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List of works by Darius P Zlotos

11-Aminostrychnine and N-(Strychnine-11-yl)propionamide: Synthesis, Configuration, and Pharmacological Evaluation at Glycine Receptors

scientific article published on 06 August 2019

6H,13H-Pyrazino[1,2-a;4,5-a']diindole analogs: probing the pharmacophore for allosteric ligands of muscarinic M2 receptors

scientific article published on 4 January 2006

A New Synthetic Approach to Pentacyclic Ring, 6,7,14,15-Tetrahydro[1,5]diazocino[1,2-a:6,5-a’]-8-dihydrodiindole

Bisquaternary Ligands of the Common Allosteric Site of M2Acetylcholine Receptors: Search for the Minimum Essential Distances between the Pharmacophoric Elements

scientific article published on 01 March 1999

Bisquaternary caracurine V and iso-caracurine V salts as ligands for the muscle type of nicotinic acetylcholine receptors: SAR and QSAR studies.

scientific article published on December 2004

Bisquaternary caracurine V derivatives as allosteric modulators of ligand binding to M2 acetylcholine receptors

scientific article published on 01 November 2000

Crystal structure of 5,11-di-hydro-pyrido[2,3-b][1,4]benzodiazepin-6-one

scientific article published on 11 April 2015

Discovery of Nanomolar Dengue and West Nile Virus Protease Inhibitors Containing a 4-Benzyloxyphenylglycine Residue

scientific article published on 12 November 2015

Drug conjugates—an emerging approach to treat breast cancer.

scientific article

Erratum to: New spectrofluorimetric methods for determination of melatonin in the presence of N-{2-[1-({3-[2-(acetylamino)ethyl]-5-methoxy-1H-indol-2-yl}methyl)-5-methoxy-1H-indol-3-yl]-ethyl}acetamide: a contaminant in commercial melatonin preparat

scientific article published on 28 September 2016

MT1 and MT2 melatonin receptors: ligands, models, oligomers, and therapeutic potential.

scientific article

Muscarinic receptor agonists and antagonists

N-Acetyl-5-arylalkoxytryptamine analogs: probing the melatonin receptors for MT(1) -selectivity.

scientific article published on 2 September 2011

Oxime Ethers of (E)-11-Isonitrosostrychnine as Highly Potent Glycine Receptor Antagonists.

scientific article

PPAR Gamma Activators: Off-Target Against Glioma Cell Migration and Brain Invasion.

scientific article published on January 2008

Pharmacological characterisation of strychnine and brucine analogues at glycine and alpha7 nicotinic acetylcholine receptors.

scientific article published on 9 May 2006

Pharmacological characteristics and binding modes of caracurine V analogues and related compounds at the neuronal alpha7 nicotinic acetylcholine receptor.

scientific article published on 28 August 2007

Probing the pharmacophore for allosteric ligands of muscarinic M2 receptors: SAR and QSAR studies in a series of bisquaternary salts of caracurine V and related ring systems

scientific article

Recent advances in melatonin receptor ligands.

scientific article

Recent advances in neuromuscular blocking agents

scientific article published on 01 June 2005

Semisynthetic analogues of toxiferine I and their pharmacological properties at α7 nAChRs, muscle-type nAChRs, and the allosteric binding site of muscarinic M2 receptors

scientific article

Stereochemistry of caracurine V

scientific article published on 01 June 2000

Structure-activity relationships of strychnine analogs at glycine receptors

scientific article

Synthesis and pharmacological evaluation of 1,2,3,4-tetrahydropyrazino[1,2-a]indole and 2-[(phenylmethylamino)methyl]-1H-indole analogues as novel melatoninergic ligands.

scientific article published on 5 May 2009

Synthesis, NMR conformational analysis and pharmacological evaluation of 7,7a,13,14-tetrahydro-6H-cyclobuta[b]pyrimido[1,2-a:3,4-a']diindole analogues as melatonin receptor ligands.

scientific article published on 25 May 2007

Update on melatonin receptors: IUPHAR Review 20.

scientific article published on 17 June 2016

[Drugs in the pipeline]

scientific article published on 01 January 2007

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