List of works - Adriana Chilin

1,4,8-trimethylfuro[2,3-H]quinolin-2(1H)-one, a new furocoumarin bioisoster.

scientific article published on May 2004

2,6-Dimethyl-9-methoxy-4H-pyrrolo[3,2,1-ij]quinolin-4-one, a new compound with unusual photosensitizing properties

scientific article published on 01 July 1994

4-Hydroxymethyl- and 4-methoxymethylfuro[2,3-h]quinolin-2(1H)-ones: synthesis and biological properties.

scientific article published in April 2003

4-hydroxymethyl-1,6,8-trimethylfuro[2,3-h]quinolin-2(1H)-one induces mitochondrial dysfunction and apoptosis upon its intracellular oxidation

scientific article published in January 2005

8-Azapsoralen derivatives: isolation and characterization of the furan-side cycloadducts with DNA

scientific article published on 01 February 1994

A novel convenient synthesis of benzoquinazolines

scientific article published on 01 January 2006

Angular furoquinolinones, psoralen analogs: novel antiproliferative agents for skin diseases. Synthesis, biological activity, mechanism of action, and computer-aided studies.

scientific article

Autogrid-based clustering of kinases: selection of representative conformations for docking purposes.

scientific article published on 29 May 2014

Benzoquinazoline derivatives as new agents affecting DNA processing.

scientific article published on 19 December 2010

Cell killing and DNA damage induced in cultured mammalian cells by some tetrahydrobenzopsoralenquinones

scientific article published on 01 January 1999

Coumarin as attractive casein kinase 2 (CK2) inhibitor scaffold: an integrate approach to elucidate the putative binding motif and explain structure-activity relationships

scientific article

DNA damage and biological effects induced by photosensitization with new N(1)-unsubstituted furo[2,3-h]quinolin-2(1H)-ones.

scientific article

DNA damage induced by 4,6,8,9-tetramethyl-2H-furo[2,3-h]quinolin-2-one, a new furocoumarin analog: biological consequences

scientific article published on 01 March 2000

DNA damage induced by 4,6,8,9-tetramethyl-2H-furo[2,3-h]quinolin-2-one, a new furocoumarin analog: photochemical mechanisms

scientific article published on 01 March 2000

Design, synthesis and biological evaluation of novel trimethylangelicin analogues targeting nuclear factor kB (NF-kB).

scientific article published on 31 March 2018

Discovery of biarylaminoquinazolines as novel tubulin polymerization inhibitors

scientific article

Mechanism of action of 4-hydroxymethyl-1,6,8-trimethylfuro[2,3-h]quinolin-2(1H)-one, a very active angular furocoumarin-like sensitizer.

scientific article

New vandetanib analogs: fused tricyclic quinazolines with antiangiogenic potential.

scientific article

New water soluble pyrroloquinoline derivatives as new potential anticancer agents

scientific article

Novel benzoquinoline derivatives via unpredicted condensation of ethyl propiolate and naphthylamines: Synthesis and topoisomerase inhibition activity

scientific article published on 14 September 2016

Pegylated enzyme entrapped in poly(vinyl alcohol) hydrogel for biocatalytic application.

scientific article

Photobiological properties of 1-(3'-hydroxypropyl)-4,6,8-trimethylfur.

scientific article

Photochemical and photobiological studies on furoquinazolines as new psoralen analogs.

scientific article

Psoralen derivatives as inhibitors of NF- $$\upkappa \hbox {B/DNA}$$ κ B/DNA interaction: the critical role of the furan ring

scientific article published on 14 April 2015

Psoralen derivatives as inhibitors of NF-κB/DNA interaction: synthesis, molecular modeling, 3D-QSAR, and biological evaluation

scientific article published on 25 February 2013

Psoralenquinones as a novel class of proteasome inhibitors: design, synthesis and biological evaluation.

scientific article published on 6 April 2011

Pyrazoloquinazoline Tricyclic System as Novel Scaffold to Design New Kinase CK2 Inhibitors

Pyrrolocoumarin derivatives: DNA-binding properties

scientific article published on 01 December 1988

Pyrroloquinolinone-based dual topoisomerase I/II inhibitor

scientific article published on March 2014

Quinazoline derivatives as potential anticancer agents: a patent review (2007 - 2010).

scientific article published on 12 March 2012

Quinazoline-based multi-tyrosine kinase inhibitors: synthesis, modeling, antitumor and antiangiogenic properties.

scientific article published on 6 July 2013

Synthesis and antitumor activity of novel amsacrine analogs: the critical role of the acridine moiety in determining their biological activity

scientific article

Synthesis and biological activity of (hydroxymethyl)- and (diethylaminomethyl)benzopsoralens

scientific article published on 01 July 1999

Synthesis and biological evaluation of a new furo[2,3-h]quinolin-2(1H)-one.

scientific article published in February 2002

The Importance of Descriptor-Based Clusterization in QSAR Models Development: Tyrosine Kinases Inhibitors as a Key Study.

scientific article published on 2 August 2011

Using the TOPS-MODE approach to fit multi-target QSAR models for tyrosine kinases inhibitors

scientific article published on 11 March 2011

List of works by Adriana Chilin

1,4,8-trimethylfuro[2,3-H]quinolin-2(1H)-one, a new furocoumarin bioisoster.

2,6-Dimethyl-9-methoxy-4H-pyrrolo[3,2,1-ij]quinolin-4-one, a new compound with unusual photosensitizing properties

4-Hydroxymethyl- and 4-methoxymethylfuro[2,3-h]quinolin-2(1H)-ones: synthesis and biological properties.

4-hydroxymethyl-1,6,8-trimethylfuro[2,3-h]quinolin-2(1H)-one induces mitochondrial dysfunction and apoptosis upon its intracellular oxidation

8-Azapsoralen derivatives: isolation and characterization of the furan-side cycloadducts with DNA

A novel convenient synthesis of benzoquinazolines

Angular furoquinolinones, psoralen analogs: novel antiproliferative agents for skin diseases. Synthesis, biological activity, mechanism of action, and computer-aided studies.

Autogrid-based clustering of kinases: selection of representative conformations for docking purposes.

Benzoquinazoline derivatives as new agents affecting DNA processing.

Cell killing and DNA damage induced in cultured mammalian cells by some tetrahydrobenzopsoralenquinones

Coumarin as attractive casein kinase 2 (CK2) inhibitor scaffold: an integrate approach to elucidate the putative binding motif and explain structure-activity relationships

DNA damage and biological effects induced by photosensitization with new N(1)-unsubstituted furo[2,3-h]quinolin-2(1H)-ones.

DNA damage induced by 4,6,8,9-tetramethyl-2H-furo[2,3-h]quinolin-2-one, a new furocoumarin analog: biological consequences

DNA damage induced by 4,6,8,9-tetramethyl-2H-furo[2,3-h]quinolin-2-one, a new furocoumarin analog: photochemical mechanisms

Design, synthesis and biological evaluation of novel trimethylangelicin analogues targeting nuclear factor kB (NF-kB).

Discovery of biarylaminoquinazolines as novel tubulin polymerization inhibitors

Mechanism of action of 4-hydroxymethyl-1,6,8-trimethylfuro[2,3-h]quinolin-2(1H)-one, a very active angular furocoumarin-like sensitizer.

New vandetanib analogs: fused tricyclic quinazolines with antiangiogenic potential.

New water soluble pyrroloquinoline derivatives as new potential anticancer agents

Novel benzoquinoline derivatives via unpredicted condensation of ethyl propiolate and naphthylamines: Synthesis and topoisomerase inhibition activity

Pegylated enzyme entrapped in poly(vinyl alcohol) hydrogel for biocatalytic application.

Photobiological properties of 1-(3'-hydroxypropyl)-4,6,8-trimethylfur.

Photochemical and photobiological studies on furoquinazolines as new psoralen analogs.

Psoralen derivatives as inhibitors of NF- $$\upkappa \hbox {B/DNA}$$ κ B/DNA interaction: the critical role of the furan ring

Psoralen derivatives as inhibitors of NF-κB/DNA interaction: synthesis, molecular modeling, 3D-QSAR, and biological evaluation

Psoralenquinones as a novel class of proteasome inhibitors: design, synthesis and biological evaluation.

Pyrazoloquinazoline Tricyclic System as Novel Scaffold to Design New Kinase CK2 Inhibitors

Pyrrolocoumarin derivatives: DNA-binding properties

Pyrroloquinolinone-based dual topoisomerase I/II inhibitor

Quinazoline derivatives as potential anticancer agents: a patent review (2007 - 2010).

Quinazoline-based multi-tyrosine kinase inhibitors: synthesis, modeling, antitumor and antiangiogenic properties.

Synthesis and antitumor activity of novel amsacrine analogs: the critical role of the acridine moiety in determining their biological activity

Synthesis and biological activity of (hydroxymethyl)- and (diethylaminomethyl)benzopsoralens

Synthesis and biological evaluation of a new furo[2,3-h]quinolin-2(1H)-one.

The Importance of Descriptor-Based Clusterization in QSAR Models Development: Tyrosine Kinases Inhibitors as a Key Study.

Using the TOPS-MODE approach to fit multi-target QSAR models for tyrosine kinases inhibitors