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List of works by Jonathan S Rosenblum

Boro-norleucine as a P1 residue for the design of selective and potent DPP7 inhibitors.

scientific article published in October 2005

DPP8 and DPP9 expression in cynomolgus monkey and Sprague Dawley rat tissues.

scientific article published on 12 July 2013

Efficient Nuclear Transport of Structurally Disturbed Cargo: Mutations in a Cargo Protein Switch Its Cognate Karyopherin ⬇️

scientific article published on February 9, 2011

Functional interrogation of kinases and other nucleotide-binding proteins.

scientific article published on 15 May 2013

Inhibitor focusing: direct selection of drug targets from proteomes using activity-based probes.

scientific article published on February 2003

Polo-like kinases inhibited by wortmannin. Labeling site and downstream effects.

scientific article published on 29 November 2006

Prolyl peptidases: a serine protease subfamily with high potential for drug discovery.

scientific article

Synergistic computational and experimental proteomics approaches for more accurate detection of active serine hydrolases in yeast

scientific article

Synthesis and activity of a potent, specific azabicyclo[3.3.0]-octane-based DPP II inhibitor.

scientific article published on 10 October 2006

Synthesis and structure-activity relationship of (1-halo-2-naphthyl) carbamate-based inhibitors of KIAA1363 (NCEH1/AADACL1).

scientific article

Synthesis and structure-activity relationship of N-alkyl Gly-boro-Pro inhibitors of DPP4, FAP, and DPP7.

scientific article published in October 2005

Synthesis and structure–activity relationship of 4-quinolone-3-carboxylic acid based inhibitors of glycogen synthase kinase-3β ⬇️

scientific article published on August 5, 2011

Wortmannin, a widely used phosphoinositide 3-kinase inhibitor, also potently inhibits mammalian polo-like kinase.

scientific article published in January 2005

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