List of works - Ioannis Papanastasiou

4-(1-Adamantyl)phenylalkylamines with Potential Antiproliferative Activity

An Overview on Target-Based Drug Design against Kinetoplastid Protozoan Infections: Human African Trypanosomiasis, Chagas Disease and Leishmaniases

scientific article published in 2021

Design and synthesis of Trypanosoma brucei active 1-alkyloxy and 1-benzyloxyadamantano 2-guanylhydrazones.

scientific article published in July 2009

Design and synthesis of new adamantyl-substituted antileishmanial ether phospholipids.

scientific article published on 22 July 2010

Fluorine substituted methoxyphenylalkyl amides as potent melatonin receptor agonists.

scientific article published on 11 February 2019

Heterocyclic rimantadine analogues with antiviral activity

scientific article published on 24 January 2006

In vitro Controlled Release from Solid Pharmaceutical Formulations of two new Adamantane Aminoethers with Antitubercular Activity (I).

scientific article published on 30 May 2017

In vitro Controlled Release of two new Tuberculocidal Adamantane Aminoethers from Solid Pharmaceutical Formulations (II)

scientific article published on 19 July 2017

Insights in Organometallic Synthesis of Various Adamantane Derivatives with Sigma Receptor-Binding Affinity and Antiproliferative/Anticancer Activity

scientific article published on 01 January 2018

Multicomponent reaction of aldehydes, amines and oxalacetate analogues leading to biologically attractive pyrrole derivatives

scientific article published on 03 January 2020

New adamantane derivatives with sigma affinity and antiproliferative activity.

scientific article published on July 2012

New adamantane phenylalkylamines with σ-receptor binding affinity and anticancer activity, associated with putative antagonism of neuropathic pain.

scientific article

Novel 1',1'-chain substituted hexahydrocannabinols: 9β-hydroxy-3-(1-hexyl-cyclobut-1-yl)-hexahydrocannabinol (AM2389) a highly potent cannabinoid receptor 1 (CB1) agonist.

scientific article

Sigma Receptor (σR) Ligands with Antiproliferative and Anticancer Activity.

scientific article published on 25 August 2017

Synthesis and Evaluation of Nifurtimox-Adamantane Adducts with Trypanocidal Activity

scientific article published on 27 May 2019

Synthesis of Adamantane Aminoethers with Antitubercular Potential

scientific article published on 01 January 2017

Synthesis of diphenoxyadamantane alkylamines with pharmacological interest

scientific article published on 06 April 2019

Synthesis, σ1, σ2-receptors binding affinity and antiproliferative action of new C1-substituted adamantanes ⬇️

scientific article published on March 24, 2012

The novel GABA adamantane derivative (AdGABA): design, synthesis, and activity relationship with gabapentin.

scientific article

List of works by Ioannis Papanastasiou

4-(1-Adamantyl)phenylalkylamines with Potential Antiproliferative Activity

An Overview on Target-Based Drug Design against Kinetoplastid Protozoan Infections: Human African Trypanosomiasis, Chagas Disease and Leishmaniases

Design and synthesis of Trypanosoma brucei active 1-alkyloxy and 1-benzyloxyadamantano 2-guanylhydrazones.

Design and synthesis of new adamantyl-substituted antileishmanial ether phospholipids.

Fluorine substituted methoxyphenylalkyl amides as potent melatonin receptor agonists.

Heterocyclic rimantadine analogues with antiviral activity

In vitro Controlled Release from Solid Pharmaceutical Formulations of two new Adamantane Aminoethers with Antitubercular Activity (I).

In vitro Controlled Release of two new Tuberculocidal Adamantane Aminoethers from Solid Pharmaceutical Formulations (II)

Insights in Organometallic Synthesis of Various Adamantane Derivatives with Sigma Receptor-Binding Affinity and Antiproliferative/Anticancer Activity

Multicomponent reaction of aldehydes, amines and oxalacetate analogues leading to biologically attractive pyrrole derivatives

New adamantane derivatives with sigma affinity and antiproliferative activity.

New adamantane phenylalkylamines with σ-receptor binding affinity and anticancer activity, associated with putative antagonism of neuropathic pain.

Novel 1',1'-chain substituted hexahydrocannabinols: 9β-hydroxy-3-(1-hexyl-cyclobut-1-yl)-hexahydrocannabinol (AM2389) a highly potent cannabinoid receptor 1 (CB1) agonist.

Sigma Receptor (σR) Ligands with Antiproliferative and Anticancer Activity.

Synthesis and Evaluation of Nifurtimox-Adamantane Adducts with Trypanocidal Activity

Synthesis of Adamantane Aminoethers with Antitubercular Potential

Synthesis of diphenoxyadamantane alkylamines with pharmacological interest

Synthesis, σ1, σ2-receptors binding affinity and antiproliferative action of new C1-substituted adamantanes ⬇️

The novel GABA adamantane derivative (AdGABA): design, synthesis, and activity relationship with gabapentin.