List of works - Anthony G Coyne

Asymmetric electrocyclic reactions

scientific article published on 12 May 2011

Correction to Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors

scientific article published on 22 July 2020

Corrigendum: Substrate Fragmentation for the Design of M. tuberculosis CYP121 Inhibitors

scientific article published on 19 December 2016

Covalent inactivation of Mycobacterium thermoresistibile inosine-5'-monophosphate dehydrogenase (IMPDH)

scientific article published on 09 November 2019

Development of Inhibitors against Mycobacterium abscessus tRNA (m1G37) Methyltransferase (TrmD) Using Fragment-Based Approaches

scientific article published on 19 July 2019

Drugging challenging targets using fragment-based approaches

scientific article

Effect of DMSO on Protein Structure and Interactions Assessed by Collision-Induced Dissociation and Unfolding

scientific article published on 13 August 2017

Fragment Profiling Approach to Inhibitors of the Orphan M. tuberculosis P450 CYP144A1.

scientific article published on 7 February 2017

Fragment Screening against the EthR-DNA Interaction by Native Mass Spectrometry.

scientific article published on 17 May 2017

Fragment-Based Approach to Targeting Inosine-5'-monophosphate Dehydrogenase (IMPDH) from Mycobacterium tuberculosis.

scientific article

Fragment-Based Approaches to the Development of Mycobacterium tuberculosis CYP121 Inhibitors

scientific article published on 22 March 2016

Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors

scientific article published on 02 April 2020

Fragment-based approaches in drug discovery and chemical biology

scientific article

Fragment-based approaches to TB drugs

scientific article published on 2 November 2016

Inhibiting Mycobacterium tuberculosis CoaBC by targeting an allosteric site

scientific article published on 08 January 2021

Organic synthesis reactions on-water at the organic-liquid water interface

scientific article

Overcoming the Limitations of Fragment Merging: Rescuing a Strained Merged Fragment Series TargetingMycobacterium tuberculosisCYP121

scientific article

Regioselective conversion of arenes to N-aryl-1,2,3-triazoles using C-H borylation

scientific article published on 22 July 2014

Small-molecule inhibitors that target protein-protein interactions in the RAD51 family of recombinases

scientific article

Spirooxindoles as novel 3D-fragment scaffolds: Synthesis and screening against CYP121 from M. tuberculosis

scientific article

Structural insights into the EthR-DNA interaction using native mass spectrometry.

scientific article published on 13 March 2017

Substrate Fragmentation for the Design of M. tuberculosis CYP121 Inhibitors.

scientific article published on 19 July 2016

Targeting of Fumarate Hydratase from Mycobacterium tuberculosis Using Allosteric Inhibitors with a Dimeric-Binding Mode

scientific article published on 27 September 2019

The Application of HETPHOX Ligands to the Intramolecular Asymmetric Heck Reaction

The influence of water on the rates of 1,3-dipolar cycloaddition reactions: trigger points for exponential rate increases in water-organic solvent mixtures. Water-super versus water-normal dipolarophiles

scientific article published in September 2004

Trapping of palindromic ligands within native transthyretin prevents amyloid formation

scientific article

Understanding "on-water" catalysis of organic reactions. Effects of H+ and Li+ ions in the aqueous phase and nonreacting competitor H-bond acceptors in the organic phase: on H2O versus on D2O for Huisgen cycloadditions

scientific article published on 26 January 2015

Water and organic synthesis: a focus on the in-water and on-water border. Reversal of the in-water Breslow hydrophobic enhancement of the normal endo-effect on crossing to on-water conditions for Huisgen cycloadditions with increasingly insoluble or

scientific article published on 6 March 2013

Water: nature's reaction enforcer--comparative effects for organic synthesis "in-water" and "on-water".

scientific article published on October 2010

List of works by Anthony G Coyne

Asymmetric electrocyclic reactions

Correction to Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors

Corrigendum: Substrate Fragmentation for the Design of M. tuberculosis CYP121 Inhibitors

Covalent inactivation of Mycobacterium thermoresistibile inosine-5'-monophosphate dehydrogenase (IMPDH)

Development of Inhibitors against Mycobacterium abscessus tRNA (m1G37) Methyltransferase (TrmD) Using Fragment-Based Approaches

Drugging challenging targets using fragment-based approaches

Effect of DMSO on Protein Structure and Interactions Assessed by Collision-Induced Dissociation and Unfolding

Fragment Profiling Approach to Inhibitors of the Orphan M. tuberculosis P450 CYP144A1.

Fragment Screening against the EthR-DNA Interaction by Native Mass Spectrometry.

Fragment-Based Approach to Targeting Inosine-5'-monophosphate Dehydrogenase (IMPDH) from Mycobacterium tuberculosis.

Fragment-Based Approaches to the Development of Mycobacterium tuberculosis CYP121 Inhibitors

Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors

Fragment-based approaches in drug discovery and chemical biology

Fragment-based approaches to TB drugs

Inhibiting Mycobacterium tuberculosis CoaBC by targeting an allosteric site

Organic synthesis reactions on-water at the organic-liquid water interface

Overcoming the Limitations of Fragment Merging: Rescuing a Strained Merged Fragment Series TargetingMycobacterium tuberculosisCYP121

Regioselective conversion of arenes to N-aryl-1,2,3-triazoles using C-H borylation

Small-molecule inhibitors that target protein-protein interactions in the RAD51 family of recombinases

Spirooxindoles as novel 3D-fragment scaffolds: Synthesis and screening against CYP121 from M. tuberculosis

Structural insights into the EthR-DNA interaction using native mass spectrometry.

Substrate Fragmentation for the Design of M. tuberculosis CYP121 Inhibitors.

Targeting of Fumarate Hydratase from Mycobacterium tuberculosis Using Allosteric Inhibitors with a Dimeric-Binding Mode

The Application of HETPHOX Ligands to the Intramolecular Asymmetric Heck Reaction

The influence of water on the rates of 1,3-dipolar cycloaddition reactions: trigger points for exponential rate increases in water-organic solvent mixtures. Water-super versus water-normal dipolarophiles

Trapping of palindromic ligands within native transthyretin prevents amyloid formation

Understanding "on-water" catalysis of organic reactions. Effects of H+ and Li+ ions in the aqueous phase and nonreacting competitor H-bond acceptors in the organic phase: on H2O versus on D2O for Huisgen cycloadditions

Water and organic synthesis: a focus on the in-water and on-water border. Reversal of the in-water Breslow hydrophobic enhancement of the normal endo-effect on crossing to on-water conditions for Huisgen cycloadditions with increasingly insoluble or

Water: nature's reaction enforcer--comparative effects for organic synthesis "in-water" and "on-water".