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List of works by Sotirios Katsamakas

Boronic Acid Group: A Cumbersome False Negative Case in the Process of Drug Design.

scientific article published on 7 September 2016

Design and Synthesis of Novel Bis-Imidazolyl Phenyl Butadiyne Derivatives as HCV NS5A Inhibitors

scientific article published on 20 May 2022

Design and synthesis of gallocyanine inhibitors of DKK1/LRP6 interactions for treatment of Alzheimer's disease

scientific article published on 12 June 2018

Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site

scientific article published on 8 July 2015

Discovery of Benzothiazole Scaffold-Based DNA Gyrase B Inhibitors

scientific article

Discovery of novel phenoxazinone derivatives as DKK1/LRP6 interaction inhibitors: Synthesis, biological evaluation and structure-activity relationships.

scientific article published on 16 January 2016

Examining barbiturate scaffold for the synthesis of new agents with biological interest

scientific article published on 01 August 2019

Mononuclear copper(II) complexes with 2-thiophene carboxylate and N-N donors; DNA interaction, antioxidant/anti-inflammatory and antitumor activity

scientific article published on 26 September 2018

Novel c(RGDyK)-based conjugates of POPAM and 5-fluorouracil for integrin-targeted cancer therapy.

scientific article published on 7 November 2017

Probing the Inhibition of Microtubule Affinity Regulating Kinase 4 by N-Substituted Acridones

scientific article published in Scientific Reports

RGD-mediated delivery of small-molecule drugs.

scientific article published on 10 April 2017

Synthesis and biological evaluation of a Platinum(II)-c(RGDyK) conjugate for integrin-targeted photodynamic therapy

scientific article published on 28 September 2017

Synthesis and evaluation of gallocyanine dyes as potential agents for the treatment of Alzheimer's disease and related neurodegenerative tauopathies

scientific article published on 22 November 2015

Synthesis, structure elucidation and biological evaluation of triple bridged dinuclear copper(II) complexes as anticancer and antioxidant/anti-inflammatory agents

scientific article

Targeting on poly(ADP-ribose) polymerase activity with DNA-damaging hybrid lactam-steroid alkylators in wild-type and BRCA1-mutated ovarian cancer cells.

scientific article