List of works - Florine Cavelier

(L)-(Trimethylsilyl)alanine synthesis exploiting hydroxypinanone-induced diastereoselective alkylation.

scientific article published on 26 April 2013

A flexible synthesis of C33-C39 polyketide region of apratoxin: Synthesis of natural and unnatural analogues

A side-reaction in the SPPS of Trp-containing peptides

scientific article published on 01 October 1999

Access to α,α-Disubstituted Disilylated Amino Acids and Their Use in Solid-Phase Peptide Synthesis

scientific article published on 08 September 2015

All-L-Leu-Pro-Leu-Pro: a challenging cyclization

scientific article published on 01 November 2000

Analysis of ochratoxin A in grapes, musts and wines by LC-MS/MS: first comparison of stable isotope dilution assay and diastereomeric dilution assay methods.

scientific article published on 11 February 2014

Biological activity of silylated amino acid containing substance P analogues.

scientific article published in March 2004

Conformational studies of proline-, thiaproline- and dimethylsilaproline-containing diketopiperazines

scholarly article by Florine Cavelier published in January 2006

Control by Metals of Staphylopine Dehydrogenase Activity during Metallophore Biosynthesis

scientific article published on 22 March 2019

Cyclization of peptides through a urea bond: application to the Arg-Gly-Asp tripeptide

scientific article

Direct Access to L-Azetidine-2-carboxylic Acid

ESI mass spectrometry of amino acid trimethylsilylethyl esters.

scientific article

Efficient Synthesis of Nicotianamine and Non-Natural Analogues

Expedient Synthesis of Fmoc-(S)-γ-Fluoroleucine and Late-Stage Fluorination of Peptides

First identification and quantification of S-3-(hexan-1-ol)-γ-glutamyl-cysteine in grape must as a potential thiol precursor, using UPLC-MS/MS analysis and stable isotope dilution assay.

scientific article published on 30 May 2017

First synthesis of a stable isotope of Ochratoxin A metabolite for a reliable detoxification monitoring

scientific article published on 24 July 2013

High yield synthesis of tentoxin, a cyclic tetrapeptide.

scientific article published in July 2002

Highly resolutive separations of hardly soluble synthetic polypeptides by capillary electrophoresis

scientific article published in January 2010

Hydrophobic α,α-Disubstituted Disilylated TESDpg Induces Incipient 310-Helix in Short Tripeptide Sequence.

scientific article

Influence of silaproline on peptide conformation and bioactivity

scientific article published in March 2002

Innovative analysis of 3-mercaptohexan-1-ol, 3-mercaptohexylacetate and their corresponding disulfides in wine by stable isotope dilution assay and nano-liquid chromatography tandem mass spectrometry.

scientific article published on 21 September 2016

N-Substituted Glycines with Functional Side-Chains for Peptoid Synthesis

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

scientific article published on 21 October 2019

Neurotensin modulates the electrical activity of frog pituitary melanotropes via activation of a G-protein-coupled receptor pharmacologically related to both the NTS1 and nts2 receptors of mammals.

scientific article

New general strategy of dimerization of bioactive molecules

Peptide Bond Formation Using Polymer-Bound BOP

article by Sorin V. Filip et al published May 2004 in European Journal of Organic Chemistry

Phospholyl(borane) Amino Acids and Peptides: Stereoselective Synthesis and Fluorescent Properties with Large Stokes Shift.

scientific article published on 20 December 2017

Prediction of pKa Using DFT: the Nicotianamine Polyacid Example

scientific article published on 19 October 2016

Replacement of a Proline with Silaproline Causes a 20-Fold Increase in the Cellular Uptake of a Pro-Rich Peptide

scientific article published in 2006

Resolution of protected silaproline for a gram scale preparation

scientific article published on 15 October 2011

Revisiting the evaluation strategy of varietal thiol biogenesis

scientific article published on 15 June 2018

Silaproline Helical Mimetics Selectively Form an All-transPPII Helix

Silicon-Containing Amino Acids: Synthetic Aspects, Conformational Studies, and Applications to Bioactive Peptides

scientific article published on 16 August 2016

Spinal NTS2 receptor activation reverses signs of neuropathic pain

scientific article published on 11 June 2013

Stereoselective Synthesis of β-(5-Arylthiazolyl) α-Amino Acids and Use in Neurotensin Analogues

Stereoselective synthesis of unsaturated α-amino acids

scientific article published on 26 February 2015

Straightforward Synthesis of Chiral Silylated Amino Acids through Hydrosilylation

Straightforward synthesis of deuterated precursors to demonstrate the biogenesis of aromatic thiols in wine.

scientific article

Study of a lipophilic captopril analogue binding to angiotensin I converting enzyme

scientific article published on 01 February 2010

Supported synthesis of oxoapratoxin A.

scientific article

Synthesis and Characterization in Vitro and in Vivo of (l)-(Trimethylsilyl)alanine Containing Neurotensin Analogues.

scientific article published on 8 September 2015

Synthesis and biological activity of nicotianamine and analogues.

scientific article published in January 2009

Synthesis and biological effects of c(Lys-Lys-Pro-Tyr-Ile-Leu-Lys-Lys-Pro-Tyr-Ile-Leu) (JMV2012), a new analogue of neurotensin that crosses the blood-brain barrier

scientific article

Synthesis of homopolypeptides with PPII structure

Synthesis of tritium labelled delta sleep-inducing peptide

scholarly article by Matthieu Giraud et al published 2001 in Journal of Labelled Compounds and Radiopharmaceuticals

Synthesis, structure, and properties of MeSer1-tentoxin, a new cyclic tetrapeptide which interacts specifically with chloroplast F1 H(+)-ATPase differentiation of inhibitory and stimulating effects

scientific article published on 01 October 1996

Tentoxin has at least two binding sites on CF1 and epsilon-depleted CF1 ATPases isolated from spinach chloroplast

scientific article published on 01 October 1996

The crystallographic structure of thermoNicotianamine synthase with a synthetic reaction intermediate highlights the sequential processing mechanism

scientific article

Toward high yield synthesis of peptide-oligonucleotide chimera through a disulfide bridge: a simplified method for oligonucleotide activation.

scientific article published in November 2005

Towards a selective Boc deprotection on acid cleavable Wang resin

Use of Molecular Modeling to Design Selective NTS2 Neurotensin Analogues.

scientific article published on 3 April 2017

Varietal thiols in wine: discovery, analysis and applications

scientific article published on 22 July 2011

alpha,alpha'-disubstituted amino acids with silylated side chains as lipophilic building blocks for the synthesis of peptaibol analogues

scientific article published in July 2008

List of works by Florine Cavelier

(L)-(Trimethylsilyl)alanine synthesis exploiting hydroxypinanone-induced diastereoselective alkylation.

A flexible synthesis of C33-C39 polyketide region of apratoxin: Synthesis of natural and unnatural analogues

A side-reaction in the SPPS of Trp-containing peptides

Access to α,α-Disubstituted Disilylated Amino Acids and Their Use in Solid-Phase Peptide Synthesis

All-L-Leu-Pro-Leu-Pro: a challenging cyclization

Analysis of ochratoxin A in grapes, musts and wines by LC-MS/MS: first comparison of stable isotope dilution assay and diastereomeric dilution assay methods.

Biological activity of silylated amino acid containing substance P analogues.

Conformational studies of proline-, thiaproline- and dimethylsilaproline-containing diketopiperazines

Control by Metals of Staphylopine Dehydrogenase Activity during Metallophore Biosynthesis

Cyclization of peptides through a urea bond: application to the Arg-Gly-Asp tripeptide

Direct Access to L-Azetidine-2-carboxylic Acid

ESI mass spectrometry of amino acid trimethylsilylethyl esters.

Efficient Synthesis of Nicotianamine and Non-Natural Analogues

Expedient Synthesis of Fmoc-(S)-γ-Fluoroleucine and Late-Stage Fluorination of Peptides

First identification and quantification of S-3-(hexan-1-ol)-γ-glutamyl-cysteine in grape must as a potential thiol precursor, using UPLC-MS/MS analysis and stable isotope dilution assay.

First synthesis of a stable isotope of Ochratoxin A metabolite for a reliable detoxification monitoring

High yield synthesis of tentoxin, a cyclic tetrapeptide.

Highly resolutive separations of hardly soluble synthetic polypeptides by capillary electrophoresis

Hydrophobic α,α-Disubstituted Disilylated TESDpg Induces Incipient 310-Helix in Short Tripeptide Sequence.

Influence of silaproline on peptide conformation and bioactivity

Innovative analysis of 3-mercaptohexan-1-ol, 3-mercaptohexylacetate and their corresponding disulfides in wine by stable isotope dilution assay and nano-liquid chromatography tandem mass spectrometry.

N-Substituted Glycines with Functional Side-Chains for Peptoid Synthesis

Neurotensin Analogues Containing Cyclic Surrogates of Tyrosine at Position 11 Improve NTS2 Selectivity Leading to Analgesia without Hypotension and Hypothermia

Neurotensin modulates the electrical activity of frog pituitary melanotropes via activation of a G-protein-coupled receptor pharmacologically related to both the NTS1 and nts2 receptors of mammals.

New general strategy of dimerization of bioactive molecules

Peptide Bond Formation Using Polymer-Bound BOP

Phospholyl(borane) Amino Acids and Peptides: Stereoselective Synthesis and Fluorescent Properties with Large Stokes Shift.

Prediction of pKa Using DFT: the Nicotianamine Polyacid Example

Replacement of a Proline with Silaproline Causes a 20-Fold Increase in the Cellular Uptake of a Pro-Rich Peptide

Resolution of protected silaproline for a gram scale preparation

Revisiting the evaluation strategy of varietal thiol biogenesis

Silaproline Helical Mimetics Selectively Form an All-transPPII Helix

Silicon-Containing Amino Acids: Synthetic Aspects, Conformational Studies, and Applications to Bioactive Peptides

Spinal NTS2 receptor activation reverses signs of neuropathic pain

Stereoselective Synthesis of β-(5-Arylthiazolyl) α-Amino Acids and Use in Neurotensin Analogues

Stereoselective synthesis of unsaturated α-amino acids

Straightforward Synthesis of Chiral Silylated Amino Acids through Hydrosilylation

Straightforward synthesis of deuterated precursors to demonstrate the biogenesis of aromatic thiols in wine.

Study of a lipophilic captopril analogue binding to angiotensin I converting enzyme

Supported synthesis of oxoapratoxin A.

Synthesis and Characterization in Vitro and in Vivo of (l)-(Trimethylsilyl)alanine Containing Neurotensin Analogues.

Synthesis and biological activity of nicotianamine and analogues.

Synthesis and biological effects of c(Lys-Lys-Pro-Tyr-Ile-Leu-Lys-Lys-Pro-Tyr-Ile-Leu) (JMV2012), a new analogue of neurotensin that crosses the blood-brain barrier

Synthesis of homopolypeptides with PPII structure

Synthesis of tritium labelled delta sleep-inducing peptide

Synthesis, structure, and properties of MeSer1-tentoxin, a new cyclic tetrapeptide which interacts specifically with chloroplast F1 H(+)-ATPase differentiation of inhibitory and stimulating effects

Tentoxin has at least two binding sites on CF1 and epsilon-depleted CF1 ATPases isolated from spinach chloroplast

The crystallographic structure of thermoNicotianamine synthase with a synthetic reaction intermediate highlights the sequential processing mechanism

Toward high yield synthesis of peptide-oligonucleotide chimera through a disulfide bridge: a simplified method for oligonucleotide activation.

Towards a selective Boc deprotection on acid cleavable Wang resin

Use of Molecular Modeling to Design Selective NTS2 Neurotensin Analogues.

Varietal thiols in wine: discovery, analysis and applications

alpha,alpha'-disubstituted amino acids with silylated side chains as lipophilic building blocks for the synthesis of peptaibol analogues