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List of works by Simone Bertini

1,2-Dihydro-2-oxopyridine-3-carboxamides: The C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor

scientific article published on 21 January 2014

4-[6-(Dansylamino)hexylamino]-7-methyl-2-phenyl-1,8-naphthyridine as a new potential fluorescent probe for studying A1-adenosine receptor

scientific article published in October 2002

7-Nitrobenzofurazan (NBD) derivatives of 5'-N-ethylcarboxamidoadenosine (NECA) as new fluorescent probes for human A(3) adenosine receptors.

scientific article published in December 2001

A comparative kinetic study of thiamphenicol in pre-ruminant lambs and calves.

scientific article published in December 2002

A theoretical study to investigate D2DAR/D4DAR selectivity: receptor modeling and molecular docking of dopaminergic ligands.

scientific article published in February 2006

Antiproliferative activity and cell cycle analysis of 2-(3,5-dihydroxyphenyl)-6-hydroxybenzothiazole on MCF-7 breast and HCT-15 colon cancer cell lines

scientific article published on 25 March 2011

Application of An Improved HPLC-FL Method to Screen Serine Palmitoyl Transferase Inhibitors

BACE1 inhibitory activities of enantiomerically pure, variously substituted N-(3-(4-benzhydrylpiperazin-1-yl)-2-hydroxypropyl) arylsulfonamides

scientific article published on 18 September 2010

Benzodiazepine poisoning in companion animals.

scientific article

CB2-selective cannabinoid receptor ligands: synthesis, pharmacological evaluation, and molecular modeling investigation of 1,8-Naphthyridin-2(1H)-one-3-carboxamides

scientific article

Carbazole-containing arylcarboxamides as BACE1 inhibitors

scientific article published on 21 September 2011

Ceramide analogues in apoptosis: a new strategy for anticancer drug development.

scientific article

Comparative bioavailability of two sustained-release theophylline formulations in the dog

scientific article published on 01 December 1998

Comparison of HPLC and GC-MS methods for determination of embutramide (a component of Tanax or T-61) in biological specimens.

scientific article

Conformationally restrained ceramide analogues: effects of lipophilic modifications on the antiproliferative activity.

scientific article published in January 2003

Design, synthesis and preliminary evaluation of 18F-labelled 1,8-naphthyridin- and quinolin-2-one-3-carboxamide derivatives for PET imaging of CB2 cannabinoid receptor

scientific article published on 25 April 2015

Determination of ochratoxin A in tissues of wild boar (Sus scrofa L.) by enzymatic digestion (ED) coupled to high-performance liquid chromatography with a fluorescence detector (HPLC-FLD).

scientific article

Development of an HPLC/UV assay for the evaluation of inhibitors of human recombinant monoacylglycerol lipase.

scientific article

Diazoxide attenuates indomethacin-induced small intestinal damage in the rat

scientific article published on 13 October 2010

Doxycycline levels and anti-Wolbachia antibodies in sera from dogs experimentally infected with Dirofilaria immitis and treated with a combination of ivermectin/doxycycline

scientific article published on 28 February 2015

Effects of beta3-adrenoceptor agonist SR 58611A on gastric acid secretion and histamine release in the dog: comparison with ritodrine.

scientific article published in October 1998

Effects of cannabinoid receptor agonists on rat gastric acid secretion: discrepancy between in vitro and in vivo data.

scientific article

Effects of histamine H4 receptor ligands in a mouse model of gastric ulceration.

scientific article

Effects of nonselective and selective cyclooxygenase inhibitors on small intestinal motility in the horse.

scientific article published on 18 June 2008

Effects of oral curcumin on indomethacin-induced small intestinal damage in the rat.

scientific article published on April 2009

Enrofloxacin-theophylline interaction: influence of enrofloxacin on theophylline steady-state pharmacokinetics in the beagle dog

scientific article published on 01 October 1995

Estrogen receptor ligands: a patent review update

scientific article

Gastric antisecretory effects of compound BP 2-94: a histamine H3-receptor agonist prodrug

scientific article published on 01 December 1999

Heavy Metals in the Muscle and Hepatopancreas of Red Swamp Crayfish (<i>Procambarus clarkii</i>) in Campania (Italy)

scientific article published on 29 June 2021

Highly selective salicylketoxime-based estrogen receptor β agonists display antiproliferative activities in a glioma model

scientific article

Inhibition of motility in isolated horse small intestine is mediated by κ but not µ opioid receptors.

scientific article published on 23 August 2011

Intestinal effects of nonselective and selective cyclooxygenase inhibitors in the rat

scientific article published on 16 September 2006

Lead and copper in hunted wild boars and radiographic evaluation of bullet fragmentation between ammunitions

scientific article published on 28 March 2019

Metabolically labile cannabinoid esters: A ‘soft drug’ approach for the development of cannabinoid-based therapeutic drugs

scientific article published on 20 June 2007

Modulation of pentagastrin-induced histamine release by histamine H3 receptors in the dog

scientific article published on 01 July 1996

Monoaryl-substituted salicylaldoximes as ligands for estrogen receptor beta

scientific article published on 13 February 2008

New quinolone- and 1,8-naphthyridine-3-carboxamides as selective CB2 receptor agonists with anticancer and immuno-modulatory activity

scientific article published on 24 April 2015

Oral single-dose pharmacokinetics of thiamphenicol in the sea-bass (Dicentrarchus labrax)

scientific article published on 01 February 2000

Oxime-based inhibitors of glucose transporter 1 displaying antiproliferative effects in cancer cells.

scientific article published on 28 September 2013

Pharmacokinetics of enrofloxacin and its metabolite ciprofloxacin after intravenous and intramuscular administrations in sheep.

scientific article published in July 1996

Pharmacological characterization of muscarinic receptors in the contractions of isolated bronchi in the horse

scientific article published on 07 March 2014

Pharmacological evidence for beta3 adrenoceptors in the control of rat gastric acid secretion

scientific article published in February 2003

Phosphonomethylphosphorylmethyl(oxy)-analogues of geranylgeranyl diphosphate as stable and selective geranylgeranyl protein transferase inhibitors

Positive Allosteric Modulation of CB1 and CB2 Cannabinoid Receptors Enhances the Neuroprotective Activity of a Dual CB1R/CB2R Orthosteric Agonist

scientific article published on 08 December 2020

Protective effects of proton pump inhibitors against indomethacin-induced lesions in the rat small intestine

scientific article published on 07 December 2006

Rational design, synthesis and anti-proliferative properties of new CB2 selective cannabinoid receptor ligands: an investigation of the 1,8-naphthyridin-2(1H)-one scaffold.

scientific article

Regulation of gastric acid secretion by histamine H3 receptors in the dog: an investigation into the site of action

scientific article published on 01 August 1994

Rifaximin is an effective alternative to metronidazole for the treatment of chronic enteropathy in dogs: a randomised trial.

scientific article

Role of muscarinic receptors in the contraction of jejunal smooth muscle in the horse: An in vitro study

scientific article published on 11 July 2017

Salicylaldoxime derivatives as new leads for the development of carbonic anhydrase inhibitors.

scientific article

Salicylaldoxime moiety as a phenolic "A-Ring" substitute in estrogen receptor ligands.

scientific article published in November 2001

Selective and potent agonists for estrogen receptor beta derived from molecular refinements of salicylaldoximes.

scientific article

Short communication: Alteration in blood parameters by enrofloxacin in juvenile lesser spotted dogfish (Scyliorhinus canicula, Linnaeus, 1758) after intramuscular injection

scientific article published on 10 August 2017

Sildenafil improves clinical signs and radiographic features in dogs with congenital idiopathic megaoesophagus: a randomised controlled trial.

scientific article published on 10 February 2017

Stable analogues of geranylgeranyl diphosphate possessing improved geranylgeranyl versus farnesyl protein transferase inhibitory selectivity.

scientific article

Stable propylphosphonic acid analogues of geranylgeranyl diphosphate possessing inhibitory activity on geranylgeranyl protein transferase

scientific article published in November 2004

Structural evolutions of salicylaldoximes as selective agonists for estrogen receptor beta

scientific article

Study of apoptosis induction and deoxycytidine kinase/cytidine deaminase modulation in the synergistic interaction of a novel ceramide analog and gemcitabine in pancreatic cancer cells.

scientific article published on June 2010

Synthesis and antiviral properties of novel analogues of monophosphate and diphosphate bioactive forms of acyclovir.

scientific article published in April 2000

Synthesis of Anthranylaldoxime Derivatives as Estrogen Receptor Ligands and Computational Prediction of Binding Modes

scientific article published on 01 August 2006

Synthesis of Stable Analogues of Geranylgeranyl Diphosphate Possessing a (Z,E,E)-Geranylgeranyl Side Chain, Docking Analysis, and Biological Assays for Prenyl Protein Transferase Inhibition

scientific article published on 01 February 2006

Synthesis of a resveratrol analogue with high ceramide-mediated proapoptotic activity on human breast cancer cells

scientific article published on November 2005

Synthesis of aniline-type analogues of farnesyl diphosphate and their biological assays for prenyl protein transferase inhibitory activity

scientific article published in December 2003

Synthesis of heterocycle-based analogs of resveratrol and their antitumor and vasorelaxing properties

scientific article published on 2 August 2010

Synthesis, antifungal activity, and molecular modeling studies of new inverted oxime ethers of oxiconazole

scientific article published in October 2002

Synthesis, antiinflammatory activity and platelet antiaggregating activity of a new series of beta-aminoxypropionic acids

scientific article published on 01 February 1995

Synthesis, biological activity and molecular modeling of new biphenylic carboxamides as potent and selective CB2 receptor ligands

scientific article published on 02 December 2014

The effect of ethanol, beer, and wine on histamine release from the dog stomach

scientific article published on 01 November 1996

The plasma kinetics and tissue distribution of enrofloxacin and its metabolite ciprofloxacin in the Muscovy duck.

scientific article published in February 1997

Traditional Uses of Cannabinoids and New Perspectives in the Treatment of Multiple Sclerosis

alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors

scientific article

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