List of works - Constantinos G Neochoritis

1,4,5-Trisubstituted Imidazole-Based p53-MDM2/MDMX Antagonists with Aliphatic Linkers for Conjugation with Biological Carriers.

scientific article

1,5-Benzoxazepines vs 1,5-benzodiazepines. one-pot microwave-assisted synthesis and evaluation for antioxidant activity and lipid peroxidation inhibition

scientific article published on 04 November 2010

2,30-Bis(10H-indole) heterocycles: New p53/MDM2/MDMX antagonists

scientific article

A fluorinated indole-based MDM2 antagonist selectively inhibits the growth of p53wt osteosarcoma cells

scientific article published on 16 February 2019

Application of Silver Nanoparticles in the Multicomponent Reaction Domain: A Combined Catalytic Reduction Methodology to Efficiently Access Potential Hypertension or Inflammation Inhibitors

Artificial Macrocycles as Potent p53-MDM2 Inhibitors.

scientific article published on 20 September 2017

Atorvastatin (Lipitor) by MCR

scientific article published on 07 February 2019

Design of a novel thiophene inhibitor of 15-lipoxygenase-1 with both anti-inflammatory and neuroprotective properties

scientific article published on 09 July 2016

Design of indole- and MCR-based macrocycles as p53-MDM2 antagonists

scientific article published on 20 February 2019

Discovery of chromenes as inhibitors of macrophage migration inhibitory factor.

scientific article published on 24 December 2017

Efficient isocyanide-less isocyanide-based multicomponent reactions

scientific article

Glycoconjugates via phosphorus ylides

scientific article published on 03 May 2019

Hitting on the move: Targeting intrinsically disordered protein states of the MDM2-p53 interaction

scientific article published on 06 August 2019

How To Design a Successful p53-MDM2/X Interaction Inhibitor: A Thorough Overview Based on Crystal Structures.

scientific article published on 16 December 2015

Isocyanide-Based Multicomponent Reactions of Free Phenylboronic Acids

scientific article published on 22 September 2019

Isocyanides as Influenza A Virus Subtype H5N1 Wild-Type M2 Channel Inhibitors

scientific article published on 7 September 2015

Leuckart-Wallach Route Toward Isocyanides and Some Applications

scientific article published on 10 August 2015

Multicomponent Peptide Stapling as a Diversity-Driven Tool for the Development of Inhibitors of Protein-Protein Interactions

scientific article published on 06 February 2020

One-pot microwave assisted synthesis of new 2-alkoxycarbonylmethylene-4-oxo-1,5-benzo-, naphtho-, and pyridodiazepines and assessment of their cytogenetic activity

scientific article published on 25 June 2013

One-pot microwave assisted synthesis under green chemistry conditions, antioxidant screening, and cytotoxicity assessments of benzimidazole Schiff bases and pyrimido[1,2-a]benzimidazol-3(4H)-ones.

scientific article published on 19 November 2010

Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination

scientific article published on 12 December 2019

Rapid approach to complex boronic acids

scientific article published on 05 July 2019

Rational Development of a Potent 15-Lipoxygenase-1 Inhibitor with in Vitro and ex Vivo Anti-inflammatory Properties

scientific article published on 2 September 2015

Rational design and synthesis of 1,5-disubstituted tetrazoles as potent inhibitors of the MDM2-p53 interaction.

scientific article published on 16 November 2016

Scaffold hopping via ANCHOR.QUERY: β-lactams as potent p53-MDM2 antagonists†.

scientific article published on 15 March 2017

Structure and Reactivity of Glycosyl Isocyanides

scientific article published on 10 January 2019

Synthesis of 2-keto-imidazoles utilizing N-arylamino-substituted N-heterocyclic carbenes

scientific article published on 20 January 2011

Tetrazoles via Multicomponent Reactions

scientific article published on 01 February 2019

Towards a facile and convenient synthesis of highly functionalized indole derivatives based on multi-component reactions.

scientific article published on March 2014

Versatile Multicomponent Reaction Macrocycle Synthesis Using α-Isocyano-ω-carboxylic Acids

scientific article published on 6 October 2015

List of works by Constantinos G Neochoritis

1,4,5-Trisubstituted Imidazole-Based p53-MDM2/MDMX Antagonists with Aliphatic Linkers for Conjugation with Biological Carriers.

1,5-Benzoxazepines vs 1,5-benzodiazepines. one-pot microwave-assisted synthesis and evaluation for antioxidant activity and lipid peroxidation inhibition

2,30-Bis(10H-indole) heterocycles: New p53/MDM2/MDMX antagonists

A fluorinated indole-based MDM2 antagonist selectively inhibits the growth of p53wt osteosarcoma cells

Application of Silver Nanoparticles in the Multicomponent Reaction Domain: A Combined Catalytic Reduction Methodology to Efficiently Access Potential Hypertension or Inflammation Inhibitors

Artificial Macrocycles as Potent p53-MDM2 Inhibitors.

Atorvastatin (Lipitor) by MCR

Design of a novel thiophene inhibitor of 15-lipoxygenase-1 with both anti-inflammatory and neuroprotective properties

Design of indole- and MCR-based macrocycles as p53-MDM2 antagonists

Discovery of chromenes as inhibitors of macrophage migration inhibitory factor.

Efficient isocyanide-less isocyanide-based multicomponent reactions

Glycoconjugates via phosphorus ylides

Hitting on the move: Targeting intrinsically disordered protein states of the MDM2-p53 interaction

How To Design a Successful p53-MDM2/X Interaction Inhibitor: A Thorough Overview Based on Crystal Structures.

Isocyanide-Based Multicomponent Reactions of Free Phenylboronic Acids

Isocyanides as Influenza A Virus Subtype H5N1 Wild-Type M2 Channel Inhibitors

Leuckart-Wallach Route Toward Isocyanides and Some Applications

Multicomponent Peptide Stapling as a Diversity-Driven Tool for the Development of Inhibitors of Protein-Protein Interactions

One-pot microwave assisted synthesis of new 2-alkoxycarbonylmethylene-4-oxo-1,5-benzo-, naphtho-, and pyridodiazepines and assessment of their cytogenetic activity

One-pot microwave assisted synthesis under green chemistry conditions, antioxidant screening, and cytotoxicity assessments of benzimidazole Schiff bases and pyrimido[1,2-a]benzimidazol-3(4H)-ones.

Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination

Rapid approach to complex boronic acids

Rational Development of a Potent 15-Lipoxygenase-1 Inhibitor with in Vitro and ex Vivo Anti-inflammatory Properties

Rational design and synthesis of 1,5-disubstituted tetrazoles as potent inhibitors of the MDM2-p53 interaction.

Scaffold hopping via ANCHOR.QUERY: β-lactams as potent p53-MDM2 antagonists†.

Structure and Reactivity of Glycosyl Isocyanides

Synthesis of 2-keto-imidazoles utilizing N-arylamino-substituted N-heterocyclic carbenes

Tetrazoles via Multicomponent Reactions

Towards a facile and convenient synthesis of highly functionalized indole derivatives based on multi-component reactions.

Versatile Multicomponent Reaction Macrocycle Synthesis Using α-Isocyano-ω-carboxylic Acids