List of works - Valentín Hornillos

A BODIPY-embedding miltefosine analog linked to cell-penetrating Tat(48-60) peptide favors intracellular delivery and visualization of the antiparasitic drug

scientific article published on 21 January 2014

An efficient, one-pot synthesis of various ceramide 1-phosphates from sphingosine 1-phosphate.

scientific article published on 9 November 2007

Asymmetric allylic alkylation of acyclic allylic ethers with organolithium reagents

scientific article published on 21 August 2012

Catalytic Asymmetric Synthesis of Phosphine Boronates

scientific article published on 7 May 2015

Catalytic Asymmetric Synthesis of Phosphine Boronates

Catalytic Direct Cross-Coupling of Organolithium Compounds with Aryl Chlorides

scientific article published on 19 September 2013

Catalytic asymmetric conjugate addition of Grignard reagents to chromones

article

Catalytic asymmetric synthesis of chromenes and tetrahydroquinolines via sequential allylic alkylation and intramolecular Heck coupling

scientific article published on 07 March 2012

ChemInform Abstract: Catalytic Asymmetric Conjugate Addition of Grignard Reagents to Chromones

article

ChemInform Abstract: Catalytic Asymmetric Synthesis of Phosphine Boronates

ChemInform Abstract: Catalytic Direct Cross-Coupling of Organolithium Compounds with Aryl Chlorides

ChemInform Abstract: Copper-Catalyzed α-Selective Allylic Alkylation of Heteroaryllithium Reagents

ChemInform Abstract: Direct Catalytic Cross-Coupling of Alkenyllithium Compounds

ChemInform Abstract: Hindered Aryllithium Reagents as Partners in Palladium-Catalyzed Cross-Coupling: Synthesis of Tri- and Tetra-ortho-Substituted Biaryls under Ambient Conditions

ChemInform Abstract: Palladium-Catalyzed Direct Cross-Coupling of Organolithium Reagents with Aryl and Vinyl Triflates

ChemInform Abstract: Palladium-Catalyzed Direct Cross-Coupling of Secondary Alkyllithium Reagents

ChemInform Abstract: Palladium-Catalyzed, tert-Butyllithium-Mediated Dimerization of Aryl Halides and Its Application in the Atropselective Total Synthesis of Mastigophorene A

ChemInform Abstract: Pd-Catalyzed Cross-Coupling of Aryllithium Reagents with 2-Alkoxy-Substituted Aryl Chlorides: Mild and Efficient Synthesis of 3,3′-Diaryl BINOLs

ChemInform Abstract: tBuLi-Mediated One-Pot Direct Highly Selective Cross-Coupling of Two Distinct Aryl Bromides

Chiral Diarylmethanes via Copper-Catalyzed Asymmetric Allylic Arylation with Organolithium Compounds

scientific article published on 23 December 2015

Copper-catalysed α-selective allylic alkylation of heteroaryllithium reagents

scientific article published on 21 October 2014

Copper-catalyzed enantioselective allyl-allyl cross-coupling

scientific article published in February 2013

Cu-catalyzed asymmetric allylic alkylation of phosphonates and phosphine oxides with Grignard reagents

scientific article published on 27 February 2013

Cu-catalyzed enantioselective allylic alkylation with organolithium reagents

scientific article published on 2 February 2017

Defeating Leishmania resistance to Miltefosine (hexadecylphosphocholine) by peptide-mediated drug smuggling: A proof of mechanism for trypanosomatid chemotherapy

Direct catalytic cross-coupling of alkenyllithium compounds.

scientific article published on 28 November 2014

Dynamic Kinetic Asymmetric Heck Reaction for the Simultaneous Generation of Central and Axial Chirality

scientific article published on 27 August 2018

Dynamic Kinetic Resolution of Heterobiaryl Ketones via Zn-catalyzed Asymmetric Hydrosilylation.

scientific article published on 13 February 2018

Fast, greener and scalable direct coupling of organolithium compounds with no additional solvents

scientific article

Fluorescent labeling of Acanthamoeba assessed in situ from corneal sectioned microscopy.

scientific article

Frontispiece: Palladium-Catalysed Direct Cross-Coupling of Organolithium Reagents with Aryl and Vinyl Triflates

Hindered Aryllithium Reagents as Partners in Palladium-Catalyzed Cross-Coupling: Synthesis of Tri- and Tetra-ortho-Substituted Biaryls under Ambient Conditions

Hindered aryllithium reagents as partners in palladium-catalyzed cross-coupling: synthesis of tri- and tetra-ortho-substituted biaryls under ambient conditions.

scientific article

Innentitelbild: Catalytic Asymmetric Synthesis of Phosphine Boronates (Angew. Chem. 27/2015)

Inside Cover: Catalytic Asymmetric Synthesis of Phosphine Boronates (Angew. Chem. Int. Ed. 27/2015)

Ir-Catalyzed Atroposelective Desymmetrization of Heterobiaryls: Hydroarylation of Vinyl Ethers and Bicycloalkenes

scientific article published on 22 January 2020

Nickel-Catalyzed Cross-Coupling of Organolithium Reagents with (Hetero)Aryl Electrophiles

scientific article published on 29 December 2015

One-pot sequential 1,2-addition, Pd-catalysed cross-coupling of organolithium reagents with Weinreb amides

article

Palladium-Catalysed Direct Cross-Coupling of Organolithium Reagents with Aryl and Vinyl Triflates

scientific article published on 11 September 2014

Palladium-Catalyzed C(sp(3))-C(sp(2)) Cross-Coupling of (Trimethylsilyl)methyllithium with (Hetero)Aryl Halides

scientific article published on 14 April 2015

Palladium-Catalyzed, tert- Butyllithium-Mediated Dimerization of Aryl Halides and Its Application in the Atropselective Total Synthesis of Mastigophorene A

scientific article published on 16 February 2016

Palladium-catalysed direct cross-coupling of secondary alkyllithium reagents

Pd-Catalyzed Cross-Coupling of Aryllithium Reagents with 2-Alkoxy-Substituted Aryl Chlorides: Mild and Efficient Synthesis of 3,3′-Diaryl BINOLs

scientific article published on 16 December 2014

Ros3 (Lem3p/CDC50) Gene Dosage Is Implicated in Miltefosine Susceptibility in <i>Leishmania (Viannia) braziliensis</i> Clinical Isolates and in <i>Leishmania (Leishmania) major</i>

scientific article published on 16 March 2021

Synthesis and biological evaluation of fluorescent leishmanicidal analogues of hexadecylphosphocholine (miltefosine) as probes of antiparasite mechanisms.

scientific article published on 31 October 2007

Synthesis and characterization of metallodendritic palladium-biscarbene complexes derived from 1,1'-methylenebis(1,2,4-triazole)

scientific article published on 07 March 2011

Synthesis of 16-mercaptohexadecylphosphocholine, a miltefosine analog with leishmanicidal activity

scientific article published in 2006

Synthesis of BODIPY-labeled alkylphosphocholines with leishmanicidal activity, as fluorescent analogues of miltefosine

scientific article

Synthesis of axially chiral heterobiaryl alkynes via dynamic kinetic asymmetric alkynylation.

scientific article published on 18 November 2016

tBuLi-Mediated One-Pot Direct Highly Selective Cross-Coupling of Two Distinct Aryl Bromides

scientific article published on 10 September 2015

List of works by Valentín Hornillos

A BODIPY-embedding miltefosine analog linked to cell-penetrating Tat(48-60) peptide favors intracellular delivery and visualization of the antiparasitic drug

An efficient, one-pot synthesis of various ceramide 1-phosphates from sphingosine 1-phosphate.

Asymmetric allylic alkylation of acyclic allylic ethers with organolithium reagents

Catalytic Asymmetric Synthesis of Phosphine Boronates

Catalytic Asymmetric Synthesis of Phosphine Boronates

Catalytic Direct Cross-Coupling of Organolithium Compounds with Aryl Chlorides

Catalytic asymmetric conjugate addition of Grignard reagents to chromones

Catalytic asymmetric synthesis of chromenes and tetrahydroquinolines via sequential allylic alkylation and intramolecular Heck coupling

ChemInform Abstract: Catalytic Asymmetric Conjugate Addition of Grignard Reagents to Chromones

ChemInform Abstract: Catalytic Asymmetric Synthesis of Phosphine Boronates

ChemInform Abstract: Catalytic Direct Cross-Coupling of Organolithium Compounds with Aryl Chlorides

ChemInform Abstract: Copper-Catalyzed α-Selective Allylic Alkylation of Heteroaryllithium Reagents

ChemInform Abstract: Direct Catalytic Cross-Coupling of Alkenyllithium Compounds

ChemInform Abstract: Hindered Aryllithium Reagents as Partners in Palladium-Catalyzed Cross-Coupling: Synthesis of Tri- and Tetra-ortho-Substituted Biaryls under Ambient Conditions

ChemInform Abstract: Palladium-Catalyzed Direct Cross-Coupling of Organolithium Reagents with Aryl and Vinyl Triflates

ChemInform Abstract: Palladium-Catalyzed Direct Cross-Coupling of Secondary Alkyllithium Reagents

ChemInform Abstract: Palladium-Catalyzed, tert-Butyllithium-Mediated Dimerization of Aryl Halides and Its Application in the Atropselective Total Synthesis of Mastigophorene A

ChemInform Abstract: Pd-Catalyzed Cross-Coupling of Aryllithium Reagents with 2-Alkoxy-Substituted Aryl Chlorides: Mild and Efficient Synthesis of 3,3′-Diaryl BINOLs

ChemInform Abstract: tBuLi-Mediated One-Pot Direct Highly Selective Cross-Coupling of Two Distinct Aryl Bromides

Chiral Diarylmethanes via Copper-Catalyzed Asymmetric Allylic Arylation with Organolithium Compounds

Copper-catalysed α-selective allylic alkylation of heteroaryllithium reagents

Copper-catalyzed enantioselective allyl-allyl cross-coupling

Cu-catalyzed asymmetric allylic alkylation of phosphonates and phosphine oxides with Grignard reagents

Cu-catalyzed enantioselective allylic alkylation with organolithium reagents

Defeating Leishmania resistance to Miltefosine (hexadecylphosphocholine) by peptide-mediated drug smuggling: A proof of mechanism for trypanosomatid chemotherapy

Direct catalytic cross-coupling of alkenyllithium compounds.

Dynamic Kinetic Asymmetric Heck Reaction for the Simultaneous Generation of Central and Axial Chirality

Dynamic Kinetic Resolution of Heterobiaryl Ketones via Zn-catalyzed Asymmetric Hydrosilylation.

Fast, greener and scalable direct coupling of organolithium compounds with no additional solvents

Fluorescent labeling of Acanthamoeba assessed in situ from corneal sectioned microscopy.

Frontispiece: Palladium-Catalysed Direct Cross-Coupling of Organolithium Reagents with Aryl and Vinyl Triflates

Hindered Aryllithium Reagents as Partners in Palladium-Catalyzed Cross-Coupling: Synthesis of Tri- and Tetra-ortho-Substituted Biaryls under Ambient Conditions

Hindered aryllithium reagents as partners in palladium-catalyzed cross-coupling: synthesis of tri- and tetra-ortho-substituted biaryls under ambient conditions.

Innentitelbild: Catalytic Asymmetric Synthesis of Phosphine Boronates (Angew. Chem. 27/2015)

Inside Cover: Catalytic Asymmetric Synthesis of Phosphine Boronates (Angew. Chem. Int. Ed. 27/2015)

Ir-Catalyzed Atroposelective Desymmetrization of Heterobiaryls: Hydroarylation of Vinyl Ethers and Bicycloalkenes

Nickel-Catalyzed Cross-Coupling of Organolithium Reagents with (Hetero)Aryl Electrophiles

One-pot sequential 1,2-addition, Pd-catalysed cross-coupling of organolithium reagents with Weinreb amides

Palladium-Catalysed Direct Cross-Coupling of Organolithium Reagents with Aryl and Vinyl Triflates

Palladium-Catalyzed C(sp(3))-C(sp(2)) Cross-Coupling of (Trimethylsilyl)methyllithium with (Hetero)Aryl Halides

Palladium-Catalyzed, tert- Butyllithium-Mediated Dimerization of Aryl Halides and Its Application in the Atropselective Total Synthesis of Mastigophorene A

Palladium-Catalyzed, tert- Butyllithium-Mediated Dimerization of Aryl Halides and Its Application in the Atropselective Total Synthesis of Mastigophorene A

Palladium-catalysed direct cross-coupling of secondary alkyllithium reagents

Pd-Catalyzed Cross-Coupling of Aryllithium Reagents with 2-Alkoxy-Substituted Aryl Chlorides: Mild and Efficient Synthesis of 3,3′-Diaryl BINOLs

Ros3 (Lem3p/CDC50) Gene Dosage Is Implicated in Miltefosine Susceptibility in <i>Leishmania (Viannia) braziliensis</i> Clinical Isolates and in <i>Leishmania (Leishmania) major</i>

Synthesis and biological evaluation of fluorescent leishmanicidal analogues of hexadecylphosphocholine (miltefosine) as probes of antiparasite mechanisms.

Synthesis and characterization of metallodendritic palladium-biscarbene complexes derived from 1,1'-methylenebis(1,2,4-triazole)

Synthesis of 16-mercaptohexadecylphosphocholine, a miltefosine analog with leishmanicidal activity

Synthesis of BODIPY-labeled alkylphosphocholines with leishmanicidal activity, as fluorescent analogues of miltefosine

Synthesis of axially chiral heterobiaryl alkynes via dynamic kinetic asymmetric alkynylation.

tBuLi-Mediated One-Pot Direct Highly Selective Cross-Coupling of Two Distinct Aryl Bromides