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List of works by Samuele Maramai

(S)-2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements, Structural and Biological Investigation

scientific article published on 16 February 2018

A stereoselective approach to peptidomimetic BACE1 inhibitors.

scientific article published on 6 October 2013

Activation of the Wnt Pathway by Small Peptides: Rational Design, Synthesis and Biological Evaluation.

scientific article published on 13 November 2017

Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain

scientific article

Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain

scholarly article by Margherita Brindisi et al published 30 August 2018 in ChemMedChem

Development of a practical and scalable route for the preparation of the deacetoxytubuvaline (dTuv) fragment of pretubulysin and analogs

Development of novel cyclic peptides as pro-apoptotic agents

scientific article published on 5 April 2016

Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases

scientific article published on 26 July 2012

Disease-modifying anti-Alzheimer's drugs: inhibitors of human cholinesterases interfering with β-amyloid aggregation.

scientific article

Dopamine D3 Receptor Antagonists as Potential Therapeutics for the Treatment of Neurological Diseases

scientific article

Harnessing the pyrroloquinoxaline scaffold for FAAH and MAGL interaction: definition of the structural determinants for enzyme inhibition

scholarly article in RSC Advances, vol. 6 no. 69, 2016

Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties

scientific article published on 22 November 2012

Multifunctional cholinesterase and amyloid Beta fibrillization modulators. Synthesis and biological investigation

scientific article

Multitarget Therapeutic Strategies for Alzheimer's Disease: Review on Emerging Target Combinations

scientific article published on 30 June 2020

Phenylpyrrole-based HDAC inhibitors: synthesis, molecular modeling and biological studies

scientific article published on 24 August 2016

Selective kainate receptor (GluK1) ligands structurally based upon 1H-cyclopentapyrimidin-2,4(1H,3H)-dione: synthesis, molecular modeling, and pharmacological and biostructural characterization

scientific article

Subtype Selective γ-Aminobutyric Acid Type A Receptor (GABAAR) Modulators Acting at the Benzodiazepine Binding Site: An Update

scientific article published on 05 December 2019

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