Search filters

List of works by Rink-Jan Lohman

A regulatory role for protease-activated receptor-2 in motivational learning in rats.

scientific article published on 4 May 2009

An HDAC6 Inhibitor Confers Protection and Selectively Inhibits B-Cell Infiltration in DSS-Induced Colitis in Mice.

scientific article published on 8 November 2016

An antagonist of human protease activated receptor-2 attenuates PAR2 signaling, macrophage activation, mast cell degranulation, and collagen-induced arthritis in rats

scientific article published on 30 March 2012

Antagonism of Protease-Activated Receptor 2 Protects against Experimental Colitis

scientific article published on 25 October 2011

Antagonism of the proinflammatory and pronociceptive actions of canonical and biased agonists of protease-activated receptor-2.

scientific article published on 16 July 2016

Benzylamide antagonists of protease activated receptor 2 with anti-inflammatory activity.

scientific article published on 17 December 2015

Cyclic Penta- and Hexaleucine Peptides without N-Methylation Are Orally Absorbed

scientific article

Diet-induced obesity, adipose inflammation, and metabolic dysfunction correlating with PAR2 expression are attenuated by PAR2 antagonism

scientific article

Differential Anti-inflammatory Activity of HDAC Inhibitors in Human Macrophages and Rat Arthritis

scientific article published on 10 December 2015

Flexibility versus Rigidity for Orally Bioavailable Cyclic Hexapeptides

scientific article published on 07 October 2015

Helix-constrained nociceptin peptides are potent agonists and antagonists of ORL-1 and nociception.

scientific article

Improving on Nature: Making a Cyclic Heptapeptide Orally Bioavailable

scientific article published on 12 September 2014

Minocycline Prevents the Development of Mechanical Allodynia in Mouse Models of Vincristine-Induced Peripheral Neuropathy

scientific article published on 27 June 2019

Mirror image pairs of cyclic hexapeptides have different oral bioavailabilities and metabolic stabilities

scientific article published on 21 October 2019

Modulating human proteinase activated receptor 2 with a novel antagonist (GB88) and agonist (GB110).

scientific article

Novel Helix-Constrained Nociceptin Derivatives Are Potent Agonists and Antagonists of ERK Phosphorylation and Thermal Analgesia in Mice ⬇️

scientific article published on November 10, 2010

PAR2 Modulators Derived from GB88.

scientific article

Pathway-selective antagonism of proteinase activated receptor 2.

scientific article

Pharmacological inhibition of protease-activated receptor-2 reduces crescent formation in rat nephrotoxic serum nephritis

scientific article published on 25 March 2019

Protease-activated receptor 2 does not contribute to renal inflammation or fibrosis in the obstructed kidney

scientific article published on 31 July 2019

Protease-activated receptor-2 regulates trypsin expression in the brain and protects against seizures and epileptogenesis.

scientific article published on 5 January 2008

Rational design and synthesis of an orally bioavailable peptide guided by NMR amide temperature coefficients

scientific article

Receptor residence time trumps drug-likeness and oral bioavailability in determining efficacy of complement C5a antagonists.

scientific article

Structure-Activity Relationships of Wollamide Cyclic Hexapeptides with Activity against Drug-Resistant and Intracellular

scientific article published on 26 February 2019

Total Synthesis, Structure, and Oral Absorption of a Thiazole Cyclic Peptide, Sanguinamide A

scientific article published on 06 November 2012

Paulina is supported by:

About Paulina

Help