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List of works by Alessandro Deplano

A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists

scientific article published on 14 May 2014

Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors

scientific article published on 01 December 2019

Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor

scientific article

Design, Synthesis and Evaluation of Antiproliferative Activity of New Benzimidazolehydrazones.

scientific article published on 30 April 2016

Design, synthesis and <i>in vitro</i> and <i>in vivo</i> biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents

scientific article published on 01 December 2021

Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 reverse transcriptase-associated RNase H and RDDP functions.

scientific article published on August 2017

Development and Validation of Molecular Overlays Derived from Three-Dimensional Hydrophobic Similarity with PharmScreen

article

Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen

scientific article published on 01 December 2020

Homology modeling of a Class A GPCR in the inactive conformation: A quantitative analysis of the correlation between model/template sequence identity and model accuracy

scientific article published on 4 October 2016

In vitro nematicidal activity of aryl hydrazones and comparative GC-MS metabolomics analysis

scientific article published on 10 November 2015

Inhibitory effect of positively charged triazine antagonists of prokineticin receptors on the transient receptor vanilloid type-1 (TRPV1) channel.

scientific article published on 17 July 2015

Interaction of the N-(3-Methylpyridin-2-yl)amide Derivatives of Flurbiprofen and Ibuprofen with FAAH: Enantiomeric Selectivity and Binding Mode

scientific article published on 13 November 2015

Novel propanamides as fatty acid amide hydrolase inhibitors.

scientific article published on 12 May 2017

Potent Nematicidal Activity of Maleimide Derivatives on Meloidogyne incognita

scientific article published on 09 June 2016

Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties

scientific article published on 21 July 2015

Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors

scientific article published on 12 August 2019

Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity

scientific article published on 26 July 2015