List of works - Somsak Ruchirawat

8-Hydroxyquinolines: a review of their metal chelating properties and medicinal applications

scientific article

A flavonoid chrysin suppresses hypoxic survival and metastatic growth of mouse breast cancer cells.

scientific article published on 20 August 2013

A new sulfoxide analog of 1,2,3,6-tetrahydrophenylpyridine and antimicrobial activity

scientific article published on 27 September 2010

A novel tricyclic polyketide and its biosynthetic precursor azaphilone derivatives from the endophytic fungus Dothideomycete sp.

scientific article

Alkaloids as important scaffolds in therapeutic drugs for the treatments of cancer, tuberculosis, and smoking cessation

scientific article

Antimalarial and antimicrobial activities of 8-Aminoquinoline-Uracils metal complexes

scientific article published on 18 February 2016

Antimicrobial and antioxidative activities of bioactive constituents from Hydnophytum formicarum Jack. ⬇️

scientific article

Antimycobacterial activity of natural products and synthetic agents: pyrrolodiquinolines and vermelhotin as anti-tubercular leads against clinical multidrug resistant isolates of Mycobacterium tuberculosis

scientific article

Antioxidant, cytotoxicity, and QSAR study of 1-adamantylthio derivatives of 3-picoline and phenylpyridines

Antiplasmodial dimeric chalcone derivatives from the roots of Uvaria siamensis

scientific article published on 15 December 2016

Aromatase inhibitory activity of 1,4-naphthoquinone derivatives and QSAR study.

scientific article

Aspergillusol A, an alpha-glucosidase inhibitor from the marine-derived fungus Aspergillus aculeatus.

scientific article

Bioactive 4-hydroxycinnamide and bioactivities of Polyalthia cerasoides

scientific article published on 08 March 2011

Bioactive azafluorenone alkaloids from Polyalthia debilis (Pierre) Finet & Gagnep ⬇️

scientific article published on 3 November 2009

Bioactive cardinane sesquiterpenes from the stems of Alangium salviifolium

scientific article

Bioactive metabolites from Spilanthes acmella Murr. ⬇️

scientific article

Coriander (Coriandrum sativum): A promising functional food toward the well-being

scientific article published on 21 November 2017

Cytotoxic Steroidal Glycosides from the Whole Plant of Calamus acanthophyllus

scientific article

Cytotoxic sesquiterpenes from the endophytic fungus Pseudolagarobasidium acaciicola.

scientific article published on 14 December 2015

Cytotoxicity and QSAR study of (thio)ureas derived from phenylalkylamines and pyridylalkylamines

Depsidones, aromatase inhibitors and radical scavenging agents from the marine-derived fungus Aspergillus unguis CRI282-03.

scientific article published on 3 February 2012

Derivatives (halogen, nitro and amino) of 8-hydroxyquinoline with highly potent antimicrobial and antioxidant activities

scientific article published on 24 March 2016

Design, synthesis and molecular docking studies of novel N-benzenesulfonyl-1,2,3,4-tetrahydroisoquinoline-based triazoles with potential anticancer activity

scientific article published on 6 May 2014

Designing new analogs for streamlining the structure of cytotoxic lamellarin natural products.

scientific article published on 20 February 2015

Discovery of novel 1,2,3-triazole derivatives as anticancer agents using QSAR and in silico structural modification

scientific article

Drimane Sesquiterpene-Conjugated Amino Acids from a Marine Isolate of the Fungus Talaromyces minioluteus (Penicillium Minioluteum) ⬇️

scientific article published on 5 June 2015

Elucidating the structure-activity relationships of the vasorelaxation and antioxidation properties of thionicotinic acid derivatives.

scientific article published on 6 January 2010

Facile and Divergent Synthesis of Lamellarins and Lactam-Containing Derivatives with Improved Drug Likeness and Biological Activities.

scientific article published on 16 July 2015

High therapeutic potential of Spilanthes acmella: A review

scientific article published on 4 April 2013

Homodimers of Vanillin and Apocynin Decrease the Metastatic Potential of Human Cancer Cells by Inhibiting the FAK/PI3K/Akt Signaling Pathway

scientific article published on March 2017

Hybrid flavan-chalcones, aromatase and lipoxygenase inhibitors, from Desmos cochinchinensis

scientific article

Investigation of aromatase inhibitory activity of metal complexes of 8-hydroxyquinoline and uracil derivatives

scientific article

Investigation on biological activities of anthranilic acid sulfonamide analogs

scientific article published on 07 October 2011

New bioactive triterpenoids and antimalarial activity of Diospyros rubra Lec.

scientific article published on 15 January 2010

Novel 1,4-naphthoquinone-based sulfonamides: Synthesis, QSAR, anticancer and antimalarial studies

scientific article published on 5 September 2015

Novel triazole-tetrahydroisoquinoline hybrids as human aromatase inhibitors

scientific article published on 28 September 2019

Overcoming multidrug resistance in human lung cancer with novel benzo[a]quinolizin-4-ones.

scientific article published on March 2011

Oxyresveratrol: Structural Modification and Evaluation of Biological Activities.

scientific article

Part 1: Antiplasmodial, cytotoxic, radical scavenging and antioxidant activities of Thai plants in the family Acanthaceae.

scientific article published on 16 June 2010

Radical scavenging and antioxidant activities of isocoumarins and a phthalide from the endophytic fungus Colletotrichum sp.

scientific article published on 21 December 2010

Roles of Pyridine and Pyrimidine Derivatives as Privileged Scaffolds in Anticancer Agents

scientific article published on 23 September 2016

Sterols from Thai Marine Sponge Petrosia (Strongylophora) sp. and Their Cytotoxicity

scientific article published on 23 February 2017

Synthesis and biological activities of azalamellarins

scientific article published on September 2010

Synthesis and cytotoxicity of novel 2,2'-bis- and 2,2',2″-tris-indolylmethanes-based bengacarboline analogs

scientific article

Synthesis and molecular docking of 1,2,3-triazole-based sulfonamides as aromatase inhibitors

scientific article published on 17 April 2015

Synthesis and molecular docking of N,N'-disubstituted thiourea derivatives as novel aromatase inhibitors

scientific article published on 04 May 2018

Synthesis and structure-activity relationship of 2-thiopyrimidine-4-one analogs as antimicrobial and anticancer agents

scientific article published on 16 December 2010

Synthesis and structure-activity relationship of mono-indole-, bis-indole-, and tris-indole-based sulfonamides as potential anticancer agents

scientific article published on 28 June 2013

Synthesis of N-substituted 5-iodouracils as antimicrobial and anticancer agents.

scientific article

Synthesis of isocryptolepine analogues and their structure-activity relationship studies as antiplasmodial and antiproliferative agents.

scientific article

Synthesis, anticancer activity and QSAR study of 1,4-naphthoquinone derivatives

scientific article

Synthesis, biological evaluation and molecular docking of novel chalcone-coumarin hybrids as anticancer and antimalarial agents

scientific article

Synthesis, cytotoxic and antimalarial activities of benzoyl thiosemicarbazone analogs of isoquinoline and related compounds.

scientific article published on 23 February 2010

Synthesis, cytotoxicity and QSAR study of N-tosyl-1,2,3,4-tetrahydroisoquinoline derivatives

scientific article published on 21 April 2013

Synthesis, molecular docking, and QSAR study of bis-sulfonamide derivatives as potential aromatase inhibitors

scientific article published on 03 August 2019

Synthesis, molecular docking, and QSAR study of sulfonamide-based indoles as aromatase inhibitors

scientific article published on 20 October 2017

Terpenoids from the roots of Drypetes hoaensis and their cytotoxic activities

scientific article published on 25 January 2014

The application of the Baker–Venkataraman rearrangement to the synthesis of benz[b]indeno[2,1-e]pyran-10,11-dione

scientific article (publication date: June 2002)

Vanillin enhances TRAIL-induced apoptosis in cancer cells through inhibition of NF-kappaB activation

scientific article published on July 1, 2010

Vasorelaxant and antioxidant activities of Spilanthes acmella Murr.

scientific article published on 18 December 2008

List of works by Somsak Ruchirawat

8-Hydroxyquinolines: a review of their metal chelating properties and medicinal applications

A flavonoid chrysin suppresses hypoxic survival and metastatic growth of mouse breast cancer cells.

A new sulfoxide analog of 1,2,3,6-tetrahydrophenylpyridine and antimicrobial activity

A novel tricyclic polyketide and its biosynthetic precursor azaphilone derivatives from the endophytic fungus Dothideomycete sp.

Alkaloids as important scaffolds in therapeutic drugs for the treatments of cancer, tuberculosis, and smoking cessation

Antimalarial and antimicrobial activities of 8-Aminoquinoline-Uracils metal complexes

Antimicrobial and antioxidative activities of bioactive constituents from Hydnophytum formicarum Jack. ⬇️

Antimycobacterial activity of natural products and synthetic agents: pyrrolodiquinolines and vermelhotin as anti-tubercular leads against clinical multidrug resistant isolates of Mycobacterium tuberculosis

Antioxidant, cytotoxicity, and QSAR study of 1-adamantylthio derivatives of 3-picoline and phenylpyridines

Antiplasmodial dimeric chalcone derivatives from the roots of Uvaria siamensis

Aromatase inhibitory activity of 1,4-naphthoquinone derivatives and QSAR study.

Aspergillusol A, an alpha-glucosidase inhibitor from the marine-derived fungus Aspergillus aculeatus.

Bioactive 4-hydroxycinnamide and bioactivities of Polyalthia cerasoides

Bioactive azafluorenone alkaloids from Polyalthia debilis (Pierre) Finet & Gagnep ⬇️

Bioactive cardinane sesquiterpenes from the stems of Alangium salviifolium

Bioactive metabolites from Spilanthes acmella Murr. ⬇️

Coriander (Coriandrum sativum): A promising functional food toward the well-being

Cytotoxic Steroidal Glycosides from the Whole Plant of Calamus acanthophyllus

Cytotoxic sesquiterpenes from the endophytic fungus Pseudolagarobasidium acaciicola.

Cytotoxicity and QSAR study of (thio)ureas derived from phenylalkylamines and pyridylalkylamines

Depsidones, aromatase inhibitors and radical scavenging agents from the marine-derived fungus Aspergillus unguis CRI282-03.

Derivatives (halogen, nitro and amino) of 8-hydroxyquinoline with highly potent antimicrobial and antioxidant activities

Design, synthesis and molecular docking studies of novel N-benzenesulfonyl-1,2,3,4-tetrahydroisoquinoline-based triazoles with potential anticancer activity

Designing new analogs for streamlining the structure of cytotoxic lamellarin natural products.

Discovery of novel 1,2,3-triazole derivatives as anticancer agents using QSAR and in silico structural modification

Drimane Sesquiterpene-Conjugated Amino Acids from a Marine Isolate of the Fungus Talaromyces minioluteus (Penicillium Minioluteum) ⬇️

Elucidating the structure-activity relationships of the vasorelaxation and antioxidation properties of thionicotinic acid derivatives.

Facile and Divergent Synthesis of Lamellarins and Lactam-Containing Derivatives with Improved Drug Likeness and Biological Activities.

High therapeutic potential of Spilanthes acmella: A review

Homodimers of Vanillin and Apocynin Decrease the Metastatic Potential of Human Cancer Cells by Inhibiting the FAK/PI3K/Akt Signaling Pathway

Hybrid flavan-chalcones, aromatase and lipoxygenase inhibitors, from Desmos cochinchinensis

Investigation of aromatase inhibitory activity of metal complexes of 8-hydroxyquinoline and uracil derivatives

Investigation on biological activities of anthranilic acid sulfonamide analogs

New bioactive triterpenoids and antimalarial activity of Diospyros rubra Lec.

Novel 1,4-naphthoquinone-based sulfonamides: Synthesis, QSAR, anticancer and antimalarial studies

Novel triazole-tetrahydroisoquinoline hybrids as human aromatase inhibitors

Overcoming multidrug resistance in human lung cancer with novel benzo[a]quinolizin-4-ones.

Oxyresveratrol: Structural Modification and Evaluation of Biological Activities.

Part 1: Antiplasmodial, cytotoxic, radical scavenging and antioxidant activities of Thai plants in the family Acanthaceae.

Radical scavenging and antioxidant activities of isocoumarins and a phthalide from the endophytic fungus Colletotrichum sp.

Roles of Pyridine and Pyrimidine Derivatives as Privileged Scaffolds in Anticancer Agents

Sterols from Thai Marine Sponge Petrosia (Strongylophora) sp. and Their Cytotoxicity

Synthesis and biological activities of azalamellarins

Synthesis and cytotoxicity of novel 2,2'-bis- and 2,2',2″-tris-indolylmethanes-based bengacarboline analogs

Synthesis and molecular docking of 1,2,3-triazole-based sulfonamides as aromatase inhibitors

Synthesis and molecular docking of N,N'-disubstituted thiourea derivatives as novel aromatase inhibitors

Synthesis and structure-activity relationship of 2-thiopyrimidine-4-one analogs as antimicrobial and anticancer agents

Synthesis and structure-activity relationship of mono-indole-, bis-indole-, and tris-indole-based sulfonamides as potential anticancer agents

Synthesis of N-substituted 5-iodouracils as antimicrobial and anticancer agents.

Synthesis of isocryptolepine analogues and their structure-activity relationship studies as antiplasmodial and antiproliferative agents.

Synthesis, anticancer activity and QSAR study of 1,4-naphthoquinone derivatives

Synthesis, biological evaluation and molecular docking of novel chalcone-coumarin hybrids as anticancer and antimalarial agents

Synthesis, cytotoxic and antimalarial activities of benzoyl thiosemicarbazone analogs of isoquinoline and related compounds.

Synthesis, cytotoxicity and QSAR study of N-tosyl-1,2,3,4-tetrahydroisoquinoline derivatives

Synthesis, molecular docking, and QSAR study of bis-sulfonamide derivatives as potential aromatase inhibitors

Synthesis, molecular docking, and QSAR study of sulfonamide-based indoles as aromatase inhibitors

Terpenoids from the roots of Drypetes hoaensis and their cytotoxic activities

The application of the Baker–Venkataraman rearrangement to the synthesis of benz[b]indeno[2,1-e]pyran-10,11-dione

Vanillin enhances TRAIL-induced apoptosis in cancer cells through inhibition of NF-kappaB activation

Vasorelaxant and antioxidant activities of Spilanthes acmella Murr.