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List of works by Frederick Monsma

Binding kinetics and mechanism of action: toward the discovery and development of better and best in class drugs

scientific article published on September 16, 2010

Characterizing cannabinoid CB2 receptor ligands using DiscoveRx PathHunter beta-arrestin assay

scientific article

Cloning and characterization of murine neuromedin U receptors.

scientific article published on September 2002

Discovery of novel chemotypes to a G-protein-coupled receptor through ligand-steered homology modeling and structure-based virtual screening.

scientific article published on 17 January 2008

Identification and characterization of a novel RF-amide peptide ligand for orphan G-protein-coupled receptor SP9155

scientific article (publication date: 25 July 2003)

Molecular modeling and site-specific mutagenesis of the histamine-binding site of the histamine H4 receptor.

scientific article

Murgocil is a highly bioactive staphylococcal-specific inhibitor of the peptidoglycan glycosyltransferase enzyme MurG.

scientific article published on 5 September 2013

P2Y(13): identification and characterization of a novel Galphai-coupled ADP receptor from human and mouse

scientific article (publication date: May 2002)

P518/Qrfp sequence polymorphisms in SAMP6 osteopenic mouse.

scientific article published on 17 September 2007

Regulation of two rat mas-related genes in a model of neuropathic pain.

scientific article published on 24 October 2005

SCH 1473759, a novel Aurora inhibitor, demonstrates enhanced anti-tumor activity in combination with taxanes and KSP inhibitors

scientific article published on February 5, 2011

Screening for antibacterial inhibitors of the UDP-3-O-(R-3-hydroxymyristoyl)-N-acetylglucosamine deacetylase (LpxC) using a high-throughput mass spectrometry assay

scientific article

The importance of drug-target residence time.

scientific article published on July 2009