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List of works by Fabian Hulpia

1-(1-Arylethylpiperidin-4-yl)thymine Analogs as Antimycobacterial TMPK Inhibitors

scientific article published on 17 June 2020

2-((3,5-Dinitrobenzyl)thio)quinazolinones: Potent Antimycobacterial Agents Activated by Deazaflavin (F<sub>420</sub>)-Dependent Nitroreductase (Ddn)

scientific article published on 21 December 2020

C6-O-alkylated 7-deazainosine nucleoside analogues: Discovery of potent and selective anti-sleeping sickness agents

scientific article published on 03 January 2020

Combining tubercidin and cordycepin scaffolds results in highly active candidates to treat late-stage sleeping sickness

scientific article published on 05 December 2019

Discovery of Novel 7-Aryl 7-Deazapurine 3′-Deoxy-ribofuranosyl Nucleosides with Potent Activity against Trypanosoma cruzi

Discovery of Pyrrolo[2,3-b]pyridine (1,7-Dideazapurine) Nucleoside Analogues as Anti-Trypanosoma cruzi Agents

scientific article published on 20 September 2019

Exploring the purine core of 3'-C-ethynyladenosine (EAdo) in search of novel nucleoside therapeutics

scientific article published on 03 March 2016

New fluoroethyl phenylalanine analogues as potential LAT1-targeting PET tracers for glioblastoma

scientific article published on 27 February 2019

Positively selected modifications in the pore of TbAQP2 allow pentamidine to enter Trypanosoma brucei

scientific article published on 07 August 2020

Report on a novel emerging class of highly potent benzimidazole NPS opioids: Chemical and in vitro functional characterization of isotonitazene

scientific article published on 08 January 2020

Revisiting tubercidin against kinetoplastid parasites: Aromatic substitutions at position 7 improve activity and reduce toxicity

article published in 2019

Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors

scientific article published on 6 March 2018

Synthesis of a 3'-C-ethynyl-β-d-ribofuranose purine nucleoside library: Discovery of C7-deazapurine analogs as potent antiproliferative nucleosides

Synthesis, in vitro and in vivo small-animal SPECT evaluation of novel technetium labeled bile acid analogues to study (altered) hepatic transporter function.

scientific article published on 12 July 2016

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