List of works - Sebastiano Intagliata

Benzimidazolone-based selective σ2 receptor ligands: Synthesis and pharmacological evaluation

scientific article published on 09 January 2019

Characterization of Sigma 1 Receptor Antagonist CM-304 and Its Analog, AZ-66: Novel Therapeutics Against Allodynia and Induced Pain.

scientific article published on 14 June 2019

Design and synthesis of new homo and hetero bis-piperazinyl-1-propanone derivatives as 5-HT7R selective ligands over 5-HT1AR.

scientific article published on 28 June 2016

Divergent Cytotoxic and Metabolically Stimulative Functions of Sigma-2 Receptors: Structure-Activity Relationships of 6-Acetyl-3-(4-(4-(4-fluorophenyl)piperazin-1-yl)butyl)benzo[d]oxazol-2(3H)-one (SN79) Derivatives

scientific article published on 07 December 2018

Ginseng and heme oxygenase-1: The link between an old herb and a new protective system

scientific article published on 17 October 2019

Heme Oxygenase-2 (HO-2) as a therapeutic target: Activators and inhibitors

scientific article published on 17 September 2019

In Vitro Antioxidant and Anti-Glycation Activity of Resveratrol and Its Novel Triester with Trolox

scientific article published on 24 December 2020

New Arylethanolimidazole Derivatives as HO-1 Inhibitors with Cytotoxicity against MCF-7 Breast Cancer Cells

scientific article published on 11 March 2020

New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies

scientific article published on 27 December 2016

Novel Structural Insight into Inhibitors of Heme Oxygenase-1 (HO-1) by New Imidazole-Based Compounds: Biochemical and In Vitro Anticancer Activity Evaluation

scientific article published on 18 May 2018

Protective Effects of Caffeic Acid Phenethyl Ester (CAPE) and Novel Cape Analogue as Inducers of Heme Oxygenase-1 in Streptozotocin-Induced Type 1 Diabetic Rats

scientific article published on 17 May 2019

Solid Lipid Nanoparticles Loading Idebenone Ester with Pyroglutamic Acid: In Vitro Antioxidant Activity and In Vivo Topical Efficacy

scientific article published on 29 December 2018

Strategies to Improve Resveratrol Systemic and Topical Bioavailability: An Update

scientific article published on 25 July 2019

Structure–Activity Relationships and Therapeutic Potentials of 5-HT7 Receptor Ligands: An Update

scientific article published on 05 June 2018

Structure–activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT7 and 5-HT1A receptor ligands

scientific article published on 07 August 2014

Synthesis and Molecular Modelling Studies of New 1,3-Diaryl-5-Oxo-Proline Derivatives as Endothelin Receptor Ligands

scientific article published on 17 April 2020

Synthesis and binding properties of new long-chain 4-substituted piperazine derivatives as 5-HT₁A and 5-HT₇ receptor ligands

scientific article published on 25 February 2015

Synthesis, in vitro and in silico studies of HO-1 inducers and lung antifibrotic agents

scientific article published on 01 July 2019

Synthesis, in vitro and in vivo characterization of new benzoxazole and benzothiazole-based sigma receptor ligands

scientific article published on 21 April 2019

Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines

scientific article published on 17 September 2018

[1]Benzothieno[3,2-d]pyrimidine derivatives as ligands for the serotonergic 5-HT7 receptor

scientific article published on 10 September 2019

List of works by Sebastiano Intagliata