List of works - Agostino Cilibrizzi

2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists.

scientific article published on 8 April 2016

3D-QSAR assisted identification of FABP4 inhibitors: An effective scaffold hopping analysis/QSAR evaluation

scientific article published on 29 November 2018

A case of extensive protein platination: the reaction of lysozyme with a Pt(ii)–terpyridine complex

scientific article published on 01 July 2018

A tri-functional vanadium(iv) complex to detect cysteine oxidation

scientific article

Cinnoline derivatives as human neutrophil elastase inhibitors

scientific article published on 21 July 2015

Correspondence: Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury

scientific article published on 7 February 2018

Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase.

scientific article published on 7 July 2011

Development of small molecule non-peptide formyl peptide receptor (FPR) ligands and molecular modeling of their recognition.

scientific article

Dihedral Angle Calculations To Elucidate the Folding of Peptides through Its Main Mechanical Forces

scientific article published on 15 February 2019

Diversity-oriented synthesis of macrocyclic peptidomimetics

scientific article

FABP4 inhibitors 3D-QSAR model and isosteric replacement of BMS309403 datasets

scientific article published on 19 December 2018

Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity.

scientific article published on 31 March 2010

Further studies on arylpiperazinyl alkyl pyridazinones: discovery of an exceptionally potent, orally active, antinociceptive agent in thermally induced pain.

scientific article published on December 2009

Further studies on pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as potent and selective human A1 adenosine receptor antagonists

scientific article published on 12 October 2014

Hydroxypyridinone Journey into Metal Chelation

scientific article published on 23 July 2018

Novel Phosphate Derivatives as Scaffolds for the Preparation of Synthetic Phosphoserine-Based Peptides Using the Fmoc/t-Bu Solid-Phase Strategy

article

Pharmacokinetics of Mephedrone Enantiomers in Whole Blood after a Controlled Intranasal Administration to Healthy Human Volunteers

scientific article published on 23 December 2020

Pyrazolo[1′,5′:1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A1 adenosine receptor ligands ⬇️

scientific article published on September 22, 2010

Repurposing strategies on pyridazinone-based series by pharmacophore- and structure-driven screening

scientific article published on 01 December 2020

Solid-Phase Synthesis and In-Silico Analysis of Iron-Binding Catecholato Chelators

scientific article published on 12 October 2020

Synthesis and Evaluation as Antitubercular Agents of 5-Arylethenyl and 5-(Hetero)aryl-3-Isoxazolecarboxylate

Synthesis and iron coordination properties of schizokinen and its imide derivative

scientific article published on 01 November 2019

Synthesis of five and six-membered heterocycles bearing an arylpiperazinylalkyl side chain as orally active antinociceptive agents

scientific article published on 02 September 2015

Synthesis, HPLC enantioresolution, and X-ray analysis of a new series of C5-methyl pyridazines as N-formyl peptide receptor (FPR) agonists.

scientific article

Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonists

scientific article published on 27 April 2012

Synthetic Approaches for Piperidone-Based Templates as Scaffolds to Access Chirally Enriched Donepezil Analogues

scientific article published on 03 February 2020

The role of mitochondrial labile iron in Friedreich's ataxia skin fibroblasts sensitivity to ultraviolet A

scientific article published on 01 March 2019

Vanadyl complexes with dansyl-labelled di-picolinic acid ligands: synthesis, phosphatase inhibition activity and cellular uptake studies

scientific article published on 23 March 2016

List of works by Agostino Cilibrizzi

2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists.

3D-QSAR assisted identification of FABP4 inhibitors: An effective scaffold hopping analysis/QSAR evaluation

A case of extensive protein platination: the reaction of lysozyme with a Pt(ii)–terpyridine complex

A tri-functional vanadium(iv) complex to detect cysteine oxidation

Cinnoline derivatives as human neutrophil elastase inhibitors

Correspondence: Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury

Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase.

Development of small molecule non-peptide formyl peptide receptor (FPR) ligands and molecular modeling of their recognition.

Dihedral Angle Calculations To Elucidate the Folding of Peptides through Its Main Mechanical Forces

Diversity-oriented synthesis of macrocyclic peptidomimetics

FABP4 inhibitors 3D-QSAR model and isosteric replacement of BMS309403 datasets

Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity.

Further studies on arylpiperazinyl alkyl pyridazinones: discovery of an exceptionally potent, orally active, antinociceptive agent in thermally induced pain.

Further studies on pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as potent and selective human A1 adenosine receptor antagonists

Hydroxypyridinone Journey into Metal Chelation

Novel Phosphate Derivatives as Scaffolds for the Preparation of Synthetic Phosphoserine-Based Peptides Using the Fmoc/t-Bu Solid-Phase Strategy

Pharmacokinetics of Mephedrone Enantiomers in Whole Blood after a Controlled Intranasal Administration to Healthy Human Volunteers

Pyrazolo[1′,5′:1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as selective human A1 adenosine receptor ligands ⬇️

Repurposing strategies on pyridazinone-based series by pharmacophore- and structure-driven screening

Solid-Phase Synthesis and In-Silico Analysis of Iron-Binding Catecholato Chelators

Synthesis and Evaluation as Antitubercular Agents of 5-Arylethenyl and 5-(Hetero)aryl-3-Isoxazolecarboxylate

Synthesis and iron coordination properties of schizokinen and its imide derivative

Synthesis of five and six-membered heterocycles bearing an arylpiperazinylalkyl side chain as orally active antinociceptive agents

Synthesis, HPLC enantioresolution, and X-ray analysis of a new series of C5-methyl pyridazines as N-formyl peptide receptor (FPR) agonists.

Synthesis, enantioresolution, and activity profile of chiral 6-methyl-2,4-disubstituted pyridazin-3(2H)-ones as potent N-formyl peptide receptor agonists

Synthetic Approaches for Piperidone-Based Templates as Scaffolds to Access Chirally Enriched Donepezil Analogues

The role of mitochondrial labile iron in Friedreich's ataxia skin fibroblasts sensitivity to ultraviolet A

Vanadyl complexes with dansyl-labelled di-picolinic acid ligands: synthesis, phosphatase inhibition activity and cellular uptake studies