List of works by Gilles Ouvry

Design of selective PI3Kα inhibitors starting from a promiscuous pan kinase scaffold

scientific article published on 29 April 2015

Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis.

scientific article published on 12 January 2018

Discovery of 1-(4-(5-(5-amino-6-(5-tert-butyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one (AZD8835): A potent and selective inhibitor of PI3Kα and PI3Kδ for the treatment of cancers

scientific article published on 9 October 2015

Discovery of Novel 3-Quinoline Carboxamides as Potent, Selective, and Orally Bioavailable Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase

scientific article

Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors

scientific article published on 10 May 2017

Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists

scientific article published on 12 October 2016

Identification of novel TACE inhibitors compatible with topical application.

scientific article

Optimization of a Series of Bivalent Triazolopyridazine Based Bromodomain and Extraterminal Inhibitors: The Discovery of (3R)-4-[2-[4-[1-(3-Methoxy-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-4-piperidyl]phenoxy]ethyl]-1,3-dimethyl-piperazin-2-one (AZD515

scientific article

Substituted allyl diphenylphosphine oxides as radical allylating agents

scientific article published on 01 July 2006

Synthesis and biological activity of anticoccidial agents: 2,3-diarylindoles.

scientific article published on 9 January 2009

Synthesis and biological activity of imidazopyridine anticoccidial agents: Part II.

scientific article published on 26 September 2007

The Identification of Potent, Selective, and Orally Available Inhibitors of Ataxia Telangiectasia Mutated (ATM) Kinase: The Discovery of AZD0156 (8-{6-[3-(Dimethylamino)propoxy]pyridin-3-yl}-3-methyl-1-(tetrahydro-2 H-pyran-4-yl)-1,3-dihydro-2 H-imi

scientific article published on 23 April 2018

beta-Nitro xanthates as olefin precursors

scientific article published on 01 August 2003

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