article published on 30 October 2013

Label-free impedance responses of endogenous and synthetic chemokine receptor CXCR3 agonists correlate with Gi-protein pathway activation.

scientific article

Metabolic profiling of ligands for the chemokine receptor CXCR3 by liquid chromatography-mass spectrometry coupled to bioaffinity assessment

scientific article published on 12 July 2015

Pharmacological characterization of [3H]VUF11211, a novel radiolabeled small-molecule inverse agonist for the chemokine receptor CXCR3

scientific article published on 09 January 2015

Pharmacological characterization of a small‐molecule agonist for the chemokine receptor CXCR3

scientific article published on June 1, 2012

Pharmacological modulation of chemokine receptor function.

scientific article published on March 2012

Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonists

scientific article published on 27 February 2012

Ubiquitination of CXCR7 controls receptor trafficking

scientific article