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List of works by Nicolas Pietrancosta

1,1'-Xylyl bis-1,4,8,11-tetraaza cyclotetradecane: a new potential copper chelator agent for neuroprotection in Alzheimer's disease. Its comparative effects with clioquinol on rat brain copper distribution.

scientific article published on 11 April 2006

5'-Methylene-triazole-substituted-aminoribosyl uridines as MraY inhibitors: synthesis, biological evaluation and molecular modeling

scientific article

Antidepressant efficacy of a selective organic cation transporter blocker in a mouse model of depression

scientific article published on 16 October 2019

Bacterial Transferase MraY, a Source of Inspiration towards New Antibiotics

scientific article published on 01 January 2018

CXCR4, master regulator of innate immune responses?

scientific article published in August 2017

CYP2U1 activity is altered by missense mutations in hereditary spastic paraplegia 56.

scientific article published on 16 October 2017

Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition

scientific article published on 06 November 2019

Characterization of a Human Point Mutation of VGLUT3 (p.A211V) in the Rodent Brain Suggests a Nonuniform Distribution of the Transporter in Synaptic Vesicles

scientific article

Clinical or ATPase domain mutations in ABCD4 disrupt the interaction between the vitamin B12-trafficking proteins ABCD4 and LMBD1.

scientific article

Ctr9, a Protein in the Transcription Complex Paf1, Regulates Dopamine Transporter Activity at the Plasma Membrane.

scientific article published on 5 June 2015

Design, synthesis and biological evaluation of small-azo-dyes as potent Vesicular Glutamate Transporters inhibitors

scientific article published on 18 March 2014

Destabilization of the human RED-SMU1 splicing complex as a basis for host-directed antiinfluenza strategy

scientific article published on 10 May 2019

Enhanced delivery of gamma-secretase inhibitor DAPT into the brain via an ascorbic acid mediated strategy.

scientific article published on 31 May 2005

Expression in yeast, new substrates, and construction of a first 3D model of human orphan cytochrome P450 2U1: Interpretation of substrate hydroxylation regioselectivity from docking studies.

scientific article published on 7 April 2015

Identification of Primary Natural Killer Cell Modulators by Chemical Library Screening with a Luciferase-Based Functional Assay

scientific article published on 05 September 2018

LSP5-2157 a new inhibitor of vesicular glutamate transporters

scientific article published on 04 December 2019

Membrane-bound human orphan cytochrome P450 2U1: Sequence singularities, construction of a full 3D model, and substrate docking

scientific article published on 22 July 2017

Naphthyl and coumarinyl biarylpiperazine derivatives as highly potent human beta-secretase inhibitors. Design, synthesis, and enzymatic BACE-1 and cell assays.

scientific article published on July 2006

Natural amines inhibit activation of human plasmacytoid dendritic cells through CXCR4 engagement

scientific article published on 09 February 2017

Pseudomonas aeruginosa Lipoxygenase LoxA Contributes to Lung Infection by Altering the Host Immune Lipid Signaling

scientific article published on 14 August 2019

Purification and characterization of recombinant human liver glycolate oxidase.

scientific article

Regulation of IRE1 RNase activity by the Ribonuclease inhibitor 1 (RNH1)

scientific article published on 05 September 2018

Reverse Immunology Approach to Define a New HIV-gp41-Neutralizing Epitope

article

Rose Bengal analogs and vesicular glutamate transporters (VGLUTs).

scientific article published on 25 June 2010

Simple Coupling Reaction between Amino Acids and Weakly Nucleophilic Heteroaromatic Amines

scientific article published on 01 September 2004

Spectral and 3D model studies of the interaction of orphan human cytochrome P450 2U1 with substrates and ligands.

scientific article published on 22 July 2016

Stimulating Type I interferon response with small molecules: revival of an old idea

scientific article published on 29 October 2015

Structural and Functional Characterization of the Interaction of Snapin with the Dopamine Transporter: Differential Modulation of Psychostimulant Actions.

scientific article

Structure of human glycolate oxidase in complex with the inhibitor 4-carboxy-5-[(4-chlorophenyl)sulfanyl]-1,2,3-thiadiazole

scientific article

Substituted thiazolamide coupled to a redox delivery system: a new gamma-secretase inhibitor with enhanced pharmacokinetic profile.

scientific article published on 10 January 2005

Successful prediction of substrate-binding pocket in SLC17 transporter sialin.

scientific article published on 13 February 2012

Synthesis and anti-HIV properties of new hydroxyquinoline–polyamine conjugates on cells infected by HIV-1 LAV and HIV-1 BaL viral strains

article

Synthesis and biological activity of N-substituted spiro[benzoxazepine-piperidine] Aβ-peptide production inhibitors

article

Synthesis of Quinoline Dicarboxylic Esters as Biocompatible Fluorescent Tags

scientific article published on September 12, 2012

[Organic cation transporters as novel therapeutic targets for depression]

scientific article published on 21 August 2020