List of works - Masaki Ohtawa

Concise asymmetric synthesis of (-)-bilobalide

scientific article published on 16 October 2019

Design and Synthesis of A-Ring Simplified Pyripyropene A Analogues as Potent and Selective Synthetic SOAT2 Inhibitors.

scientific article published on 11 January 2018

Design, synthesis, and biological evaluation of air-stable nafuredin-γ analogs as complex I inhibitors

scientific article published on 22 January 2015

Development of a new air-stable structure-simplified nafuredin-γ analog as a potent and selective nematode complex I inhibitor.

scientific article

In vitro metabolism of pyripyropene A and ACAT inhibitory activity of its metabolites.

scientific article

New pyripyropene A derivatives, highly SOAT2-selective inhibitors, improve hypercholesterolemia and atherosclerosis in atherogenic mouse models

scientific article

Pharmacological characterization of the neurotrophic sesquiterpene jiadifenolide reveals a non-convulsant signature and potential for progression in neurodegenerative disease studies

scientific article published on 22 June 2018

Potentiation of bleomycin in Jurkat cells by fungal pycnidione.

scientific article published in January 2012

Scopranones with Two Atypical Scooplike Moieties Produced by Streptomyces sp. BYK-11038

scientific article published on 24 October 2017

Selectivity of pyripyropene derivatives in inhibition toward acyl-CoA:cholesterol acyltransferase 2 isozyme

scientific article published in August 2008

Simplifungin and Valsafungins, Antifungal Antibiotics of Fungal Origin.

scientific article

Stereoselective total synthesis of atpenins a4 and b, harzianopyridone, and NBRI23477 B

scientific article published on 01 January 2012

Synthesis and Structural Revision of Cyslabdan.

scientific article

Synthesis and biological activity of 5-(4-methoxyphenyl)-oxazole derivatives.

scientific article

Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 1

scientific article published on 09 January 2013

Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 2

scientific article published on 06 March 2013

Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 3

scientific article published on 08 May 2013

Synthesis of (-)-11-O-Debenzoyltashironin: Neurotrophic Sesquiterpenes Cause Hyperexcitation.

scientific article published on 23 June 2017

Total Synthesis and Absolute Configuration of Simpotentin, a Potentiator of Amphotericin B Activity

scientific article published on 27 June 2019

List of works by Masaki Ohtawa

Concise asymmetric synthesis of (-)-bilobalide

Design and Synthesis of A-Ring Simplified Pyripyropene A Analogues as Potent and Selective Synthetic SOAT2 Inhibitors.

Design, synthesis, and biological evaluation of air-stable nafuredin-γ analogs as complex I inhibitors

Development of a new air-stable structure-simplified nafuredin-γ analog as a potent and selective nematode complex I inhibitor.

In vitro metabolism of pyripyropene A and ACAT inhibitory activity of its metabolites.

New pyripyropene A derivatives, highly SOAT2-selective inhibitors, improve hypercholesterolemia and atherosclerosis in atherogenic mouse models

Pharmacological characterization of the neurotrophic sesquiterpene jiadifenolide reveals a non-convulsant signature and potential for progression in neurodegenerative disease studies

Potentiation of bleomycin in Jurkat cells by fungal pycnidione.

Scopranones with Two Atypical Scooplike Moieties Produced by Streptomyces sp. BYK-11038

Selectivity of pyripyropene derivatives in inhibition toward acyl-CoA:cholesterol acyltransferase 2 isozyme

Simplifungin and Valsafungins, Antifungal Antibiotics of Fungal Origin.

Stereoselective total synthesis of atpenins a4 and b, harzianopyridone, and NBRI23477 B

Synthesis and Structural Revision of Cyslabdan.

Synthesis and biological activity of 5-(4-methoxyphenyl)-oxazole derivatives.

Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 1

Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 2

Synthesis and structure-activity relationship of pyripyropene A derivatives as potent and selective acyl-CoA:cholesterol acyltransferase 2 (ACAT2) inhibitors: part 3

Synthesis of (-)-11-O-Debenzoyltashironin: Neurotrophic Sesquiterpenes Cause Hyperexcitation.

Total Synthesis and Absolute Configuration of Simpotentin, a Potentiator of Amphotericin B Activity