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List of works by Emilio Lence

A New Pathway for Protein Haptenation by β-Lactams.

scientific article published on 9 August 2017

A selective resin for trans-diequatorial-1,2-diols

Chemical Modification of a Dehydratase Enzyme Involved in Bacterial Virulence by an Ammonium Derivative: Evidence of its Active Site Covalent Adduct

scientific article

Freezing the Dynamic Gap for Selectivity: Motion-Based Design of Inhibitors of the Shikimate Kinase Enzyme.

scientific article published on 4 October 2016

Frontispiece: Freezing the Dynamic Gap for Selectivity: Motion-Based Design of Inhibitors of the Shikimate Kinase Enzyme

Insights into substrate binding and catalysis in bacterial type I dehydroquinase

scientific article

Irreversible covalent modification of type I dehydroquinase with a stable Schiff base

scientific article

Mapping a protein recognition centre with chiral photoactive ligands. An integrated approach combining photophysics, reactivity, proteomics and molecular dynamics simulation studies

scientific article

Mechanistic basis of the inhibition of type II dehydroquinase by (2S)- and (2R)-2-benzyl-3-dehydroquinic acids

scientific article

Mechanistic insight into the reaction catalysed by bacterial type II dehydroquinases

scientific article published on 01 March 2014

Metal-Assisted Ring-Closing/Opening Process of a Chiral Tetrahydroquinazoline

scientific article published on 23 January 2012

Mycobacterium tuberculosis shikimate kinase inhibitors: design and simulation studies of the catalytic turnover

scientific article

Parallel solid-phase synthesis and evaluation of inhibitors of Streptomyces coelicolor type II dehydroquinase

scientific article

Photogeneration of Quinone-Methides as Latent Electrophiles for Lysine-Targeting

QM/MM simulations identify the determinants of catalytic activity differences between type II dehydroquinase enzymes

scientific article published on 01 June 2018

Structural variety of zinc and copper complexes based on a 2,3-disubstituted 1,2,3,4-tetrahydroquinazoline ligand

scientific article published on 27 April 2012

Study of the Phosphoryl-Transfer Mechanism of Shikimate Kinase by NMR Spectroscopy.

scientific article

Targeting the Motion of Shikimate Kinase: Development of Competitive Inhibitors that Stabilize an Inactive Open Conformation of the Enzyme.

scientific article

The conformational rigidity of butane-1,2-diacetals as a powerful synthetic tool

scientific article published on 17 June 2008