List of works - Emilia Caselli

(S)-(+)-N-acetylphenylglycineboronic acid: a chiral derivatizing agent for Ee determination of 1,2-diols

scientific article published on 01 December 2003

Alpha-aminoester-derived imidazoles by 1,5-electrocyclization of azavinyl azomethine ylides

scientific article published on 01 July 2009

Chemo-enzymatic synthesis of levodropropizine.

scientific article published in October 2003

Design, Synthesis, Crystal Structures, and Antimicrobial Activity of Sulfonamide Boronic Acids as β-Lactamase Inhibitors ⬇️

scientific article published on November 11, 2010

Exploring sequence requirements for C3/C4 carboxylate recognition in the Pseudomonas aeruginosa cephalosporinase: Insights into plasticity of the AmpC β‐lactamase ⬇️

scientific article published on May 3, 2011

Fragment-guided design of subnanomolar -lactamase inhibitors active in vivo

scientific article

Inhibiting the β-Lactamase of Mycobacterium tuberculosis (Mtb) with Novel Boronic Acid Transition-State Inhibitors (BATSIs)

scientific article (publication date: 12 June 2015)

Inhibition of Acinetobacter-Derived Cephalosporinase: Exploring the Carboxylate Recognition Site Using Novel β-Lactamase Inhibitors.

scientific article published on 16 November 2017

Inhibition of the class C beta-lactamase from Acinetobacter spp.: insights into effective inhibitor design

scientific article

Interactions of oximino-substituted boronic acids and β-lactams with the CMY-2-derived extended-spectrum cephalosporinases CMY-30 and CMY-42

scientific article published on 10 December 2012

Negative Epistasis and Evolvability in TEM-1 β-Lactamase--The Thin Line between an Enzyme's Conformational Freedom and Disorder

scientific article published on 22 May 2015

One-Pot Synthesis of Imidazole-4-Carboxylates by Microwave-Assisted 1,5-Electrocyclization of Azavinyl Azomethine Ylides

scientific article published on August 2010

Recognition and resistance in TEM beta-lactamase

scientific article

Structure-Based Analysis of Boronic Acids as Inhibitors of Acinetobacter-Derived Cephalosporinase-7, a Unique Class C β-Lactamase.

scientific article published on 16 November 2017

Structure-based design and in-parallel synthesis of inhibitors of AmpC beta-lactamase

scientific article

Structures of FOX-4 Cephamycinase in Complex with Transition-State Analog Inhibitors

scientific article published on 27 April 2020

Structures of ceftazidime and its transition-state analogue in complex with AmpC beta-lactamase: implications for resistance mutations and inhibitor design

scientific article

Synthesis of 1,2,3-triazol-1-yl-methaneboronic acids via click chemistry: an easy access to a new potential scaffold for protease inhibitors.

scientific article published in February 2015

List of works by Emilia Caselli

(S)-(+)-N-acetylphenylglycineboronic acid: a chiral derivatizing agent for Ee determination of 1,2-diols

Alpha-aminoester-derived imidazoles by 1,5-electrocyclization of azavinyl azomethine ylides

Chemo-enzymatic synthesis of levodropropizine.

Design, Synthesis, Crystal Structures, and Antimicrobial Activity of Sulfonamide Boronic Acids as β-Lactamase Inhibitors ⬇️

Exploring sequence requirements for C3/C4 carboxylate recognition in the Pseudomonas aeruginosa cephalosporinase: Insights into plasticity of the AmpC β‐lactamase ⬇️

Fragment-guided design of subnanomolar -lactamase inhibitors active in vivo

Inhibiting the β-Lactamase of Mycobacterium tuberculosis (Mtb) with Novel Boronic Acid Transition-State Inhibitors (BATSIs)

Inhibition of Acinetobacter-Derived Cephalosporinase: Exploring the Carboxylate Recognition Site Using Novel β-Lactamase Inhibitors.

Inhibition of the class C beta-lactamase from Acinetobacter spp.: insights into effective inhibitor design

Interactions of oximino-substituted boronic acids and β-lactams with the CMY-2-derived extended-spectrum cephalosporinases CMY-30 and CMY-42

Negative Epistasis and Evolvability in TEM-1 β-Lactamase--The Thin Line between an Enzyme's Conformational Freedom and Disorder

One-Pot Synthesis of Imidazole-4-Carboxylates by Microwave-Assisted 1,5-Electrocyclization of Azavinyl Azomethine Ylides

Recognition and resistance in TEM beta-lactamase

Structure-Based Analysis of Boronic Acids as Inhibitors of Acinetobacter-Derived Cephalosporinase-7, a Unique Class C β-Lactamase.

Structure-based design and in-parallel synthesis of inhibitors of AmpC beta-lactamase

Structures of FOX-4 Cephamycinase in Complex with Transition-State Analog Inhibitors

Structures of ceftazidime and its transition-state analogue in complex with AmpC beta-lactamase: implications for resistance mutations and inhibitor design

Synthesis of 1,2,3-triazol-1-yl-methaneboronic acids via click chemistry: an easy access to a new potential scaffold for protease inhibitors.