List of works by Nicolas Lebegue

A Phosphosite Mutant Approach on LRRK2 Links Phosphorylation and Dephosphorylation to Protective and Deleterious Markers, Respectively

scientific article published on 17 March 2022

Anti-diabetic activity of fused PPARγ-SIRT1 ligands with limited body-weight gain by mimicking calorie restriction and decreasing SGK1 expression

scientific article published on 10 June 2017

Antimicrobial Properties of Compounds Isolated from <i>Syzygium malaccense</i> (L.) Merr. and L.M. Perry and Medicinal Plants Used in French Polynesia

scientific article published on 14 May 2022

Antioxidant activity of benzoxazolinonic and benzothiazolinonic derivatives in the LDL oxidation model.

scientific article published on 15 September 2009

Antioxydant activity of β-carboline derivatives in the LDL oxidation model

scientific article published on 30 March 2011

Docking study of ligands into the colchicine binding site of tubulin.

scientific article published on December 2004

EGF-Containing Membrane-Bound Mucins: A Hidden ErbB2 Targeting Pathway?

scientific article published on 13 February 2020

Effect of 6-Benzoyl-benzothiazol-2-one scaffold on the pharmacological profile of α-alkoxyphenylpropionic acid derived PPAR agonists

scientific article published on 01 December 2020

Effect of oxime ether incorporation in acyl indole derivatives on PPAR subtype selectivity

scientific article

In vitro pharmacokinetic profile of a benzopyridooxathiazepine derivative using rat microsomes and hepatocytes: identification of phases I and II metabolites.

scientific article published on 7 March 2013

Lipid-lowering properties of 6-benzoyl-2(3H)-benzothiazolone and structurally related compounds

scientific article published in December 2005

MUC4-ErbB2 Oncogenic Complex: Binding studies using Microscale Thermophoresis

scientific article published on 13 November 2019

Novel 1,3-dicarbonyl compounds having 2(3H)-benzazolonic heterocycles as PPARgamma agonists

scientific article published on 02 August 2006

Novel benzopyridothiadiazepines as potential active antitumor agents

scientific article published on November 2005

Pharmacokinetic evaluation of a novel benzopyridooxathiazepine derivative as a potential anticancer agent

scientific article published on 22 October 2014

Publisher Correction: MUC4-ErbB2 Oncogenic Complex: Binding studies using Microscale Thermophoresis

scientific article published on 14 April 2020

S26948, a new specific peroxisome proliferator activated receptor gamma modulator improved in vivo hepatic insulin sensitivity in 48 h lipid infused rats.

scientific article published on 26 February 2009

Scavenging of reactive oxygen species by letosteine, a molecule with two blocked-SH groups. Comparison with free-SH drugs

scientific article published on 01 May 1995

Stereoselective synthesis of enantiopure N-protected-3-arylpiperazines from keto-esters

Structural elucidation of degradation products of a benzopyridooxathiazepine under stress conditions using electrospray orbitrap mass spectrometry - study of degradation kinetic.

scientific article

Synthesis and Biological Evaluation of N-[2-(4-Hydroxyphenylamino)-pyridin-3-yl]-4-methoxy-benzenesulfonamide (ABT-751) Tricyclic Analogues as Antimitotic and Antivascular Agents with Potent in Vivo Antitumor Activity.

scientific article published on 18 August 2016

Synthesis of a novel series of (Z)-3,5-disubstituted thiazolidine-2,4-diones as promising anti-breast cancer agents

scientific article published on 15 January 2020

Synthesis of triazoloquinazolinone based compounds as tubulin polymerization inhibitors and vascular disrupting agents.

scientific article published on 22 March 2016

Synthesis, biological evaluation and docking studies of 4-amino-tetrahydroquinazolino[3,2-e]purine derivatives.

scientific article published on 17 September 2010

Targeting peroxisome proliferator-activated receptors (PPARs): development of modulators.

scientific article published on 27 February 2012